BIOMARKERS

Molecular Biopsy of Human Tumors

- a resource for Precision Medicine *

130 related articles for article (PubMed ID: 10733601)

  • 1. Carbonic anhydrase activators - part 21. Novel activators of isozymes I, II and IV incorporating carboxamido and ureido histamine moieties.
    Scozzafava A; Supuran CT
    Eur J Med Chem; 2000 Jan; 35(1):31-9. PubMed ID: 10733601
    [TBL] [Abstract][Full Text] [Related]  

  • 2. Carbonic anhydrase activators: synthesis of high affinity isozymes I, II and IV activators, derivatives of 4-(4-tosylureido-amino acyl)ethyl-1H-imidazole (histamine derivatives).
    Scozzafava A; Iorga B; Supuran CT
    J Enzyme Inhib; 2000; 15(2):139-61. PubMed ID: 10938540
    [TBL] [Abstract][Full Text] [Related]  

  • 3. Carbonic anhydrase activators: amino acyl/dipeptidyl histamine derivatives bind with high affinity to isozymes I, II and IV and act as efficient activators.
    Supuran CT; Scozzafava A
    Bioorg Med Chem; 1999 Dec; 7(12):2915-23. PubMed ID: 10658596
    [TBL] [Abstract][Full Text] [Related]  

  • 4. Carbonic anhydrase activators: synthesis of high affinity isozymes I, II and IV activators, derivatives of 4-(arylsulfonylureido-amino acyl)ethyl-1H-imidazole.
    Supuran CT; Scozzafava A
    J Enzyme Inhib; 2000; 15(5):471-86. PubMed ID: 11030087
    [TBL] [Abstract][Full Text] [Related]  

  • 5. Carbonic anhydrase activators. Part 24. High affinity isozymes I, II and IV activators, derivatives of 4-(4-chlorophenylsulfonylureido-amino acyl)ethyl-1H-imidazole.
    Scozzafava A; Supuran CT
    Eur J Pharm Sci; 2000 Mar; 10(1):29-41. PubMed ID: 10699381
    [TBL] [Abstract][Full Text] [Related]  

  • 6. Carbonic anhydrase activators: high affinity isozymes I, II, and IV activators, incorporating a beta-alanyl-histidine scaffold.
    Scozzafava A; Supuran CT
    J Med Chem; 2002 Jan; 45(2):284-91. PubMed ID: 11784133
    [TBL] [Abstract][Full Text] [Related]  

  • 7. Synthesis and biological evaluation of histamine Schiff bases as carbonic anhydrase I, II, IV, VII, and IX activators.
    Akocak S; Lolak N; Vullo D; Durgun M; Supuran CT
    J Enzyme Inhib Med Chem; 2017 Dec; 32(1):1305-1312. PubMed ID: 29072105
    [TBL] [Abstract][Full Text] [Related]  

  • 8. Carbonic anhydrase activators: design of high affinity isozymes I, II, and IV activators, incorporating tri-/tetrasubstituted-pyridinium-azole moieties.
    Ilies M; Banciu MD; Ilies MA; Scozzafava A; Caproiu MT; Supuran CT
    J Med Chem; 2002 Jan; 45(2):504-10. PubMed ID: 11784154
    [TBL] [Abstract][Full Text] [Related]  

  • 9. Novel carbonic anhydrase isozymes I, II and IV activators incorporating sulfonyl-histamino moieties.
    Briganti F; Scozzafava A; Supuran CT
    Bioorg Med Chem Lett; 1999 Jul; 9(14):2043-8. PubMed ID: 10450978
    [TBL] [Abstract][Full Text] [Related]  

  • 10. Pyridinium derivatives of histamine are potent activators of cytosolic carbonic anhydrase isoforms I, II and VII.
    Dave K; Scozzafava A; Vullo D; Supuran CT; Ilies MA
    Org Biomol Chem; 2011 Apr; 9(8):2790-800. PubMed ID: 21369613
    [TBL] [Abstract][Full Text] [Related]  

