BIOMARKERS

Molecular Biopsy of Human Tumors

- a resource for Precision Medicine *

118 related articles for article (PubMed ID: 10212389)

  • 1. Dicarba-closo-dodecaboranes as a pharmacophore. Retinoidal antagonists and potential agonists.
    Iijima T; Endo Y; Tsuji M; Kawachi E; Kagechika H; Shudo K
    Chem Pharm Bull (Tokyo); 1999 Mar; 47(3):398-404. PubMed ID: 10212389
    [TBL] [Abstract][Full Text] [Related]  

  • 2. Dicarba-closo-dodecaboranes as a pharmacophore. Novel potent retinoidal agonists.
    Endo Y; Iijima T; Kagechika H; Ohta K; Kawachi E; Shudo K
    Chem Pharm Bull (Tokyo); 1999 Apr; 47(4):585-7. PubMed ID: 10319433
    [TBL] [Abstract][Full Text] [Related]  

  • 3. Structure-Activity study of retinoid agonists bearing substituted dicarba-closo-dodecaborane. Relation between retinoidal activity and conformation of two aromatic nuclei.
    Endo Y; Iijima T; Yaguchi K; Kawachi E; Inoue N; Kagechika H; Kubo A; Itai A
    Bioorg Med Chem Lett; 2001 May; 11(10):1307-11. PubMed ID: 11392543
    [TBL] [Abstract][Full Text] [Related]  

  • 4. Polyenylidene thiazolidinedione derivatives with retinoidal activities.
    Tashima T; Kagechika H; Tsuji M; Fukasawa H; Kawachi E; Hashimoto Y; Shudo K
    Chem Pharm Bull (Tokyo); 1997 Nov; 45(11):1805-13. PubMed ID: 9396157
    [TBL] [Abstract][Full Text] [Related]  

  • 5. Estrogenic antagonists bearing dicarba-closo-dodecaborane as a hydrophobic pharmacophore.
    Endo Y; Yoshimi T; Iijima T; Yamakoshi Y
    Bioorg Med Chem Lett; 1999 Dec; 9(24):3387-92. PubMed ID: 10617077
    [TBL] [Abstract][Full Text] [Related]  

  • 6. Novel retinoid X receptor (RXR) antagonists having a dicarba-closo-dodecaborane as a hydrophobic moiety.
    Ohta K; Iijima T; Kawachi E; Kagechika H; Endo Y
    Bioorg Med Chem Lett; 2004 Dec; 14(23):5913-8. PubMed ID: 15501068
    [TBL] [Abstract][Full Text] [Related]  

  • 7. New estrogenic antagonists bearing dicarba-closo-dodecaborane as a hydrophobic pharmacophore.
    Endo Y; Yoshimi T; Yamakoshi Y
    Chem Pharm Bull (Tokyo); 2000 Feb; 48(2):312-4. PubMed ID: 10705532
    [TBL] [Abstract][Full Text] [Related]  

  • 8. Polymethylcarborane as a novel bioactive moiety: derivatives with potent retinoid antagonistic activity.
    Endo Y; Yaguchi K; Kawachi E; Kagechika H
    Bioorg Med Chem Lett; 2000 Aug; 10(15):1733-6. PubMed ID: 10937735
    [TBL] [Abstract][Full Text] [Related]  

  • 9. Structure-activity study of estrogenic agonists bearing dicarba-closo-dodecaborane. Effect of geometry and separation distance of hydroxyl groups at the ends of molecules.
    Endo Y; Iijima T; Amakoshi Y; Kubo A; Itai A
    Bioorg Med Chem Lett; 1999 Dec; 9(23):3313-8. PubMed ID: 10612591
    [TBL] [Abstract][Full Text] [Related]  

  • 10. Design, synthesis and evaluation of retinoids with novel bulky hydrophobic partial structures.
    Amano Y; Noguchi M; Nakagomi M; Muratake H; Fukasawa H; Shudo K
    Bioorg Med Chem; 2013 Jul; 21(14):4342-50. PubMed ID: 23685180
    [TBL] [Abstract][Full Text] [Related]  

