These tools will no longer be maintained as of December 31, 2024. Archived website can be found here. PubMed4Hh GitHub repository can be found here. Contact NLM Customer Service if you have questions.


BIOMARKERS

Molecular Biopsy of Human Tumors

- a resource for Precision Medicine *

101 related articles for article (PubMed ID: 10571146)

  • 1. 3-Acyloxy-2-phenalkylpropyl amides and esters of homovanillic acid as novel vanilloid receptor agonists.
    Lee J; Park SU; Kim JY; Kim JK; Lee J; Oh U; Marquez VE; Beheshti M; Wang QJ; Modarres S; Blumberg PM
    Bioorg Med Chem Lett; 1999 Oct; 9(20):2909-14. PubMed ID: 10571146
    [TBL] [Abstract][Full Text] [Related]  

  • 2. Phenolic modification as an approach to improve the pharmacology of the 3-acyloxy-2-benzylpropyl homovanillic amides and thioureas, a promising class of vanilloid receptor agonists and analgesics.
    Lee J; Lee J; Kang MS; Kim KP; Chung SJ; Blumberg PM; Yi JB; Park YH
    Bioorg Med Chem; 2002 Apr; 10(4):1171-9. PubMed ID: 11836128
    [TBL] [Abstract][Full Text] [Related]  

  • 3. Synthesis and evaluation of phorboid 20-homovanillates: discovery of a class of ligands binding to the vanilloid (capsaicin) receptor with different degrees of cooperativity.
    Appendino G; Cravotto G; Palmisano G; Annunziata R; Szallasi A
    J Med Chem; 1996 Aug; 39(16):3123-31. PubMed ID: 8759633
    [TBL] [Abstract][Full Text] [Related]  

  • 4. N-(3-Acyloxy-2-benzylpropyl)-N'-(4-hydroxy-3-methoxybenzyl) thiourea derivatives as potent vanilloid receptor agonists and analgesics.
    Lee J; Lee J; Kim J; Kim SY; Chun MW; Cho H; Hwang SW; Oh U; Park YH; Marquez VE; Beheshti M; Szabo T; Blumberg PM
    Bioorg Med Chem; 2001 Jan; 9(1):19-32. PubMed ID: 11197340
    [TBL] [Abstract][Full Text] [Related]  

  • 5. Structure-activity relationships of simplified resiniferatoxin analogues with potent VR1 agonism elucidates an active conformation of RTX for VR1 binding.
    Lee J; Kim SY; Park S; Lim JO; Kim JM; Kang M; Lee J; Kang SU; Choi HK; Jin MK; Welter JD; Szabo T; Tran R; Pearce LV; Toth A; Blumberg PM
    Bioorg Med Chem; 2004 Mar; 12(5):1055-69. PubMed ID: 14980619
    [TBL] [Abstract][Full Text] [Related]  

  • 6. N-(3-acyloxy-2-benzylpropyl)-N'-dihydroxytetrahydrobenzazepine and tetrahydroisoquinoline thiourea analogues as vanilloid receptor ligands.
    Lee J; Lee J; Szabo T; Gonzalez AF; Welter JD; Blumberg PM
    Bioorg Med Chem; 2001 Jul; 9(7):1713-20. PubMed ID: 11425572
    [TBL] [Abstract][Full Text] [Related]  

  • 7. 7-Hydroxynaphthalen-1-yl-urea and -amide antagonists of human vanilloid receptor 1.
    McDonnell ME; Zhang SP; Nasser N; Dubin AE; Dax SL
    Bioorg Med Chem Lett; 2004 Jan; 14(2):531-4. PubMed ID: 14698197
    [TBL] [Abstract][Full Text] [Related]  

  • 8. 2-(Anilinomethyl)imidazolines as alpha(1)-adrenoceptor agonists: the identification of alpha(1A) subtype selective 2'-carboxylic acid esters and amides.
    Bishop MJ; Berman J; Bigham EC; Garrison DT; Gobel MJ; Hodson SJ; Irving PE; Liacos JA; Minick DJ; Navas F; Saussy DL; Speake JD
    Bioorg Med Chem Lett; 2001 Nov; 11(21):2871-4. PubMed ID: 11597419
    [TBL] [Abstract][Full Text] [Related]  

  • 9. N-Acylvanillamides: development of an expeditious synthesis and discovery of new acyl templates for powerful activation of the vanilloid receptor.
    Appendino G; Minassi A; Morello AS; De Petrocellis L; Di Marzo V
    J Med Chem; 2002 Aug; 45(17):3739-45. PubMed ID: 12166946
    [TBL] [Abstract][Full Text] [Related]  