  • 11. Carbonic anhydrase activators. Activation of isozymes I, II, IV, VA, VII, and XIV with l- and d-histidine and crystallographic analysis of their adducts with isoform II: engineering proton-transfer processes within the active site of an enzyme.
    Temperini C; Scozzafava A; Vullo D; Supuran CT
    Chemistry; 2006 Sep; 12(27):7057-66. PubMed ID: 16807956
    [TBL] [Abstract][Full Text] [Related]  

  • 12. Carbonic anhydrase activators: X-ray crystal structure of the adduct of human isozyme II with L-histidine as a platform for the design of stronger activators.
    Temperini C; Scozzafava A; Puccetti L; Supuran CT
    Bioorg Med Chem Lett; 2005 Dec; 15(23):5136-41. PubMed ID: 16214338
    [TBL] [Abstract][Full Text] [Related]  

  • 13. Carbonic anhydrase activators: gold nanoparticles coated with derivatized histamine, histidine, and carnosine show enhanced activatory effects on several mammalian isoforms.
    Saada MC; Montero JL; Vullo D; Scozzafava A; Winum JY; Supuran CT
    J Med Chem; 2011 Mar; 54(5):1170-7. PubMed ID: 21291238
    [TBL] [Abstract][Full Text] [Related]  

  • 14. Carbonic anhydrase inhibitors: novel sulfonamides incorporating 1,3,5-triazine moieties as inhibitors of the cytosolic and tumour-associated carbonic anhydrase isozymes I, II and IX.
    Garaj V; Puccetti L; Fasolis G; Winum JY; Montero JL; Scozzafava A; Vullo D; Innocenti A; Supuran CT
    Bioorg Med Chem Lett; 2005 Jun; 15(12):3102-8. PubMed ID: 15905091
    [TBL] [Abstract][Full Text] [Related]  

  • 15. Carbonic anhydrase activators: L-Adrenaline plugs the active site entrance of isozyme II, activating better isoforms I, IV, VA, VII, and XIV.
    Temperini C; Innocenti A; Scozzafava A; Mastrolorenzo A; Supuran CT
    Bioorg Med Chem Lett; 2007 Feb; 17(3):628-35. PubMed ID: 17127057
    [TBL] [Abstract][Full Text] [Related]  

  • 16. Carbonic anhydrase activators. The selective serotonin reuptake inhibitors fluoxetine, sertraline and citalopram are strong activators of isozymes I and II.
    Casini A; Caccia S; Scozzafava A; Supuran CT
    Bioorg Med Chem Lett; 2003 Aug; 13(16):2765-8. PubMed ID: 12873510
    [TBL] [Abstract][Full Text] [Related]  

  • 17. Carbonic anhydrase inhibitors: N-cyanosulfonamides, a new class of high affinity isozyme II and IV inhibitors.
    Supuran CT; Scozzafava A; Briganti F
    J Enzyme Inhib; 1999; 14(4):289-306. PubMed ID: 10445050
    [TBL] [Abstract][Full Text] [Related]  

  • 18. Carbonic anhydrase inhibitors: ureido and thioureido derivatives of aromatic sulfonamides possessing increased affinities for isozyme I. A novel route to 2,5-disubstituted-1,3,4-thiadiazoles via thioureas, and their interaction with isozymes I, II and IV.
    Scozzafava A; Supuran CT
    J Enzyme Inhib; 1998 Apr; 13(2):103-23. PubMed ID: 9629531
    [TBL] [Abstract][Full Text] [Related]  

  • 19. α-Carbonic anhydrases are strongly activated by spinaceamine derivatives.
    Akocak S; Lolak N; Bua S; Nocentini A; Karakoc G; Supuran CT
    Bioorg Med Chem; 2019 Mar; 27(5):800-804. PubMed ID: 30683554
    [TBL] [Abstract][Full Text] [Related]  

  • 20. Mono- and di-halogenated histamine, histidine and carnosine derivatives are potent carbonic anhydrase I, II, VII, XII and XIV activators.
    Saada MC; Vullo D; Montero JL; Scozzafava A; Supuran CT; Winum JY
    Bioorg Med Chem; 2014 Sep; 22(17):4752-8. PubMed ID: 25082511
    [TBL] [Abstract][Full Text] [Related]  

    [Next]    [New Search]
    of 7.