These tools will no longer be maintained as of December 31, 2024. Archived website can be found here. PubMed4Hh GitHub repository can be found here. Contact NLM Customer Service if you have questions.


BIOMARKERS

Molecular Biopsy of Human Tumors

- a resource for Precision Medicine *

131 related articles for article (PubMed ID: 11008374)

  • 1. beta-Lactam derivatives as enzyme inhibitors: 1-peptidyl derivatives of 4-phenylazetidin-2-one as inhibitors of elastase and papain.
    Achilles K; Schirmeister T; Otto HH
    Arch Pharm (Weinheim); 2000 Aug; 333(8):243-53. PubMed ID: 11008374
    [TBL] [Abstract][Full Text] [Related]  

  • 2. beta-Lactam derivatives as enzyme inhibitors: N-substituted derivatives of (S)-4-oxoazetidine-2-carboxylate as inhibitors of elastase and papain.
    Achilles K; Schneider M; Schirmeister T; Otto HH
    Pharmazie; 2000 Nov; 55(11):798-802. PubMed ID: 11125993
    [TBL] [Abstract][Full Text] [Related]  

  • 3. beta-Lactam derivatives as enzyme inhibitors: derivatives of (E)-2-[(RS)-1-(4-methoxyphenyl)-2-oxo-4-phenylazetidin-3-ylidene]propionic acid.
    Venz C; Otto HH
    Pharmazie; 2001 Sep; 56(9):686-90. PubMed ID: 11593986
    [TBL] [Abstract][Full Text] [Related]  

  • 4. Irreversible inhibition of serine proteases by peptide derivatives of (alpha-aminoalkyl)phosphonate diphenyl esters.
    Oleksyszyn J; Powers JC
    Biochemistry; 1991 Jan; 30(2):485-93. PubMed ID: 1988040
    [TBL] [Abstract][Full Text] [Related]  

  • 5. beta-lactam derivatives as enzyme inhibitors: carboxy peptidyl derivatives of (S)-4-oxoazetidine-2-carboxylate as peptidomimetics.
    Schneider M; Otto HH
    Arch Pharm (Weinheim); 2001 May; 334(5):167-72. PubMed ID: 11413823
    [TBL] [Abstract][Full Text] [Related]  

  • 6. In vitro evaluation of the antielastase activity of polycyclic β-lactams.
    Monleón LM; Díez-García F; Zamora H; Anaya J; Grande M; de Diego JG; Rodríguez FD
    Bioorg Chem; 2012 Dec; 45():29-35. PubMed ID: 23064125
    [TBL] [Abstract][Full Text] [Related]  

  • 7. The novel serpin endopin 2 demonstrates cross-class inhibition of papain and elastase: localization of endopin 2 to regulated secretory vesicles of neuroendocrine chromaffin cells.
    Hwang SR; Steineckert B; Toneff T; Bundey R; Logvinova AV; Goldsmith P; Hook VY
    Biochemistry; 2002 Aug; 41(33):10397-405. PubMed ID: 12173926
    [TBL] [Abstract][Full Text] [Related]  

  • 8. 1-Alkoxycarbonyl-3-halogenoazetidin-2-ones as elastase (PPE) inhibitors.
    Gérard S; Nollet G; Vande Put J; Marchand-Brynaert J
    Bioorg Med Chem; 2002 Dec; 10(12):3955-64. PubMed ID: 12413847
    [TBL] [Abstract][Full Text] [Related]  

  • 9. Orally active beta-lactam inhibitors of human leukocyte elastase. 3. Stereospecific synthesis and structure-activity relationships for 3,3-dialkylazetidin-2-ones.
    Finke PE; Shah SK; Fletcher DS; Ashe BM; Brause KA; Chandler GO; Dellea PS; Hand KM; Maycock AL; Osinga DG
    J Med Chem; 1995 Jun; 38(13):2449-62. PubMed ID: 7608910
    [TBL] [Abstract][Full Text] [Related]  

