These tools will no longer be maintained as of December 31, 2024. Archived website can be found here. PubMed4Hh GitHub repository can be found here. Contact NLM Customer Service if you have questions.


BIOMARKERS

Molecular Biopsy of Human Tumors

- a resource for Precision Medicine *

105 related articles for article (PubMed ID: 11073597)

  • 1. Conformational studies on (17alpha,20Z)-21-(X-Phenyl)-19-norpregna-1, 3,5(10),20-tetraene-3,17beta-diols using 1D and 2D NMR spectroscopy and GIAO calculations of (13)C shieldings.
    Sebag AB; Friel CJ; Hanson RN; Forsyth DA
    J Org Chem; 2000 Nov; 65(23):7902-12. PubMed ID: 11073597
    [TBL] [Abstract][Full Text] [Related]  

  • 2. Synthesis and evaluation of 17alpha-20E-21-(4-substituted phenyl)-19-norpregna-1,3,5(10),20-tetraene-3,17beta-diols as probes for the estrogen receptor alpha hormone binding domain.
    Hanson RN; Lee CY; Friel CJ; Dilis R; Hughes A; DeSombre ER
    J Med Chem; 2003 Jul; 46(14):2865-76. PubMed ID: 12825929
    [TBL] [Abstract][Full Text] [Related]  

  • 3. Synthesis and evaluation of (17alpha,20Z)-21-(4-substituted-phenyl)-19-norpregna-1,3,5(10),20-tetraene-3,17beta-diols as ligands for the estrogen receptor-alpha hormone binding domain: comparison with 20E-isomers.
    Hanson RN; Friel CJ; Dilis R; Hughes A; DeSombre ER
    J Med Chem; 2005 Jun; 48(13):4300-11. PubMed ID: 15974584
    [TBL] [Abstract][Full Text] [Related]  

  • 4. Evaluation of 17alpha-E-(trifluoromethylphenyl)vinyl estradiols as novel estrogen receptor ligands.
    Hanson RN; Lee CY; Friel C; Hughes A; DeSombre ER
    Steroids; 2003 Feb; 68(2):143-8. PubMed ID: 12606005
    [TBL] [Abstract][Full Text] [Related]  

  • 5. Synthesis and evaluation of 11beta-substituted 21-chloro/iodo-(17alpha,20E/Z)-19-norpregna-1,3,5(10),20-te traene-3, 17beta-diols: high-affinity ligands for the estrogen receptor.
    Hanson RN; Napolitano E; Fiaschi R
    J Med Chem; 1998 Nov; 41(24):4686-92. PubMed ID: 9822539
    [TBL] [Abstract][Full Text] [Related]  

  • 6. Synthesis and estrogen receptor binding of (17 alpha, 20E)- and (17 alpha, 20Z)-21-phenylthio- and 21-phenylseleno-19-norpregna-1,3,5(10),20-tetraene-3,17 beta-diols.
    Napolitano E; Fiaschi R; Herman LW; Hanson RN
    Steroids; 1996 Jun; 61(6):384-9. PubMed ID: 8776802
    [TBL] [Abstract][Full Text] [Related]  

  • 7. Stereochemical probes for the estrogen receptor: synthesis and receptor binding of (17 alpha,20E/Z)-21-phenyl-19-norpregna-1,3,5(10), 20-tetraene-3,17 beta-diols.
    Hanson RN; Herman LW; Fiaschi R; Napolitano E
    Steroids; 1996 Dec; 61(12):718-22. PubMed ID: 8987141
    [TBL] [Abstract][Full Text] [Related]  

  • 8. Structure-activity relationships of estrogenic ligands: synthesis and evaluation of (17 alpha, 20E)- and (17 alpha, 20Z)-21-halo-19-norpregna-1,3,5(10),20-tetraene-3,17 beta-diols.
    Napolitano E; Fiaschi R; Hanson RN
    J Med Chem; 1991 Sep; 34(9):2754-9. PubMed ID: 1895295
    [TBL] [Abstract][Full Text] [Related]  

  • 9. Synthesis and biological properties of 7alpha-cyano derivatives of the (17alpha,20E/Z)-[125I]iodovinyl- and 16alpha-[125I]iodo-estradiols.
    Ali H; Rousseau J; Paquette B; Dubé C; Marko B; van Lier JE
    Steroids; 2003 Dec; 68(14):1189-200. PubMed ID: 14643881
    [TBL] [Abstract][Full Text] [Related]  

  • 10. Synthesis, receptor binding, and tissue distribution of 7 alpha- and 11 beta-substituted (17 alpha,20E)- and (17 alpha,20Z)-21-[125I]iodo-19-norpregna-1,3,5(10),20-tetraene-3,17-diols.
    Ali H; Rousseau J; Ghaffari MA; van Lier JE
    J Med Chem; 1991 Feb; 34(2):854-60. PubMed ID: 1995909
    [TBL] [Abstract][Full Text] [Related]  

