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9. Analgesic and anti-inflammatory effects of A-286501, a novel orally active adenosine kinase inhibitor. Jarvis MF; Yu H; McGaraughty S; Wismer CT; Mikusa J; Zhu C; Chu K; Kohlhaas K; Cowart M; Lee CH; Stewart AO; Cox BF; Polakowski J; Kowaluk EA Pain; 2002 Mar; 96(1-2):107-18. PubMed ID: 11932067 [TBL] [Abstract][Full Text] [Related]
10. Comparison of the ability of adenosine kinase inhibitors and adenosine receptor agonists to attenuate thermal hyperalgesia and reduce motor performance in rats. Jarvis MF; Mikusa J; Chu KL; Wismer CT; Honore P; Kowaluk EA; McGaraughty S Pharmacol Biochem Behav; 2002 Oct; 73(3):573-81. PubMed ID: 12151032 [TBL] [Abstract][Full Text] [Related]
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13. Discovery and optimization of 2-aryl oxazolo-pyrimidines as adenosine kinase inhibitors using liquid phase parallel synthesis. Bauser M; Delapierre G; Hauswald M; Flessner T; D'Urso D; Hermann A; Beyreuther B; De Vry J; Spreyer P; Reissmüller E; Meier H Bioorg Med Chem Lett; 2004 Apr; 14(8):1997-2000. PubMed ID: 15050645 [TBL] [Abstract][Full Text] [Related]
14. ABT-702 (4-amino-5-(3-bromophenyl)-7-(6-morpholino-pyridin- 3-yl)pyrido[2,3-d]pyrimidine), a novel orally effective adenosine kinase inhibitor with analgesic and anti-inflammatory properties. II. In vivo characterization in the rat. Kowaluk EA; Mikusa J; Wismer CT; Zhu CZ; Schweitzer E; Lynch JJ; Lee CH; Jiang M; Bhagwat SS; Gomtsyan A; McKie J; Cox BF; Polakowski J; Reinhart G; Williams M; Jarvis MF J Pharmacol Exp Ther; 2000 Dec; 295(3):1165-74. PubMed ID: 11082454 [TBL] [Abstract][Full Text] [Related]
15. A-134974: a novel adenosine kinase inhibitor, relieves tactile allodynia via spinal sites of action in peripheral nerve injured rats. Zhu CZ; Mikusa J; Chu KL; Cowart M; Kowaluk EA; Jarvis MF; McGaraughty S Brain Res; 2001 Jun; 905(1-2):104-10. PubMed ID: 11423084 [TBL] [Abstract][Full Text] [Related]
16. Discovery of 4-amino-5-(3-bromophenyl)-7-(6-morpholino-pyridin-3-yl)pyrido[2,3-d]pyrimidine, an orally active, non-nucleoside adenosine kinase inhibitor. Lee CH; Jiang M; Cowart M; Gfesser G; Perner R; Kim KH; Gu YG; Williams M; Jarvis MF; Kowaluk EA; Stewart AO; Bhagwat SS J Med Chem; 2001 Jun; 44(13):2133-8. PubMed ID: 11405650 [TBL] [Abstract][Full Text] [Related]
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20. ABT-702 (4-amino-5-(3-bromophenyl)-7-(6-morpholinopyridin-3-yl)pyrido[2, 3-d]pyrimidine), a novel orally effective adenosine kinase inhibitor with analgesic and anti-inflammatory properties: I. In vitro characterization and acute antinociceptive effects in the mouse. Jarvis MF; Yu H; Kohlhaas K; Alexander K; Lee CH; Jiang M; Bhagwat SS; Williams M; Kowaluk EA J Pharmacol Exp Ther; 2000 Dec; 295(3):1156-64. PubMed ID: 11082453 [TBL] [Abstract][Full Text] [Related] [Next] [New Search]