112 related articles for article (PubMed ID: 11164381)
1. Stereochemistry and molecular pharmacology of (S)-thio-ATPA, a new potent and selective GluR5 agonist.
Stensbøl TB; Jensen HS; Nielsen B; Johansen TN; Egebjerg J; Frydenvang K; Krogsgaard-Larsen P
Eur J Pharmacol; 2001 Jan; 411(3):245-53. PubMed ID: 11164381
[TBL] [Abstract][Full Text] [Related]
2. Resolution, absolute stereochemistry and molecular pharmacology of the enantiomers of ATPA.
Stensbøl TB; Borre L; Johansen TN; Egebjerg J; Madsen U; Ebert B; Krogsgaard-Larsen P
Eur J Pharmacol; 1999 Sep; 380(2-3):153-62. PubMed ID: 10513575
[TBL] [Abstract][Full Text] [Related]
3. (S)-2-Amino-3-(3-hydroxy-7,8-dihydro-6H-cyclohepta[d]isoxazol-4-yl)propionic acid, a potent and selective agonist at the GluR5 subtype of ionotropic glutamate receptors. Synthesis, modeling, and molecular pharmacology.
Brehm L; Greenwood JR; Hansen KB; Nielsen B; Egebjerg J; Stensbøl TB; Bräuner-Osborne H; Sløk FA; Kronborg TT; Krogsgaard-Larsen P
J Med Chem; 2003 Apr; 46(8):1350-8. PubMed ID: 12672235
[TBL] [Abstract][Full Text] [Related]
4. Resolution, configurational assignment, and enantiopharmacology of 2-amino-3-[3-hydroxy-5-(2-methyl-2H- tetrazol-5-yl)isoxazol-4-yl]propionic acid, a potent GluR3- and GluR4-preferring AMPA receptor agonist.
Vogensen SB; Jensen HS; Stensbøl TB; Frydenvang K; Bang-Andersen B; Johansen TN; Egebjerg J; Krogsgaard-Larsen P
Chirality; 2000 Nov; 12(10):705-13. PubMed ID: 11054828
[TBL] [Abstract][Full Text] [Related]
5. Excitatory amino acid receptor ligands: resolution, absolute stereochemistry, and enantiopharmacology of 2-amino-3-(4-butyl-3-hydroxyisoxazol-5-yl)propionic acid.
Johansen TN; Ebert B; Bräuner-Osborne H; Didriksen M; Christensen IT; Søby KK; Madsen U; Krogsgaard-Larsen P; Brehm L
J Med Chem; 1998 Mar; 41(6):930-9. PubMed ID: 9526567
[TBL] [Abstract][Full Text] [Related]
6. Resolution, absolute stereochemistry, and enantiopharmacology of the GluR1-4 and GluR5 antagonist 2-amino-3-[5-tert-butyl-3-(phosphonomethoxy)-4-isoxazolyl]propionic acid.
Møller EH; Egebjerg J; Brehm L; Stensbøl TB; Johansen TN; Madsen U; Krogsgaard-Larsen P
Chirality; 1999; 11(10):752-9. PubMed ID: 10561704
[TBL] [Abstract][Full Text] [Related]
7. Tetrazolyl isoxazole amino acids as ionotropic glutamate receptor antagonists: synthesis, modelling and molecular pharmacology.
Frølund B; Greenwood JR; Holm MM; Egebjerg J; Madsen U; Nielsen B; Bräuner-Osborne H; Stensbøl TB; Krogsgaard-Larsen P
Bioorg Med Chem; 2005 Sep; 13(18):5391-8. PubMed ID: 16043357
[TBL] [Abstract][Full Text] [Related]
8. Pharmacology and toxicology of ATOA, an AMPA receptor antagonist and a partial agonist at GluR5 receptors.
Wahl P; Frandsen A; Madsen U; Schousboe A; Krogsgaard-Larsen P
Neuropharmacology; 1998; 37(10-11):1205-10. PubMed ID: 9849658
[TBL] [Abstract][Full Text] [Related]
9. AMPA receptor agonists: resolution, configurational assignment, and pharmacology of (+)-(S)- and (-)-(R)-2-amino-3-[3-hydroxy-5-(2-pyridyl)-isoxazol-4-yl]-propionic acid (2-Py-AMPA).
Johansen TN; Ebert B; Falch E; Krogsgaard-Larsen P
Chirality; 1997; 9(3):274-80. PubMed ID: 9176992
[TBL] [Abstract][Full Text] [Related]
10. Heteroaryl analogues of AMPA. 2. Synthesis, absolute stereochemistry, photochemistry, and structure-activity relationships.
