These tools will no longer be maintained as of December 31, 2024. Archived website can be found here. PubMed4Hh GitHub repository can be found here. Contact NLM Customer Service if you have questions.


BIOMARKERS

Molecular Biopsy of Human Tumors

- a resource for Precision Medicine *

114 related articles for article (PubMed ID: 10636236)

  • 1. 6-Acylamino-2-[(alkylsulfonyl)oxy]-1H-isoindole-1,3-dione mechanism-based inhibitors of human leukocyte elastase.
    Kerrigan JE; Walters MC; Forrester KJ; Crowder JB; Christopher LJ
    Bioorg Med Chem Lett; 2000 Jan; 10(1):27-30. PubMed ID: 10636236
    [TBL] [Abstract][Full Text] [Related]  

  • 2. 6-Acylamino-2-1[(ethylsulfonyl)oxy]-1H-isoindole-1,3-diones mechanism-based inhibitors of human leukocyte elastase and cathepsin G: effect of chirality in the 6-acylamino substituent on inhibitory potency and selectivity.
    Vagnoni LM; Gronostaj M; Kerrigan JE
    Bioorg Med Chem; 2001 Mar; 9(3):637-45. PubMed ID: 11310598
    [TBL] [Abstract][Full Text] [Related]  

  • 3. The serpin MNEI inhibits elastase-like and chymotrypsin-like serine proteases through efficient reactions at two active sites.
    Cooley J; Takayama TK; Shapiro SD; Schechter NM; Remold-O'Donnell E
    Biochemistry; 2001 Dec; 40(51):15762-70. PubMed ID: 11747453
    [TBL] [Abstract][Full Text] [Related]  

  • 4. N-Acyl and N-sulfonyloxazolidine-2,4-diones are pseudo-irreversible inhibitors of serine proteases.
    Santana AB; Lucas SD; Gonçalves LM; Correia HF; Cardote TA; Guedes RC; Iley J; Moreira R
    Bioorg Med Chem Lett; 2012 Jun; 22(12):3993-7. PubMed ID: 22595175
    [TBL] [Abstract][Full Text] [Related]  

  • 5. Inhibition of serine proteases: activity of 1,3-diazetidine-2,4-diones.
    Aoyama Y; Uenaka M; Konoike T; Hayasaki-Kajiwara Y; Naya N; Nakajima M
    Bioorg Med Chem Lett; 2001 Jul; 11(13):1691-4. PubMed ID: 11425539
    [TBL] [Abstract][Full Text] [Related]  

  • 6. Leucine-phenylalanine dipeptide-based N-mesyloxysuccinimides: synthesis of all four stereoisomers and their assay against serine proteases.
    Abell AD; Oldham MD
    Bioorg Med Chem Lett; 1999 Feb; 9(3):497-500. PubMed ID: 10091709
    [TBL] [Abstract][Full Text] [Related]  

  • 7. Succinimide and saccharin-based enzyme-activated inhibitors of serine proteases.
    Martyn DC; Moore MJ; Abell AD
    Curr Pharm Des; 1999 Jun; 5(6):405-15. PubMed ID: 10390606
    [TBL] [Abstract][Full Text] [Related]  

  • 8. Esters and amides of 6-(chloromethyl)-2-oxo-2H-1-benzopyran-3-carboxylic acid as inhibitors of alpha-chymotrypsin: significance of the "aromatic" nature of the novel ester-type coumarin for strong inhibitory activity.
    Pochet L; Doucet C; Schynts M; Thierry N; Boggetto N; Pirotte B; Jiang KY; Masereel B; de Tullio P; Delarge J; Reboud-Ravaux M
    J Med Chem; 1996 Jun; 39(13):2579-85. PubMed ID: 8691456
    [TBL] [Abstract][Full Text] [Related]  

  • 9. Potent and specific inhibition of human leukocyte elastase, cathepsin G and proteinase 3 by sulfone derivatives employing the 1,2,5-thiadiazolidin-3-one 1,1 dioxide scaffold.
    Groutas WC; Kuang R; Ruan S; Epp JB; Venkataraman R; Truong TM
    Bioorg Med Chem; 1998 Jun; 6(6):661-71. PubMed ID: 9681132
    [TBL] [Abstract][Full Text] [Related]  

