These tools will no longer be maintained as of December 31, 2024. Archived website can be found here. PubMed4Hh GitHub repository can be found here. Contact NLM Customer Service if you have questions.


BIOMARKERS

Molecular Biopsy of Human Tumors

- a resource for Precision Medicine *

690 related articles for article (PubMed ID: 10911016)

  • 1. Novel approaches for designing 5'-O-ester prodrugs of 3'-azido-2', 3'-dideoxythymidine (AZT).
    Parang K; Wiebe LI; Knaus EE
    Curr Med Chem; 2000 Oct; 7(10):995-1039. PubMed ID: 10911016
    [TBL] [Abstract][Full Text] [Related]  

  • 2. Design of new mononucleotide prodrugs: aryl (SATE) phosphotriester derivatives.
    Peyrottes S; Schlienger N; Beltran T; Lefebvre I; Pompon A; Gosselin G; Aubertin AM; Imbach JL; Périgaud C
    Nucleosides Nucleotides Nucleic Acids; 2001; 20(4-7):315-21. PubMed ID: 11563043
    [TBL] [Abstract][Full Text] [Related]  

  • 3. Characterization of the activation pathway of phosphoramidate triester prodrugs of stavudine and zidovudine.
    Saboulard D; Naesens L; Cahard D; Salgado A; Pathirana R; Velazquez S; McGuigan C; De Clercq E; Balzarini J
    Mol Pharmacol; 1999 Oct; 56(4):693-704. PubMed ID: 10496951
    [TBL] [Abstract][Full Text] [Related]  

  • 4. S-Acyl-2-thioethyl aryl phosphotriester derivatives as mononucleotide prodrugs.
    Schlienger N; Peyrottes S; Kassem T; Imbach JL; Gosselin G; Aubertin AM; Périgaud C
    J Med Chem; 2000 Nov; 43(23):4570-4. PubMed ID: 11087582
    [TBL] [Abstract][Full Text] [Related]  

  • 5. New 3'-azido-3'-deoxythymidin-5'-yl O-(omega-hydroxyalkyl) carbonate prodrugs: synthesis and anti-HIV evaluation.
    Vlieghe P; Bihel F; Clerc T; Pannecouque C; Witvrouw M; De Clercq E; Salles JP; Chermann JC; Kraus JL
    J Med Chem; 2001 Mar; 44(5):777-86. PubMed ID: 11262088
    [TBL] [Abstract][Full Text] [Related]  

  • 6. A step further in the SATE mononucleotide prodrug approach.
    Peyrottes S; Villard AL; Coussot G; Augustijns P; Lefebvre I; Aubertin AM; Gosselin G; Périgaud C
    Nucleic Acids Symp Ser (Oxf); 2008; (52):539-40. PubMed ID: 18776492
    [TBL] [Abstract][Full Text] [Related]  

  • 7. Dipeptide derivatives of AZT: synthesis, chemical stability, activation in human plasma, hPEPT1 affinity, and antiviral activity.
    Santos C; Morais J; Gouveia L; de Clercq E; Pannecouque C; Nielsen CU; Steffansen B; Moreira R; Gomes P
    ChemMedChem; 2008 Jun; 3(6):970-8. PubMed ID: 18389514
    [TBL] [Abstract][Full Text] [Related]  

  • 8. In vitro anti-hepatitis B virus activities of 5"-O-myristoyl analogue derivatives of 3"-fluoro-2",3"-dideoxythymidine (FLT) and 3"-azido-2",3"-dideoxythymidine (AZT).
    Parang K; Wiebe LI; Knaus EE; Huang JS; Tyrrell DL
    J Pharm Pharm Sci; 1998; 1(3):108-14. PubMed ID: 10948398
    [TBL] [Abstract][Full Text] [Related]  

  • 9. Synthesis and anti-HIV activity of steroidal prodrugs of 3'-azido-3'-deoxythymidine (AZT).
    Balagopala MI; Ollapally AP; Lee HJ
    Cell Mol Biol (Noisy-le-grand); 1995; 41 Suppl 1():S1-7. PubMed ID: 8574137
    [TBL] [Abstract][Full Text] [Related]  

  • 10. Phenyl phosphotriester derivatives of AZT: variations upon the SATE moiety.
    Villard AL; Coussot G; Lefebvre I; Augustijns P; Aubertin AM; Gosselin G; Peyrottes S; Périgaud C
    Bioorg Med Chem; 2008 Aug; 16(15):7321-9. PubMed ID: 18585917
    [TBL] [Abstract][Full Text] [Related]  