  • 11. Regulation of retinoidal actions by diazepinylbenzoic acids. Retinoid synergists which activate the RXR-RAR heterodimers.
    Umemiya H; Fukasawa H; Ebisawa M; Eyrolles L; Kawachi E; Eisenmann G; Gronemeyer H; Hashimoto Y; Shudo K; Kagechika H
    J Med Chem; 1997 Dec; 40(26):4222-34. PubMed ID: 9435893
    [TBL] [Abstract][Full Text] [Related]  

  • 12. Novel iodinated carboranes: synthesis of the 8-iodo-7,9-dicarba-nido-undecaborate anion and 2-iodo-1,7-dicarba-closo-dodecaborane.
    Safronov AV; Kabytaev KZ; Jalisatgi SS; Hawthorne MF
    Dalton Trans; 2014 Sep; 43(33):12467-9. PubMed ID: 24782077
    [TBL] [Abstract][Full Text] [Related]  

  • 13. Novel retinoidal tropolone derivatives. Bioisosteric relationship of tropolone ring with benzoic acid moiety in retinoid structure.
    Ebisawa M; Ohta K; Kawachi E; Fukasawa H; Hashimoto Y; Kagechika H
    Chem Pharm Bull (Tokyo); 2001 Apr; 49(4):501-3. PubMed ID: 11310685
    [TBL] [Abstract][Full Text] [Related]  

  • 14. Syntheses and structure-activity relationships of 5,6,7, 8-tetrahydro-5,5,8,8-tetramethyl-2-quinoxaline derivatives with retinoic acid receptor alpha agonistic activity.
    Kikuchi K; Hibi S; Yoshimura H; Tokuhara N; Tai K; Hida T; Yamauchi T; Nagai M
    J Med Chem; 2000 Feb; 43(3):409-19. PubMed ID: 10669568
    [TBL] [Abstract][Full Text] [Related]  

  • 15. Protein kinase C modulators bearing dicarba-CLOSO-dodecaborane as a hydrophobic pharmacophore.
    Endo Y; Yoshimi T; Kimura K; Itai A
    Bioorg Med Chem Lett; 1999 Sep; 9(17):2561-4. PubMed ID: 10498208
    [TBL] [Abstract][Full Text] [Related]  

  • 16. Potent estrogen agonists based on carborane as a hydrophobic skeletal structure. A new medicinal application of boron clusters.
    Endo Y; Iijima T; Yamakoshi Y; Fukasawa H; Miyaura C; Inada M; Kubo A; Itai A
    Chem Biol; 2001 Apr; 8(4):341-55. PubMed ID: 11325590
    [TBL] [Abstract][Full Text] [Related]  

  • 17. Synthesis and 11C-Radiolabelling of 2-Carboranyl Benzothiazoles.
    Gona KB; Thota JL; Baz Z; Gómez-Vallejo V; Llop J
    Molecules; 2015 Apr; 20(5):7495-508. PubMed ID: 25915463
    [TBL] [Abstract][Full Text] [Related]  

  • 18. Potent androgen antagonists based on carborane as a hydrophobic core structure.
    Fujii S; Goto T; Ohta K; Hashimoto Y; Suzuki T; Ohta S; Endo Y
    J Med Chem; 2005 Jul; 48(14):4654-62. PubMed ID: 16000001
    [TBL] [Abstract][Full Text] [Related]  

  • 19. Utility of boron clusters for drug design. Hansch-fujita hydrophobic parameters pi of dicarba-closo-dodecaboranyl groups.
    Yamamoto K; Endo Y
    Bioorg Med Chem Lett; 2001 Sep; 11(17):2389-92. PubMed ID: 11527738
    [TBL] [Abstract][Full Text] [Related]  

  • 20. Modulators of tumor necrosis factor alpha production bearing dicarba-closo-dodecaborane as a hydrophobic pharmacophore.
    Tsuji M; Koiso Y; Takahashi H; Hashimoto Y; Endo Y
    Biol Pharm Bull; 2000 Apr; 23(4):513-6. PubMed ID: 10784439
    [TBL] [Abstract][Full Text] [Related]  

    [Next]    [New Search]
    of 6.