  • 10. Mechanism-based isocoumarin inhibitors for human leukocyte elastase. Effect of the 7-amino substituent and 3-alkoxy group in 3-alkoxy-7-amino-4-chloroisocoumarins on inhibitory potency.
    Kerrigan JE; Oleksyszyn J; Kam CM; Selzler J; Powers JC
    J Med Chem; 1995 Feb; 38(3):544-52. PubMed ID: 7853347
    [TBL] [Abstract][Full Text] [Related]  

  • 11. Effect of YM-47141, a new inhibitor produced by Flexibactor sp. Q17897, on elastase.
    Teramura K; Yasumuro K; Abe K
    J Enzyme Inhib; 1996 Aug; 11(1):33-8. PubMed ID: 9204394
    [TBL] [Abstract][Full Text] [Related]  

  • 12. Synthesis of a trihexacontapeptide corresponding to the sequence 8-70 of eglin c and studies on the relationship between the structure and the inhibitory activity against human leukocyte elastase, cathepsin G and alpha-chymotrypsin.
    Okada Y; Tsuboi S; Tsuda Y; Nagamatsu Y; Yamamoto J
    FEBS Lett; 1990 Oct; 272(1-2):113-6. PubMed ID: 2226822
    [TBL] [Abstract][Full Text] [Related]  

  • 13. Potential of pyrazolooxadiazinone derivatives as serine protease inhibitors.
    Vicentini CB; Guarneri M; Andrisano V; Guccione S; Langer T; Marschhofer R; Chabin R; Edison AM; Huang X; Knight WB; Giori P
    J Enzyme Inhib; 2001 Jan; 16(1):15-34. PubMed ID: 11496832
    [TBL] [Abstract][Full Text] [Related]  

  • 14. Synthesis and mechanism of action of novel thiocarbamate inhibitors of human leukocyte elastase.
    Li-Pan ZS; Joshi HV; Digenis GA
    J Enzyme Inhib; 2000; 15(1):63-77. PubMed ID: 10850955
    [TBL] [Abstract][Full Text] [Related]  

  • 15. Glycosaminoglycans regulate elastase inhibition by oxidized secretory leukoprotease inhibitor.
    Ying QL; Kemme M; Saunders D; Simon SR
    Am J Physiol; 1997 Mar; 272(3 Pt 1):L533-41. PubMed ID: 9124611
    [TBL] [Abstract][Full Text] [Related]  

  • 16. 2,4,5-Triphenylisothiazol-3 (2H)-one 1,1-dioxides as inhibitors of human leukocyte elastase.
    Gütschow M; Pietsch M; Themann A; Fahrig J; Schulze B
    J Enzyme Inhib Med Chem; 2005 Aug; 20(4):341-7. PubMed ID: 16206828
    [TBL] [Abstract][Full Text] [Related]  

  • 17. Phosphonic pseudopeptides as human neutrophil elastase inhibitors--a combinatorial approach.
    Sieńczyk M; Podgórski D; Błażejewska A; Kulbacka J; Saczko J; Oleksyszyn J
    Bioorg Med Chem; 2011 Feb; 19(3):1277-84. PubMed ID: 21216608
    [TBL] [Abstract][Full Text] [Related]  

  • 18. alpha-Aminoalkylphosphonate di(chlorophenyl) esters as inhibitors of serine proteases.
    Boduszek B; Brown AD; Powers JC
    J Enzyme Inhib; 1994; 8(3):147-58. PubMed ID: 7539484
    [TBL] [Abstract][Full Text] [Related]  

  • 19. Reactive sites of the 21-kD protein inhibitor of serine proteinases from potato tubers.
    Valueva TA; Revina TA; Mosolov VV
    Biochemistry (Mosc); 1999 Sep; 64(9):1074-8. PubMed ID: 10521725
    [TBL] [Abstract][Full Text] [Related]  

  • 20. Amino acid-derived phthalimide and saccharin derivatives as inhibitors of human leukocyte elastase, cathepsin G, and proteinase 3.
    Groutas WC; Chong LS; Venkataraman R; Kuang R; Epp JB; Houser-Archield N; Huang H; Hoidal JR
    Arch Biochem Biophys; 1996 Aug; 332(2):335-40. PubMed ID: 8806743
    [TBL] [Abstract][Full Text] [Related]  

    [Next]    [New Search]
    of 6.