  • 10. Respiratory actions of vanilloid receptor agonists in the nucleus of the solitary tract: comparison of resiniferatoxin with non-pungent agents and anandamide.
    Geraghty DP; Mazzone SB
    Br J Pharmacol; 2002 Nov; 137(6):919-27. PubMed ID: 12411424
    [TBL] [Abstract][Full Text] [Related]  

  • 11. Mechanisms underlying tissue selectivity of anandamide and other vanilloid receptor agonists.
    Andersson DA; Adner M; Högestätt ED; Zygmunt PM
    Mol Pharmacol; 2002 Sep; 62(3):705-13. PubMed ID: 12181448
    [TBL] [Abstract][Full Text] [Related]  

  • 12. Isosteric replacement of amide by ester function. Synthesis and benzodiazepine receptor affinity of indol-3-ylglyoxylyl ester derivatives.
    Da Settimo A; Primofiore G; Marini AM; Da Settimo F; Nuti V; Martini C; Trincavelli L; Lucacchini A
    Farmaco; 1997; 52(6-7):421-8. PubMed ID: 9372593
    [TBL] [Abstract][Full Text] [Related]  

  • 13. Pyrrolizidine esters and amides as 5-HT4 receptor agonists and antagonists.
    Becker DP; Flynn DL; Moormann AE; Nosal R; Villamil CI; Loeffler R; Gullikson GW; Moummi C; Yang DC
    J Med Chem; 2006 Feb; 49(3):1125-39. PubMed ID: 16451077
    [TBL] [Abstract][Full Text] [Related]  

  • 14. Indolyl esters and amides related to indomethacin are selective COX-2 inhibitors.
    Kalgutkar AS; Crews BC; Saleh S; Prudhomme D; Marnett LJ
    Bioorg Med Chem; 2005 Dec; 13(24):6810-22. PubMed ID: 16169736
    [TBL] [Abstract][Full Text] [Related]  

  • 15. N-isoquinolin-5-yl-N'-aralkyl-urea and -amide antagonists of human vanilloid receptor 1.
    Jetter MC; Youngman MA; McNally JJ; Zhang SP; Dubin AE; Nasser N; Dax SL
    Bioorg Med Chem Lett; 2004 Jun; 14(12):3053-6. PubMed ID: 15149643
    [TBL] [Abstract][Full Text] [Related]  

  • 16. Cannabinoid receptor binding and agonist activity of amides and esters of arachidonic acid.
    Pinto JC; Potié F; Rice KC; Boring D; Johnson MR; Evans DM; Wilken GH; Cantrell CH; Howlett AC
    Mol Pharmacol; 1994 Sep; 46(3):516-22. PubMed ID: 7935333
    [TBL] [Abstract][Full Text] [Related]  

  • 17. Mass spectrometric decompositions of copper complexes with esters and amides of nicotinic acid.
    Borowiak-Resterna A; Frański R; Klonowska K; Olszanowski A
    Rapid Commun Mass Spectrom; 2005; 19(2):283-6. PubMed ID: 15609363
    [TBL] [Abstract][Full Text] [Related]  

  • 18. Condensation reactions and formation of amides, esters, and nitriles under hydrothermal conditions.
    Rushdi AI; Simoneit BR
    Astrobiology; 2004; 4(2):211-24. PubMed ID: 15253839
    [TBL] [Abstract][Full Text] [Related]  

  • 19. Synthesis of novel naphthoquinone aliphatic amides and esters and their anticancer evaluation.
    Kongkathip B; Akkarasamiyo S; Hasitapan K; Sittikul P; Boonyalai N; Kongkathip N
    Eur J Med Chem; 2013 Feb; 60():271-84. PubMed ID: 23313636
    [TBL] [Abstract][Full Text] [Related]  

  • 20. Analysis of structure-activity relationships with the N-(3-acyloxy-2-benzylpropyl)-N'-[4-(methylsulfonylamino)benzyl]thiourea template for vanilloid receptor 1 antagonism.
    Lee J; Kim SY; Lee J; Kang M; Kil MJ; Choi HK; Jin MK; Wang Y; Toth A; Pearce LV; Lundberg DJ; Tran R; Blumberg PM
    Bioorg Med Chem; 2004 Jul; 12(13):3411-20. PubMed ID: 15186827
    [TBL] [Abstract][Full Text] [Related]  

    [Next]    [New Search]
    of 6.