BIOMARKERS

Molecular Biopsy of Human Tumors

- a resource for Precision Medicine *

135 related articles for article (PubMed ID: 10071856)

  • 1. Synthesis of 2-phenylbenzofuran derivatives as testosterone 5 alpha-reductase inhibitor.
    Ishibashi K; Nakajima K; Sugioka Y; Sugiyama M; Hamada T; Horikoshi H; Nishi T
    Chem Pharm Bull (Tokyo); 1999 Feb; 47(2):226-40. PubMed ID: 10071856
    [TBL] [Abstract][Full Text] [Related]  

  • 2. Synthesis and 5 alpha-reductase inhibitory activities of benzofuran derivatives with a carbamoyl group.
    Ishibashi K; Nakajima K; Sugioka Y; Sugiyama M; Hamada T; Horikoshi H; Nishi T
    Bioorg Med Chem Lett; 1998 Mar; 8(6):561-6. PubMed ID: 9871560
    [TBL] [Abstract][Full Text] [Related]  

  • 3. Synthesis and testosterone 5 alpha-reductase-inhibitory activity of 4-aza-5 alpha-androstane-17-carboxamide compound with an aromatic moiety in the C-17 carbamoyl group.
    Kurata H; Ishibashi K; Saito S; Hamada T; Horikoshi H; Furukawa Y; Kojima K
    Chem Pharm Bull (Tokyo); 1996 Jan; 44(1):115-21. PubMed ID: 8582030
    [TBL] [Abstract][Full Text] [Related]  

  • 4. Pyrrole butyric acid derivatives as inhibitors of steroid 5 alpha-reductase.
    Kato M; Komoda K; Namera A; Sakai Y; Okada S; Yamada A; Yokoyama K; Migita E; Minobe Y; Tani T
    Chem Pharm Bull (Tokyo); 1997 Nov; 45(11):1767-76. PubMed ID: 9396152
    [TBL] [Abstract][Full Text] [Related]  

  • 5. N-substituted 4-(4-carboxyphenoxy)benzamides. Synthesis and evaluation as inhibitors of steroid-5alpha-reductase type 1 and 2.
    Picard F; Hartmann RW
    J Enzyme Inhib Med Chem; 2002 Jun; 17(3):187-96. PubMed ID: 12443045
    [TBL] [Abstract][Full Text] [Related]  

  • 6. Effect of C-ring modifications in benzo[c]quinolizin-3-ones, new selective inhibitors of human 5 alpha-reductase 1.
    Guarna A; Occhiato EG; Machetti F; Trabocchi A; Scarpi D; Danza G; Mancina R; Comerci A; Serio M
    Bioorg Med Chem; 2001 Jun; 9(6):1385-93. PubMed ID: 11408159
    [TBL] [Abstract][Full Text] [Related]  

  • 7. Benzofuranyl 3,5-bis-polyamine derivatives as time-dependent inhibitors of trypanothione reductase.
    Hamilton CJ; Saravanamuthu A; Fairlamb AH; Eggleston IM
    Bioorg Med Chem; 2003 Aug; 11(17):3683-93. PubMed ID: 12901914
    [TBL] [Abstract][Full Text] [Related]  

  • 8. A novel class of inhibitors for human steroid 5 alpha-reductase: phenoxybenzoic acid derivatives. I.
    Igarashi S; Kimura T; Naito R; Hara H; Fujii M; Koutoku H; Oritani H; Mase T
    Chem Pharm Bull (Tokyo); 1999 Aug; 47(8):1073-80. PubMed ID: 10478462
    [TBL] [Abstract][Full Text] [Related]  

  • 9. Design and synthesis of 3-pyrrol-3-yl-3H-isobenzofuran-1-ones as inhibitors of human cytosolic phospholipase A2alpha.
    Hess M; Schulze Elfringhoff A; Lehr M
    J Enzyme Inhib Med Chem; 2008 Dec; 23(6):946-57. PubMed ID: 18608744
    [TBL] [Abstract][Full Text] [Related]  

  • 10. In vivo and in vitro effect of novel 4,16-pregnadiene-6,20-dione derivatives, as 5alpha-reductase inhibitors.
    Bratoeff E; Cabeza M; Pérez-Ornelas V; Recillas S; Heuze I
    J Steroid Biochem Mol Biol; 2008 Sep; 111(3-5):275-81. PubMed ID: 18644453
    [TBL] [Abstract][Full Text] [Related]  

