These tools will no longer be maintained as of December 31, 2024. Archived website can be found here. PubMed4Hh GitHub repository can be found here. Contact NLM Customer Service if you have questions.


BIOMARKERS

Molecular Biopsy of Human Tumors

- a resource for Precision Medicine *

125 related articles for article (PubMed ID: 11206453)

  • 21. Characterization of the mechanism of anticonvulsant activity for a selected set of putative AMPA receptor antagonists.
    Grasso S; Micale N; Zappalà M; Galli A; Costagli C; Menniti FS; De Micheli C
    Bioorg Med Chem Lett; 2003 Feb; 13(3):443-6. PubMed ID: 12565947
    [TBL] [Abstract][Full Text] [Related]  

  • 22. Structural investigation of the 7-chloro-3-hydroxy-1H-quinazoline-2,4-dione scaffold to obtain AMPA and kainate receptor selective antagonists. Synthesis, pharmacological, and molecular modeling studies.
    Colotta V; Catarzi D; Varano F; Lenzi O; Filacchioni G; Costagli C; Galli A; Ghelardini C; Galeotti N; Gratteri P; Sgrignani J; Deflorian F; Moro S
    J Med Chem; 2006 Oct; 49(20):6015-26. PubMed ID: 17004715
    [TBL] [Abstract][Full Text] [Related]  

  • 23. Synthesis and anticonvulsant evaluation of N-substituted isoquinoline AMPA receptor antagonists.
    Gitto R; De Luca L; Pagano B; Citraro R; De Sarro G; Costa L; Ciranna L; Chimirri A
    Bioorg Med Chem; 2008 Mar; 16(5):2379-84. PubMed ID: 18077172
    [TBL] [Abstract][Full Text] [Related]  

  • 24. Design and synthesis of some new quinazolin-4-(3H)-ones as anticonvulsant and antidepressant agents.
    Amir M; Ali I; Hassan MZ
    Arch Pharm Res; 2013 Jan; 36(1):61-8. PubMed ID: 23325491
    [TBL] [Abstract][Full Text] [Related]  

  • 25. Design and Synthesis of Selurampanel, a Novel Orally Active and Competitive AMPA Receptor Antagonist.
    Orain D; Tasdelen E; Haessig S; Koller M; Picard A; Dubois C; Lingenhoehl K; Desrayaud S; Floersheim P; Carcache D; Urwyler S; Kallen J; Mattes H
    ChemMedChem; 2017 Feb; 12(3):197-201. PubMed ID: 27863026
    [TBL] [Abstract][Full Text] [Related]  

  • 26. Synthesis and anticonvulsant activity of novel and potent 6,7-methylenedioxyphthalazin-1(2H)-ones.
    Grasso S; De Sarro G; De Sarro A; Micale N; Zappalà M; Puja G; Baraldi M; De Micheli C
    J Med Chem; 2000 Jul; 43(15):2851-9. PubMed ID: 10956193
    [TBL] [Abstract][Full Text] [Related]  

  • 27. New 7,8-ethylenedioxy-2,3-benzodiazepines as noncompetitive AMPA receptor antagonists.
    Zappalà M; Pellicanò A; Micale N; Menniti FS; Ferreri G; De Sarro G; Grasso S; De Micheli C
    Bioorg Med Chem Lett; 2006 Jan; 16(1):167-70. PubMed ID: 16216501
    [TBL] [Abstract][Full Text] [Related]  

  • 28. Synthesis and evaluation of pharmacological and pharmacokinetic properties of 11H-[1,2,4]triazolo[4,5-c][2,3]benzodiazepin-3(2H)-ones.
    Zappalà M; Gitto R; Bevacqua F; Quartarone S; Chimirri A; Rizzo M; De Sarro G; De Sarro A
    J Med Chem; 2000 Dec; 43(25):4834-9. PubMed ID: 11123993
    [TBL] [Abstract][Full Text] [Related]  

  • 29. Synthesis, chiral resolution, and enantiopharmacology of a potent 2,3-benzodiazepine derivative as noncompetitive AMPA receptor antagonist.
    Zappalà M; Postorino G; Micale N; Caccamese S; Parrinello N; Grazioso G; Roda G; Menniti FS; De Sarro G; Grasso S
    J Med Chem; 2006 Jan; 49(2):575-81. PubMed ID: 16420043
    [TBL] [Abstract][Full Text] [Related]  

  • 30. Excitatory amino acid neurotransmission through both NMDA and non-NMDA receptors is involved in the anticonvulsant activity of felbamate in DBA/2 mice.
    De Sarro G; Ongini E; Bertorelli R; Aguglia U; De Sarro A
    Eur J Pharmacol; 1994 Sep; 262(1-2):11-9. PubMed ID: 7529182
    [TBL] [Abstract][Full Text] [Related]  

