BIOMARKERS

Molecular Biopsy of Human Tumors

- a resource for Precision Medicine *

276 related articles for article (PubMed ID: 33236468)

  • 1. Design and in Vitro Characterization of Tricyclic Benzodiazepine Derivatives as Potent and Selective Antileukemic Agents.
    Mieczkowski A; Frączyk T; Psurski M; Wińska P; Siedlecki P; Dziełak M; Trzybiński D; Wilczek M; Bagiński M; Bieszczad B; Woźniak K
    Chem Biodivers; 2021 Jan; 18(1):e2000733. PubMed ID: 33236468
    [TBL] [Abstract][Full Text] [Related]  

  • 2. Novel (S)-1,3,4,12a-tetrahydropyrazino[2,1-c][1,4]benzodiazepine-6,12(2H,11H)-dione derivatives: Selective inhibition of MV-4-11 biphenotypic B myelomonocytic leukemia cells' growth is accompanied by reactive oxygen species overproduction and apoptosis.
    Mieczkowski A; Psurski M; Bagiński M; Bieszczad B; Mroczkowska M; Wilczek M; Czajkowska J; Trzybiński D; Woźniak K; Wietrzyk J
    Bioorg Med Chem Lett; 2018 Feb; 28(4):618-625. PubMed ID: 29395971
    [TBL] [Abstract][Full Text] [Related]  

  • 3. Design, synthesis, and biologic evaluation of novel chrysin derivatives as cytotoxic agents and caspase-3/7 activators.
    Al-Oudat BA; Alqudah MA; Audat SA; Al-Balas QA; El-Elimat T; Hassan MA; Frhat IN; Azaizeh MM
    Drug Des Devel Ther; 2019; 13():423-433. PubMed ID: 30774307
    [TBL] [Abstract][Full Text] [Related]  

  • 4. Selective Cytotoxic Effects of 5-Trifluoromethoxy-1H-indole-2,3-dione 3-Thiosemicarbazone Derivatives on Lymphoid-originated Cells.
    Danışman-Kalındemirtaş F; Erdem-Kuruca S; Akgün-Dar K; Karakaş Z; Soylu Ö; Karali N
    Anticancer Agents Med Chem; 2022; 22(2):349-355. PubMed ID: 33653255
    [TBL] [Abstract][Full Text] [Related]  

  • 5. Novel benzotriazole N-acylarylhydrazone hybrids: Design, synthesis, anticancer activity, effects on cell cycle profile, caspase-3 mediated apoptosis and FAK inhibition.
    Kassab AE; Hassan RA
    Bioorg Chem; 2018 Oct; 80():531-544. PubMed ID: 30014921
    [TBL] [Abstract][Full Text] [Related]  

  • 6. Design, synthesis, and biological evaluation of novel benzodiazepine derivatives as anticancer agents through inhibition of tubulin polymerization in vitro and in vivo.
    Pang Y; Lin H; Ou C; Cao Y; An B; Yan J; Li X
    Eur J Med Chem; 2019 Nov; 182():111670. PubMed ID: 31499359
    [TBL] [Abstract][Full Text] [Related]  

  • 7. The Synthesis, Anticancer Activity, Structure-Activity Relationships and Molecular Modelling Studies of Novel Isoindole-1,3(2H)-dione Compounds Containing Different Functional Groups.
    Tan A; Kizilkaya S; Kelestemur U; Akdemir A; Kara Y
    Anticancer Agents Med Chem; 2020; 20(11):1368-1378. PubMed ID: 32275494
    [TBL] [Abstract][Full Text] [Related]  

  • 8. Evaluation of Cytotoxic Potentials of Some Isoindole-1, 3-Dione Derivatives on HeLa, C6 and A549 Cancer Cell Lines.
    Tan A; Yaglioglu AS; Kishali NH; Sahin E; Kara Y
    Med Chem; 2020; 16(1):69-77. PubMed ID: 30520382
    [TBL] [Abstract][Full Text] [Related]  

  • 9. Biological Activity, Apoptotic Induction and Cell Cycle Arrest of New Hydrazonoyl Halides Derivatives.
    Mohamed MF; Hassaneen HM; Elzayat EM; El-Hallouty SM; El-Manawaty M; Saleh FM; Mohamed Y; El-Zohiry D; Fahmy G; Abdelaal N; Hassanin N; Hossam N
    Anticancer Agents Med Chem; 2019; 19(9):1141-1149. PubMed ID: 30843494
    [TBL] [Abstract][Full Text] [Related]  

