154 related articles for article (PubMed ID: 10658575)
1. Synthesis and BZR affinity of pyrazolo[1,5-a]pyrimidine derivatives. Part 1: study of the structural features for BZR recognition.
Selleri S; Bruni F; Costagli C; Costanzo A; Guerrini G; Ciciani G; Costa B; Martini C
Bioorg Med Chem; 1999 Dec; 7(12):2705-11. PubMed ID: 10658575
[TBL] [Abstract][Full Text] [Related]
2. New 2,3-substituted 4,7-dihydro-6-(1'H-pyrazol-3'-yl)pyrazolo[1,5-a] pyrimidin-7-ones and related compounds: synthesis and benzodiazepine receptor binding study.
Selleri S; Bruni F; Costanzo A; Guerrini G; Casilli ML; Giusti L; Lucacchini A; Martini C
Farmaco; 1995 Oct; 50(10):679-87. PubMed ID: 8590575
[TBL] [Abstract][Full Text] [Related]
3. Synthesis of 7-(2-dimethylaminovinyl) derivatives of pyrazolo[1,5-a] pyrimidines, as precursors of new tricyclic series. Binding studies of BDZ receptor.
Bruni F; Costanzo A; Selleri S; Guerrini G; Giusti L; Martini C; Lucacchini A
Farmaco; 1993 Feb; 48(2):309-19. PubMed ID: 8388217
[TBL] [Abstract][Full Text] [Related]
4. Structure-activity relationship studies of novel pyrazolo[1,5-c][1,3]benzoxazines: synthesis and benzodiazepine receptor affinity.
Varano F; Catarzi D; Colotta V; Cecchi L; Filacchioni G; Galli A; Costagli C
Arch Pharm (Weinheim); 1996 Dec; 329(12):529-34. PubMed ID: 9038420
[TBL] [Abstract][Full Text] [Related]
5. Synthesis and pharmacological evaluation of pyrazolo[1,5-a]pyrimidin-7(4H)-one derivatives as potential GABA
Guerrini G; Ciciani G; Daniele S; Di Cesare Mannelli L; Ghelardini C; Martini C; Selleri S
Bioorg Med Chem; 2017 Mar; 25(6):1901-1906. PubMed ID: 28237554
[TBL] [Abstract][Full Text] [Related]
6. Pyrazolo[1,5-a]pyrimidine CRF-1 receptor antagonists.
Wustrow DJ; Capiris T; Rubin R; Knobelsdorf JA; Akunne H; Davis MD; MacKenzie R; Pugsley TA; Zoski KT; Heffner TG; Wise LD
Bioorg Med Chem Lett; 1998 Aug; 8(16):2067-70. PubMed ID: 9873487
[TBL] [Abstract][Full Text] [Related]
7. Pyrazolo[4,3-e]-1,2,4-triazolo[1,5-c]pyrimidine derivatives as highly potent and selective human A(3) adenosine receptor antagonists.
Baraldi PG; Cacciari B; Romagnoli R; Spalluto G; Klotz KN; Leung E; Varani K; Gessi S; Merighi S; Borea PA
J Med Chem; 1999 Nov; 42(22):4473-8. PubMed ID: 10579811
[No Abstract] [Full Text] [Related]
8. Design, synthesis, and biological evaluation of C9- and C2-substituted pyrazolo[4,3-e]-1,2,4-triazolo[1,5-c]pyrimidines as new A2A and A3 adenosine receptors antagonists.
Baraldi PG; Fruttarolo F; Tabrizi MA; Preti D; Romagnoli R; El-Kashef H; Moorman A; Varani K; Gessi S; Merighi S; Borea PA
J Med Chem; 2003 Mar; 46(7):1229-41. PubMed ID: 12646033
[TBL] [Abstract][Full Text] [Related]
9. Tricyclic heteroaromatic systems. Pyrazolo[3,4-c]quinolin-4-ones and pyrazolo[3,4-c]quinoline-1,4-diones: synthesis and benzodiazepine receptor activity.
Catarzi D; Colotta V; Varano F; Cecchi L; Filacchioni G; Galli A; Costagli C
Arch Pharm (Weinheim); 1997 Dec; 330(12):383-6. PubMed ID: 9474897
[TBL] [Abstract][Full Text] [Related]
10. Synthesis and biological evaluation of 7-(aminoalkyl)pyrazolo[1,5-a]pyrimidine derivatives as cathepsin K inhibitors.