  • 31. 1-Aryl-3,5-dihydro-4H-2,3-benzodiazepin-4-ones: novel AMPA receptor antagonists.
    Chimirri A; De Sarro G; De Sarro A; Gitto R; Grasso S; Quartarone S; Zappalà M; Giusti P; Libri V; Constanti A; Chapman AG
    J Med Chem; 1997 Apr; 40(8):1258-69. PubMed ID: 9111300
    [TBL] [Abstract][Full Text] [Related]  

  • 32. 9-Carboxymethyl-5H,10H-imidazo[1,2-a]indeno[1,2-e]pyrazin-4-one-2-carbocylic acid (RPR117824): selective anticonvulsive and neuroprotective AMPA antagonist.
    Mignani S; Bohme GA; Birraux G; Boireau A; Jimonet P; Damour D; Genevois-Borella A; Debono MW; Pratt J; Vuilhorgne M; Wahl F; Stutzmann JM
    Bioorg Med Chem; 2002 May; 10(5):1627-37. PubMed ID: 11886824
    [TBL] [Abstract][Full Text] [Related]  

  • 33. A new pyrrolyl-quinoxalinedione series of non-NMDA glutamate receptor antagonists: pharmacological characterization and comparison with NBQX and valproate in the kindling model of epilepsy.
    Löscher W; Lehmann H; Behl B; Seemann D; Teschendorf HJ; Hofmann HP; Lubisch W; Höger T; Lemaire HG; Gross G
    Eur J Neurosci; 1999 Jan; 11(1):250-62. PubMed ID: 9987029
    [TBL] [Abstract][Full Text] [Related]  

  • 34. Synthesis and anticonvulsant activity of N-3 substituted 2,3-benzodiazepines.
    Quartarone S; Caruso R; Orlando V; Russo E; De Sarro G; Chimirri A
    Farmaco; 2004 May; 59(5):353-8. PubMed ID: 15120314
    [TBL] [Abstract][Full Text] [Related]  

  • 35. Design and synthesis of enantiomers of 3,5-dinitro-o-tyrosine: alpha-amino-3-hydroxy-5-methyl-4-isoxazolepropanoic acid (AMPA) receptor antagonists.
    Sun G; Slavica M; Uretsky NJ; Wallace LJ; Shams G; Weinstein DM; Miller JC; Miller DD
    J Med Chem; 1998 Mar; 41(7):1034-41. PubMed ID: 9544203
    [TBL] [Abstract][Full Text] [Related]  

  • 36. Synthesis of 7,8-(methylenedioxy)-1-phenyl-3,5-dihydro-4H-2, 3-benzodiazepin-4-ones as novel and potent noncompetitive AMPA receptor antagonists.
    Wang Y; Konkoy CS; Ilyin VI; Vanover KE; Carter RB; Weber E; Keana JF; Woodward RM; Cai SX
    J Med Chem; 1998 Jul; 41(14):2621-5. PubMed ID: 9651166
    [TBL] [Abstract][Full Text] [Related]  

  • 37. Novel potent anticonvulsant agent containing a tetrahydroisoquinoline skeleton.
    Gitto R; Caruso R; Pagano B; De Luca L; Citraro R; Russo E; De Sarro G; Chimirri A
    J Med Chem; 2006 Sep; 49(18):5618-22. PubMed ID: 16942035
    [TBL] [Abstract][Full Text] [Related]  

  • 38. Design, synthesis and anticonvulsant evaluation of N-(benzo[d]thiazol-2-ylcarbamoyl)-2-methyl-4-oxoquinazoline-3(4H)-carbothioamide derivatives: a hybrid pharmacophore approach.
    Malik S; Bahare RS; Khan SA
    Eur J Med Chem; 2013 Sep; 67():1-13. PubMed ID: 23831504
    [TBL] [Abstract][Full Text] [Related]  

  • 39. Synthesis and evaluation of pharmacological properties of novel annelated 2,3-benzodiazepine derivatives.
    Gitto R; Orlando V; Quartarone S; De Sarro G; De Sarro A; Russo E; Ferreri G; Chimirri A
    J Med Chem; 2003 Aug; 46(17):3758-61. PubMed ID: 12904081
    [TBL] [Abstract][Full Text] [Related]  

  • 40. 8-Methylureido-10-amino-10-methyl-imidazo[1,2-a]indeno[1,2-e] pyrazine-4-ones: highly in vivo potent and selective AMPA receptor antagonists.
    Jimonet P; Chevé M; Bohme GA; Boireau A; Damour D; Debono MW; Genevois-Borella A; Imperato A; Pratt J; Randle JC; Ribeill Y; Stutzmann JM; Vuilhorgne M; Mignani S
    Bioorg Med Chem; 2000 Aug; 8(8):2211-7. PubMed ID: 11003165
    [TBL] [Abstract][Full Text] [Related]  

    [Previous]   [Next]    [New Search]
    of 7.