  • 11. Synthesis and evaluation of 17α-E-20-(heteroaryl)norpregn-1,3,5(10),20 tetraene-3,17β-diols [17α-(heteroaryl)vinyl estradiols] as ligands for the estrogen receptor-α ligand binding domain (ERα-LBD).
    Olmsted SL; Tongcharoensirikul P; McCaskill E; Gandiaga K; Labaree D; Hochberg RB; Hanson RN
    Bioorg Med Chem Lett; 2012 Jan; 22(2):977-9. PubMed ID: 22178552
    [TBL] [Abstract][Full Text] [Related]  

  • 12. Synthesis of 3-phenyl-4-phenylvinyl benzopyranones and the corresponding 2,2-dimethyl-benzopyrans with structural similarity to estradiol, as estrogen receptor ligands.
    Gupta A; Raghunandan R; Kumar A; Maulik PR; Dwivedyc A; Keshri G; Singh MM; Ray S
    Med Chem; 2007 Sep; 3(5):446-54. PubMed ID: 17897069
    [TBL] [Abstract][Full Text] [Related]  

  • 13. Synthesis and evaluation of isomeric (17alpha,20E)-11beta-methoxy-21-(trifluoromethylphenyl)-19-norpregna-1,3,5(10),20-tetraene-3,17beta-diols as ERalpha-hormone binding domain ligands: effect of the methoxy group on receptor binding and uterotrophic growth.
    Hanson RN; Tongcharoensirikul P; Dilis R; Hughes A; Desombre ER
    J Med Chem; 2007 Feb; 50(3):472-9. PubMed ID: 17266199
    [TBL] [Abstract][Full Text] [Related]  

  • 14. The novel estrogen 17alpha-20Z-21-[(4-amino)phenyl]-19-norpregna-1,3,5(10),20-tetraene-3,17beta-diol induces apoptosis in prostate cancer cell lines at nanomolar concentrations in vitro.
    Mobley JA; L'Esperance JO; Wu M; Friel CJ; Hanson RH; Ho SM
    Mol Cancer Ther; 2004 May; 3(5):587-95. PubMed ID: 15141016
    [TBL] [Abstract][Full Text] [Related]  

  • 15. Synthesis of benzoylbenzamide derivatives of 17α-E-vinyl estradiol and evaluation as ligands for the estrogen receptor-α ligand binding domain.
    Hanson RN; McCaskill E; Hua E; Tongcharoensirikul P; Dilis R; Silver JL; Coulther TA; Ondrechen MJ; Labaree D; Hochberg RB
    Steroids; 2019 Apr; 144():15-20. PubMed ID: 30738075
    [TBL] [Abstract][Full Text] [Related]  

  • 16. Synthesis and evaluation of 17α-(dimethylphenyl)vinyl estradiols as probes of the estrogen receptor-α ligand binding domain.
    Hanson RN; McCaskill E; Tongcharoensirikul P; Dilis R; Labaree D; Hochberg RB
    Steroids; 2012 Apr; 77(5):471-6. PubMed ID: 22273809
    [TBL] [Abstract][Full Text] [Related]  

  • 17. Estrogen receptor binding characteristics of 1,11 beta-ethanoestradiol: effect of a 1,11 beta-bridge on steroidal estrogen.
    Napolitano E; Fiaschi R; Hanson RN
    J Steroid Biochem Mol Biol; 1990 Oct; 37(2):295-300. PubMed ID: 2268562
    [TBL] [Abstract][Full Text] [Related]  

  • 18. Synthesis, receptor binding, and tissue distribution of (17 alpha,20E)- and (17 alpha,20Z)-21-[125I]iodo-19-norpregna-1,3,5(10), 20-tetraene-3,17-diol .
    Ali H; Rousseau J; Ghaffari MA; van Lier JE
    J Med Chem; 1988 Oct; 31(10):1946-50. PubMed ID: 3172127
    [TBL] [Abstract][Full Text] [Related]  

  • 19. Novel 7α-alkoxy-17α-(4'-halophenylethynyl)estradiols as potential SPECT/PET imaging agents for estrogen receptor expressing tumours: synthesis and binding affinity evaluation.
    Neto C; Oliveira MC; Gano L; Marques F; Yasuda T; Thiemann T; Kniess T; Santos I
    Steroids; 2012 Sep; 77(11):1123-32. PubMed ID: 22633985
    [TBL] [Abstract][Full Text] [Related]  

  • 20. Impact of estradiol structural modifications (18-methyl and/or 17-hydroxy inversion of configuration) on the in vitro and in vivo estrogenic activity.
    Ayan D; Roy J; Maltais R; Poirier D
    J Steroid Biochem Mol Biol; 2011 Nov; 127(3-5):324-30. PubMed ID: 21827856
    [TBL] [Abstract][Full Text] [Related]  

    [Next]    [New Search]
    of 6.