Petek N; Štefane B; Novinec M; Svete J
Bioorg Chem; 2019 Mar; 84():226-238. PubMed ID: 30502634
[TBL] [Abstract][Full Text] [Related]
11. Design and synthesis of 3-(2-pyridyl)pyrazolo[1,5-a]pyrimidines as potent CRF1 receptor antagonists.
Huang CQ; Wilcoxen KM; Grigoriadis DE; McCarthy JR; Chen C
Bioorg Med Chem Lett; 2004 Aug; 14(15):3943-7. PubMed ID: 15225703
[TBL] [Abstract][Full Text] [Related]
12. Ether analogues of DPA-714 with subnanomolar affinity for the translocator protein (TSPO).
Banister SD; Beinat C; Wilkinson SM; Shen B; Bartoli C; Selleri S; Da Pozzo E; Martini C; Chin FT; Kassiou M
Eur J Med Chem; 2015 Mar; 93():392-400. PubMed ID: 25725375
[TBL] [Abstract][Full Text] [Related]
13. Structure-activity relationship studies at the benzodiazepine receptor (BZR): a comparison of the substitutent effects of pyrazoloquinolinone analogs.
Fryer RI; Zhang P; Rios R; Gu ZQ; Basile AS; Skolnick P
J Med Chem; 1993 May; 36(11):1669-73. PubMed ID: 8388472
[TBL] [Abstract][Full Text] [Related]
14. Design, synthesis and anticancer evaluation of novel pyrazole, pyrazolo[3,4-d]pyrimidine and their glycoside derivatives.
Nassar IF; El Farargy AF; Abdelrazek FM; Ismail NSM
Nucleosides Nucleotides Nucleic Acids; 2017 Apr; 36(4):275-291. PubMed ID: 28323527
[TBL] [Abstract][Full Text] [Related]
15. Synthesis and isomerization of some novel pyrazolopyrimidine and pyrazolotriazolopyrimidine derivatives.
Rashad AE; Shamroukh AH; Abdel-Megeid RE; Ali HS
Molecules; 2014 Apr; 19(5):5459-69. PubMed ID: 24776812
[TBL] [Abstract][Full Text] [Related]
16. Structure-activity relationship studies of pyrazolo[3,4-d]pyrimidine derivatives leading to the discovery of a novel multikinase inhibitor that potently inhibits FLT3 and VEGFR2 and evaluation of its activity against acute myeloid leukemia in vitro and in vivo.
Yang LL; Li GB; Ma S; Zou C; Zhou S; Sun QZ; Cheng C; Chen X; Wang LJ; Feng S; Li LL; Yang SY
J Med Chem; 2013 Feb; 56(4):1641-55. PubMed ID: 23362959
[TBL] [Abstract][Full Text] [Related]
17. Synthesis of 1H-pyrazolo[4,3-d]pyrimidine-7(6H)-ones and pyrazolo-5-carboxamides and interaction with benzodiazepine and adenosine A1 receptors in rat cerebral cortex.
Baraldi PG; Casolari A; Manfredini S; Periotto V; Zanirato V; Florio C; Traversa V; Bertelli GM; Borea PA
Arzneimittelforschung; 1988 Sep; 38(9):1262-5. PubMed ID: 2852012
[TBL] [Abstract][Full Text] [Related]
18. A facile and novel synthesis of N(2)-, C(6)-substituted pyrazolo[3,4-d]pyrimidine-4 carboxylate derivatives as adenosine receptor antagonists.
Venkatesan G; Paira P; Cheong SL; Federico S; Klotz KN; Spalluto G; Pastorin G
Eur J Med Chem; 2015 Mar; 92():784-98. PubMed ID: 25633494
[TBL] [Abstract][Full Text] [Related]
19. Synthesis and structure-activity relationship of pyrazolo[3,4-d]pyrimidines: potent and selective adenosine A1 receptor antagonists.
Poulsen SA; Quinn RJ
J Med Chem; 1996 Oct; 39(21):4156-61. PubMed ID: 8863792
[TBL] [Abstract][Full Text] [Related]
20. Synthesis and benzodiazepine receptor affinity of pyrazolo[1,5-a]pyrimidine derivatives. 3. New 6-(3-thienyl) series as alpha 1 selective ligands.
Selleri S; Bruni F; Costagli C; Costanzo A; Guerrini G; Ciciani G; Gratteri P; Bonaccini C; Malmberg Aiello P; Besnard F; Renard S; Costa B; Martini C
J Med Chem; 2003 Jan; 46(2):310-3. PubMed ID: 12519068
[TBL] [Abstract][Full Text] [Related]
[Next] [New Search]
