BIOMARKERS

Molecular Biopsy of Human Tumors

- a resource for Precision Medicine *

135 related articles for article (PubMed ID: 10587102)

  • 1. Synthesis and evaluation of [123I]labelled analogues of the partial inverse agonist Ro 15-4513 for the study of diazepam-insensitive benzodiazepine receptors.
    Katsifis A; Mardon K; McPhee M; Mattner F; Dikic B; Ridley D
    Nucl Med Biol; 1999 Aug; 26(6):641-9. PubMed ID: 10587102
    [TBL] [Abstract][Full Text] [Related]  

  • 2. Labelling of diazepam-sensitive and -insensitive benzodiazepine receptors with [3H]tert-butyl-8-chloro-5,6-dihydro-5-methyl-6-oxo-4H-imidazo [1,5-a][1,4]benzodiazepine 3-carboxylate (ZG-63).
    Wong G; Gu ZQ; de Costa B; Skolnick P
    Eur J Pharmacol; 1993 Sep; 247(1):57-63. PubMed ID: 8258361
    [TBL] [Abstract][Full Text] [Related]  

  • 3. Characterization of novel ligands for wild-type and natural mutant diazepam-insensitive benzodiazepine receptors.
    Wong G; Uusi-Oukari M; Hansen HC; Suzdak PD; Korpi ER
    Eur J Pharmacol; 1995 Apr; 289(2):335-42. PubMed ID: 7621907
    [TBL] [Abstract][Full Text] [Related]  

  • 4. Diazepam sensitivity of the binding of an imidazobenzodiazepine, [3H]Ro 15-4513, in cerebellar membranes from two rat lines developed for high and low alcohol sensitivity.
    Uusi-Oukari M; Korpi ER
    J Neurochem; 1990 Jun; 54(6):1980-7. PubMed ID: 2159982
    [TBL] [Abstract][Full Text] [Related]  

  • 5. Synthesis and evaluation of imidazo[1,5-a][1,4]benzodiazepine esters with high affinities and selectivities at "diazepam-insensitive" benzodiazepine receptors.
    Gu ZQ; Wong G; Dominguez C; de Costa BR; Rice KC; Skolnick P
    J Med Chem; 1993 Apr; 36(8):1001-6. PubMed ID: 8386769
    [TBL] [Abstract][Full Text] [Related]  

  • 6. The benzodiazepine/alcohol antagonist Ro 15-4513: binding to a GABAA receptor subtype that is insensitive to diazepam.
    Turner DM; Sapp DW; Olsen RW
    J Pharmacol Exp Ther; 1991 Jun; 257(3):1236-42. PubMed ID: 1646328
    [TBL] [Abstract][Full Text] [Related]  

  • 7. Characterization of diazepam-insensitive [3H]Ro 15-4513 binding in rodent brain and cultured cerebellar neuronal cells.
    Ito Y; Abiko E; Mitani K; Fukuda H
    Neurochem Res; 1994 Mar; 19(3):289-95. PubMed ID: 8177368
    [TBL] [Abstract][Full Text] [Related]  

  • 8. Synthesis and structure-activity relationships of 3,5-disubstituted 4,5-dihydro-6H-imidazo[1,5-a][1,4]benzodiazepin-6-ones at diazepam-sensitive and diazepam-insensitive benzodiazepine receptors.
    Ananthan S; Clayton SD; Ealick SE; Wong G; Evoniuk GE; Skolnick P
    J Med Chem; 1993 Feb; 36(4):479-90. PubMed ID: 8386247
    [TBL] [Abstract][Full Text] [Related]  

  • 9. Localization and pharmacological characterization of pigeon diazepam-insensitive GABAA receptors.
    Acri JB; Wong G; Lyon T; Witkin JM; Basile AS
    Neuroscience; 1997 Mar; 77(2):371-8. PubMed ID: 9472397
    [TBL] [Abstract][Full Text] [Related]  