  • 10. Peptidyl beta-homo-aspartals (3-amino-4-carboxybutyraldehydes): new specific inhibitors of caspases.
    Bajusz S; Fauszt I; Németh K; Barabás E; Juhász A; Patthy M; Bauer PI
    Biopolymers; 1999; 51(1):109-18. PubMed ID: 10380358
    [TBL] [Abstract][Full Text] [Related]  

  • 11. Synthesis and evaluation of N1/C4-substituted beta-lactams as PPE and HLE inhibitors.
    Gérard S; Galleni M; Dive G; Marchand-Brynaert J
    Bioorg Med Chem; 2004 Jan; 12(1):129-38. PubMed ID: 14697778
    [TBL] [Abstract][Full Text] [Related]  

  • 12. Inhibition of elastase by N-sulfonylaryl beta-lactams: anatomy of a stable acyl-enzyme complex.
    Wilmouth RC; Westwood NJ; Anderson K; Brownlee W; Claridge TD; Clifton IJ; Pritchard GJ; Aplin RT; Schofield CJ
    Biochemistry; 1998 Dec; 37(50):17506-13. PubMed ID: 9860865
    [TBL] [Abstract][Full Text] [Related]  

  • 13. Azapeptides as inhibitors and active site titrants for cysteine proteinases.
    Xing R; Hanzlik RP
    J Med Chem; 1998 Apr; 41(8):1344-51. PubMed ID: 9548822
    [TBL] [Abstract][Full Text] [Related]  

  • 14. New peptidic cysteine protease inhibitors derived from the electrophilic alpha-amino acid aziridine-2,3-dicarboxylic acid.
    Schirmeister T
    J Med Chem; 1999 Feb; 42(4):560-72. PubMed ID: 10052963
    [TBL] [Abstract][Full Text] [Related]  

  • 15. alpha-Aminoalkylphosphonate di(chlorophenyl) esters as inhibitors of serine proteases.
    Boduszek B; Brown AD; Powers JC
    J Enzyme Inhib; 1994; 8(3):147-58. PubMed ID: 7539484
    [TBL] [Abstract][Full Text] [Related]  

  • 16. Inhibition of human serine proteases by substituted 2-azetidinones.
    Knight WB; Chabin R; Green B
    Arch Biochem Biophys; 1992 Aug; 296(2):704-8. PubMed ID: 1632655
    [TBL] [Abstract][Full Text] [Related]  

  • 17. Structure-activity studies of fluoroketone inhibitors of alpha-lytic protease and human leukocyte elastase.
    Govardhan CP; Abeles RH
    Arch Biochem Biophys; 1990 Jul; 280(1):137-46. PubMed ID: 2353815
    [TBL] [Abstract][Full Text] [Related]  

  • 18. Azetidine-2,4-diones (4-oxo-beta-lactams) as scaffolds for designing elastase inhibitors.
    Mulchande J; Guedes RC; Tsang WY; Page MI; Moreira R; Iley J
    J Med Chem; 2008 Mar; 51(6):1783-90. PubMed ID: 18290604
    [TBL] [Abstract][Full Text] [Related]  

  • 19. 3-Acylamino-azetidin-2-one as a novel class of cysteine proteases inhibitors.
    Zhou NE; Guo D; Thomas G; Reddy AV; Kaleta J; Purisima E; Menard R; Micetich RG; Singh R
    Bioorg Med Chem Lett; 2003 Jan; 13(1):139-41. PubMed ID: 12467634
    [TBL] [Abstract][Full Text] [Related]  

  • 20. Orally active beta-lactam inhibitors of human leukocyte elastase-1. Activity of 3,3-diethyl-2-azetidinones.
    Shah SK; Dorn CP; Finke PE; Hale JJ; Hagmann WK; Brause KA; Chandler GO; Kissinger AL; Ashe BM; Weston H
    J Med Chem; 1992 Oct; 35(21):3745-54. PubMed ID: 1433189
    [TBL] [Abstract][Full Text] [Related]  

    [Next]    [New Search]
    of 7.