Falch E; Brehm L; Mikkelsen I; Johansen TN; Skjaerbaek N; Nielsen B; Stensbøl TB; Ebert B; Krogsgaard-Larsen P
J Med Chem; 1998 Jul; 41(14):2513-23. PubMed ID: 9651156
[TBL] [Abstract][Full Text] [Related]
11. Structural determinants of agonist-specific kinetics at the ionotropic glutamate receptor 2.
Holm MM; Lunn ML; Traynelis SF; Kastrup JS; Egebjerg J
Proc Natl Acad Sci U S A; 2005 Aug; 102(34):12053-8. PubMed ID: 16099829
[TBL] [Abstract][Full Text] [Related]
12. AMPA receptor agonists: synthesis, protolytic properties, and pharmacology of 3-isothiazolol bioisosteres of glutamic acid.
Matzen L; Engesgaard A; Ebert B; Didriksen M; Frølund B; Krogsgaard-Larsen P; Jaroszewski JW
J Med Chem; 1997 Feb; 40(4):520-7. PubMed ID: 9046343
[TBL] [Abstract][Full Text] [Related]
13. Synthesis, theoretical and structural analyses, and enantiopharmacology of 3-carboxy homologs of AMPA.
Brehm L; Greenwood JR; Sløk FA; Holm MM; Nielsen B; Geneser U; Stensbøl TB; Bräuner-Osborne H; Begtrup M; Egebjerg J; Krogsgaard-Larsen P
Chirality; 2004 Aug; 16(7):452-66. PubMed ID: 15236343
[TBL] [Abstract][Full Text] [Related]
14. Resolution, configurational assignment, and enantiopharmacology at glutamate receptors of 2-amino-3-(3-carboxy-5-methyl-4-isoxazolyl)propionic acid (ACPA) and demethyl-ACPA.
Johansen TN; Stensbøl TB; Nielsen B; Vogensen SB; Frydenvang K; Sløk FA; Bräüner-Osborne H; Madsen U; Krogsgaard-Larsen P
Chirality; 2001; 13(9):523-32. PubMed ID: 11579444
[TBL] [Abstract][Full Text] [Related]
15. The selective activation of the glutamate receptor GluR5 by ATPA is controlled by serine 741.
Nielsen MM; Liljefors T; Krogsgaard-Larsen P; Egebjerg J
Mol Pharmacol; 2003 Jan; 63(1):19-25. PubMed ID: 12488532
[TBL] [Abstract][Full Text] [Related]
16. The glutamate receptor GluR5 agonist (S)-2-amino-3-(3-hydroxy-7,8-dihydro-6H-cyclohepta[d]isoxazol-4-yl)propionic acid and the 8-methyl analogue: synthesis, molecular pharmacology, and biostructural characterization.
Clausen RP; Naur P; Kristensen AS; Greenwood JR; Strange M; Bräuner-Osborne H; Jensen AA; Nielsen AS; Geneser U; Ringgaard LM; Nielsen B; Pickering DS; Brehm L; Gajhede M; Krogsgaard-Larsen P; Kastrup JS
J Med Chem; 2009 Aug; 52(15):4911-22. PubMed ID: 19588945
[TBL] [Abstract][Full Text] [Related]
17. Comparison of excitotoxic profiles of ATPA, AMPA, KA and NMDA in organotypic hippocampal slice cultures.
Kristensen BW; Noraberg J; Zimmer J
Brain Res; 2001 Oct; 917(1):21-44. PubMed ID: 11602227
[TBL] [Abstract][Full Text] [Related]
18. Molecular pharmacology of the AMPA agonist, (S)-2-amino-3-(3-hydroxy-5-phenyl-4-isoxazolyl)propionic acid [(S)-APPA] and the AMPA antagonist, (R)-APPA.
Ebert B; Madsen U; Lund TM; Lenz SM; Krogsgaard-Larsen P
Neurochem Int; 1994 Jun; 24(6):507-15. PubMed ID: 7526921
[TBL] [Abstract][Full Text] [Related]
19. Pharmacological characterization of a GluR6 kainate receptor in cultured hippocampal neurons.
Bleakman D; Ogden AM; Ornstein PL; Hoo K
Eur J Pharmacol; 1999 Aug; 378(3):331-7. PubMed ID: 10493110
[TBL] [Abstract][Full Text] [Related]
20. Functional partial agonism at ionotropic excitatory amino acid receptors.
Ebert B; Madsen U; Søby KK; Krogsgaard-Larsen P
Neurochem Int; 1996 Sep; 29(3):309-16. PubMed ID: 8885290
[TBL] [Abstract][Full Text] [Related]
[Next] [New Search]