  • 11. Synthesis and in vitro activity of long-chain 5'-O-[(alkoxycarbonyl)phosphinyl]-3'-azido-3'-deoxythymidines against wild-type and AZT- and foscarnet-resistant strains of HIV-1.
    Rosowsky A; Fu H; Pai N; Mellors J; Richman DD; Hostetler KY
    J Med Chem; 1997 Aug; 40(16):2482-90. PubMed ID: 9258355
    [TBL] [Abstract][Full Text] [Related]  

  • 12. New bis(SATE) prodrug of AZT 5'-monophosphate: in vitro anti-HIV activity, stability, and potential oral absorption.
    Shafiee M; Deferme S; Villard AL; Egron D; Gosselin G; Imbach JL; Lioux T; Pompon A; Varray S; Aubertin AM; Van Den Mooter G; Kinget R; Périgaud C; Augustijns P
    J Pharm Sci; 2001 Apr; 90(4):448-63. PubMed ID: 11170035
    [TBL] [Abstract][Full Text] [Related]  

  • 13. Synthesis, in vitro anti-human immunodeficiency virus structure-activity relationships and biological stability of 5'-O-myristoyl analogue derivatives of 3'-azido-2',3'-dideoxythymidine (AZT) as potential prodrugs.
    Parang K; Wiebe LI; Knaus EE
    Antivir Chem Chemother; 1998 Jul; 9(4):311-23. PubMed ID: 9875410
    [TBL] [Abstract][Full Text] [Related]  

  • 14. Probing the mechanism of action and decomposition of amino acid phosphomonoester amidates of antiviral nucleoside prodrugs.
    McIntee EJ; Remmel RP; Schinazi RF; Abraham TW; Wagner CR
    J Med Chem; 1997 Oct; 40(21):3323-31. PubMed ID: 9341906
    [TBL] [Abstract][Full Text] [Related]  

  • 15. New 3'-azido-3'-deoxythymidin-5'-yl O-(4-hydroxyalkyl or -alkenyl or -alkylepoxide) carbonate prodrugs: synthesis and anti-HIV evaluation.
    Vlieghe P; Clerc T; Pannecouque C; Witvrouw M; De Clercq E; Salles JP; Kraus JL
    J Med Chem; 2001 Aug; 44(18):3014-21. PubMed ID: 11520210
    [TBL] [Abstract][Full Text] [Related]  

  • 16. Synthesis and anti-retroviral activity of O,O'-bis(3'-azido-2',3'-dideoxythymidin-5'-yl) phosphoramidate derivatives.
    Kers I; Stawiński J; Girardet JL; Imbach JL; Périgaud C; Gosselin G; Aubertin AM
    Nucleosides Nucleotides; 1999 Oct; 18(10):2317-25. PubMed ID: 10616733
    [TBL] [Abstract][Full Text] [Related]  

  • 17. Intracellular metabolism of CycloSaligenyl 3'-azido-2', 3'-dideoxythymidine monophosphate, a prodrug of 3'-azido-2', 3'-dideoxythymidine (zidovudine).
    Balzarini J; Naesens L; Aquaro S; Knispel T; Perno C; De Clercq E; Meier C
    Mol Pharmacol; 1999 Dec; 56(6):1354-61. PubMed ID: 10570065
    [TBL] [Abstract][Full Text] [Related]  

  • 18. Amino acid phosphoramidate monoesters of 3'-azido-3'-deoxythymidine: relationship between antiviral potency and intracellular metabolism.
    Chang S; Griesgraber GW; Southern PJ; Wagner CR
    J Med Chem; 2001 Jan; 44(2):223-31. PubMed ID: 11170632
    [TBL] [Abstract][Full Text] [Related]  

  • 19. Anti-HIV pronucleotides: decomposition pathways and correlation with biological activities.
    Egron D; Lefebvre I; Périgaud C; Beltran T; Pompon A; Gosselin G; Aubertin AM; Imbach JL
    Bioorg Med Chem Lett; 1998 May; 8(9):1045-50. PubMed ID: 9871705
    [TBL] [Abstract][Full Text] [Related]  

  • 20. Antiretroviral activity and cytotoxicity of novel zidovudine (AZT) derivatives and the relation to their chemical structure.
    Turk G; Moroni G; Pampuro S; Briñón MC; Salomón H
    Int J Antimicrob Agents; 2002 Oct; 20(4):282-8. PubMed ID: 12385685
    [TBL] [Abstract][Full Text] [Related]  

    [Next]    [New Search]
    of 35.