  • 10. High affinity ligands for 'diazepam-insensitive' benzodiazepine receptors.
    Wong G; Skolnick P
    Eur J Pharmacol; 1992 Jan; 225(1):63-8. PubMed ID: 1311690
    [TBL] [Abstract][Full Text] [Related]  

  • 11. Synthesis of novel imidazobenzodiazepines as probes of the pharmacophore for "diazepam-insensitive" GABAA receptors.
    Zhang P; Zhang W; Liu R; Harris B; Skolnick P; Cook JM
    J Med Chem; 1995 May; 38(10):1679-88. PubMed ID: 7752192
    [TBL] [Abstract][Full Text] [Related]  

  • 12. Characterization of two cerebellar binding sites of [3H]Ro 15-4513.
    Uusi-Oukari M
    J Neurochem; 1992 Aug; 59(2):568-74. PubMed ID: 1321231
    [TBL] [Abstract][Full Text] [Related]  

  • 13. Effect of diethyl pyrocarbonate modification of benzodiazepine receptors on [3H]Ro 15-4513 binding.
    Uusi-Oukari M
    J Neurochem; 1992 Aug; 59(2):560-7. PubMed ID: 1321230
    [TBL] [Abstract][Full Text] [Related]  

  • 14. Contribution of "diazepam-insensitive" GABAA receptors to the alcohol antagonist properties of Ro 15-4513 and related imidazobenzodiazepines.
    Harris BD; Moody EJ; Gu ZQ; Skolnick P
    Pharmacol Biochem Behav; 1995 Sep; 52(1):113-8. PubMed ID: 7501652
    [TBL] [Abstract][Full Text] [Related]  

  • 15. Ro 15-4513 binding to GABAA receptors: subunit composition determines ligand efficacy.
    Wong G; Skolnick P
    Pharmacol Biochem Behav; 1992 May; 42(1):107-10. PubMed ID: 1326771
    [TBL] [Abstract][Full Text] [Related]  

  • 16. Synthetic and computer-assisted analysis of the structural requirements for selective, high-affinity ligand binding to diazepam-insensitive benzodiazepine receptors.
    Wong G; Koehler KF; Skolnick P; Gu ZQ; Ananthan S; Schönholzer P; Hunkeler W; Zhang W; Cook JM
    J Med Chem; 1993 Jun; 36(13):1820-30. PubMed ID: 8390574
    [TBL] [Abstract][Full Text] [Related]  

  • 17. Ex vivo binding of t-[35S )butylbicyclophosphorothionate: a biochemical tool to study the pharmacology of ethanol at the gamma-aminobutyric acid-coupled chloride channel.
    Sanna E; Concas A; Serra M; Santoro G; Biggio G
    J Pharmacol Exp Ther; 1991 Mar; 256(3):922-8. PubMed ID: 1706433
    [TBL] [Abstract][Full Text] [Related]  

  • 18. Binding of 1,4-benzodiazepines to a novel [3H]Ro15-4513 binding site in the rat spinal cord.
    Maguire PA; Davies MF; Loew GH
    Eur J Pharmacol; 1995 Jul; 280(2):167-73. PubMed ID: 7589182
    [TBL] [Abstract][Full Text] [Related]  

  • 19. Postnatal development of diazepam-insensitive [3H]Ro 15-4513 binding sites.
    Korpi ER; Uusi-Oukari M; Kaivola J
    Neuroscience; 1993 Mar; 53(2):483-8. PubMed ID: 8388087
    [TBL] [Abstract][Full Text] [Related]  

  • 20. Chronic benzodiazepine antagonist treatment and its withdrawal upregulates components of GABA-benzodiazepine receptor ionophore complex in cerebral cortex of rat.
    Kulkarni SK; Ticku MK
    Brain Res; 1990 Jun; 519(1-2):6-11. PubMed ID: 2168788
    [TBL] [Abstract][Full Text] [Related]  

    [Next]    [New Search]
    of 7.