  • 10. Mild C(sp
    Romo-Pérez A; Miranda LD; Chávez-Blanco AD; Dueñas-González A; Camacho-Corona MDR; Acosta-Huerta A; García A
    Eur J Med Chem; 2017 Sep; 138():1-12. PubMed ID: 28641156
    [TBL] [Abstract][Full Text] [Related]  

  • 11. Inclusion of a 5-fluorouracil moiety in nitrogenous bases derivatives as human carbonic anhydrase IX and XII inhibitors produced a targeted action against MDA-MB-231 and T47D breast cancer cells.
    Petreni A; Bonardi A; Lomelino C; Osman SM; ALOthman ZA; Eldehna WM; El-Haggar R; McKenna R; Nocentini A; Supuran CT
    Eur J Med Chem; 2020 Mar; 190():112112. PubMed ID: 32044580
    [TBL] [Abstract][Full Text] [Related]  

  • 12. Discovery of novel 1,5-benzodiazepine-2,4-dione derivatives as potential anticancer agents.
    Chen Y; Le V; Xu X; Shao X; Liu J; Li Z
    Bioorg Med Chem Lett; 2014 Aug; 24(16):3948-51. PubMed ID: 25017036
    [TBL] [Abstract][Full Text] [Related]  

  • 13. Synthesis, in vitro cytotoxicity and apoptosis inducing study of 2-aryl-3-nitro-2H-chromene derivatives as potent anti-breast cancer agents.
    Rahmani-Nezhad S; Safavi M; Pordeli M; Ardestani SK; Khosravani L; Pourshojaei Y; Mahdavi M; Emami S; Foroumadi A; Shafiee A
    Eur J Med Chem; 2014 Oct; 86():562-9. PubMed ID: 25216378
    [TBL] [Abstract][Full Text] [Related]  

  • 14. Design, Synthesis, In Vitro Anti-cancer Activity, ADMET Profile and Molecular Docking of Novel Triazolo[3,4-a]phthalazine Derivatives Targeting VEGFR-2 Enzyme.
    El-Helby AA; Sakr H; Ayyad RRA; El-Adl K; Ali MM; Khedr F
    Anticancer Agents Med Chem; 2018; 18(8):1184-1196. PubMed ID: 29651967
    [TBL] [Abstract][Full Text] [Related]  

  • 15. Synthesis and Antitumor Activity of a Series of Novel 1-Oxa-4-azaspiro[4,5]deca-6,9-diene-3,8-dione Derivatives.
    Yang Z; Zhong Q; Zheng S; Wang G; He L
    Molecules; 2019 Mar; 24(5):. PubMed ID: 30866506
    [TBL] [Abstract][Full Text] [Related]  

  • 16. Novel selenadiazole derivatives as selective antitumor and radical scavenging agents.
    Ruberte AC; Plano D; Encío I; Aydillo C; Sharma AK; Sanmartín C
    Eur J Med Chem; 2018 Sep; 157():14-27. PubMed ID: 30071406
    [TBL] [Abstract][Full Text] [Related]  

  • 17. Design, synthesis, and molecular docking study of new monastrol analogues as kinesin spindle protein inhibitors.
    El-Hamamsy MH; Sharafeldin NA; El-Moselhy TF; Tawfik HO
    Arch Pharm (Weinheim); 2020 Aug; 353(8):e2000060. PubMed ID: 32452567
    [TBL] [Abstract][Full Text] [Related]  

  • 18. Design, synthesis and antitumor evaluation of novel 5-methylpyrazolo[1,5-a]pyrimidine derivatives as potential c-Met inhibitors.
    Luo G; Ma Y; Liang X; Xie G; Luo Y; Zha D; Wang S; Yu L; Zheng X; Wu W; Zhang C
    Bioorg Chem; 2020 Nov; 104():104356. PubMed ID: 33142417
    [TBL] [Abstract][Full Text] [Related]  

  • 19. Assessment of elementary derivatives of 1,5-benzodiazepine as anticancer agents with synergy potential.
    Gawandi SJ; Desai VG; Joshi S; Shingade S; Pissurlenkar RR
    Bioorg Chem; 2021 Dec; 117():105331. PubMed ID: 34689084
    [TBL] [Abstract][Full Text] [Related]  

  • 20. Design, Synthesis, and Preliminary Bioactivity Evaluation of 2,7-Substituted Carbazole Derivatives as Potent Autotaxin Inhibitors and Antitumor Agents†.
    Wang W; Zhao F; Zhao Y; Pan W; Cao P; Wu L; Wang Z; Zhao X; Zhao Y; Wang H
    Anticancer Agents Med Chem; 2019; 19(2):256-264. PubMed ID: 30173652
    [TBL] [Abstract][Full Text] [Related]  

    [Next]    [New Search]
    of 14.