  • 11. Benzo[c]quinolizin-3-ones: a novel class of potent and selective nonsteroidal inhibitors of human steroid 5alpha-reductase 1.
    Guarna A; Machetti F; Occhiato EG; Scarpi D; Comerci A; Danza G; Mancina R; Serio M; Hardy K
    J Med Chem; 2000 Oct; 43(20):3718-35. PubMed ID: 11020287
    [TBL] [Abstract][Full Text] [Related]  

  • 12. Type-1 steroid 5 alpha-reductase is functionally active in the hair follicle as evidenced by new selective inhibitors of either type-1 or type-2 human steroid 5 alpha-reductase.
    Gerst C; Dalko M; Pichaud P; Galey JB; Buan B; Bernard BA
    Exp Dermatol; 2002 Feb; 11(1):52-8. PubMed ID: 11962492
    [TBL] [Abstract][Full Text] [Related]  

  • 13. Synthesis of 8-chloro-benzo[c]quinolizin-3-ones as potent and selective inhibitors of human steroid 5alpha-reductase 1.
    Guarna A; Occhiato EG; Scarpi D; Zorn C; Danza G; Comerci A; Mancina R; Serio M
    Bioorg Med Chem Lett; 2000 Feb; 10(4):353-6. PubMed ID: 10714498
    [TBL] [Abstract][Full Text] [Related]  

  • 14. A novel class of inhibitors for human steroid 5alpha-reductase: synthesis and biological evaluation of indole derivatives. II.
    Igarashi S; Inami H; Hara H; Fujii M; Koutoku H; Oritani H; Mase T
    Chem Pharm Bull (Tokyo); 2000 Mar; 48(3):382-8. PubMed ID: 10726862
    [TBL] [Abstract][Full Text] [Related]  

  • 15. Synthesis and structure-activity relationships of novel benzofuran farnesyltransferase inhibitors.
    Asoh K; Kohchi M; Hyoudoh I; Ohtsuka T; Masubuchi M; Kawasaki K; Ebiike H; Shiratori Y; Fukami TA; Kondoh O; Tsukaguchi T; Ishii N; Aoki Y; Shimma N; Sakaitani M
    Bioorg Med Chem Lett; 2009 Mar; 19(6):1753-7. PubMed ID: 19217288
    [TBL] [Abstract][Full Text] [Related]  

  • 16. A practical synthesis of 3-substituted delta 3,5(6)-steroids as new potential 5 alpha-reductase inhibitor.
    Tian W; Zhu Z; Liao Q; Wu Y
    Bioorg Med Chem Lett; 1998 Aug; 8(15):1949-52. PubMed ID: 9873464
    [TBL] [Abstract][Full Text] [Related]  

  • 17. Synthetic models related to methoxalen and menthofuran-cytochrome P450 (CYP) 2A6 interactions. benzofuran and coumarin derivatives as potent and selective inhibitors of CYP2A6.
    Yamaguchi Y; Akimoto I; Motegi K; Yoshimura T; Wada K; Nishizono N; Oda K
    Chem Pharm Bull (Tokyo); 2013; 61(10):997-1001. PubMed ID: 23902929
    [TBL] [Abstract][Full Text] [Related]  

  • 18. Pharmacokinetic parameters and mechanisms of inhibition of rat type 1 and 2 steroid 5alpha-reductases: determinants for different in vivo activities of GI198745 and finasteride in the rat.
    Stuart JD; Lee FW; Simpson Noel D; Kadwell SH; Overton LK; Hoffman CR; Kost TA; Tippin TK; Yeager RL; Batchelor KW; Bramson HN
    Biochem Pharmacol; 2001 Oct; 62(7):933-42. PubMed ID: 11543729
    [TBL] [Abstract][Full Text] [Related]  

  • 19. MAO inhibitory activity of 2-arylbenzofurans versus 3-arylcoumarins: synthesis, in vitro study, and docking calculations.
    Ferino G; Cadoni E; Matos MJ; Quezada E; Uriarte E; Santana L; Vilar S; Tatonetti NP; Yáñez M; Viña D; Picciau C; Serra S; Delogu G
    ChemMedChem; 2013 Jun; 8(6):956-66. PubMed ID: 23589499
    [TBL] [Abstract][Full Text] [Related]  

  • 20. Synthesis and evaluation of 2'-substituted 4-(4'-carboxy- or 4'-carboxymethylbenzylidene)-N-acylpiperidines: highly potent and in vivo active steroid 5alpha-reductase type 2 inhibitors.
    Picard F; Barassin S; Mokhtarian A; Hartmann RW
    J Med Chem; 2002 Aug; 45(16):3406-17. PubMed ID: 12139451
    [TBL] [Abstract][Full Text] [Related]  

    [Next]    [New Search]
    of 7.