118 related articles for article (PubMed ID: 11259030)
1. Convenient synthesis and diversification of dehydroalaninyl phosphinic peptide analogues.
Matziari M; Georgiadis D; Dive V; Yiotakis A
Org Lett; 2001 Mar; 3(5):659-62. PubMed ID: 11259030
[TBL] [Abstract][Full Text] [Related]
2. Efficient synthesis of Fmoc-protected phosphinic pseudodipeptides: Building blocks for the synthesis of matrix metalloproteinase inhibitors.
Bhowmick M; Sappidi RR; Fields GB; Lepore SD
Biopolymers; 2011; 96(1):1-3. PubMed ID: 20225219
[TBL] [Abstract][Full Text] [Related]
3. A synthetic method for diversification of the P1' substituent in phosphinic dipeptides as a tool for exploration of the specificity of the S1' binding pockets of leucine aminopeptidases.
Vassiliou S; Xeilari M; Yiotakis A; Grembecka J; Pawełczak M; Kafarski P; Mucha A
Bioorg Med Chem; 2007 May; 15(9):3187-200. PubMed ID: 17337192
[TBL] [Abstract][Full Text] [Related]
4. Synthesis of a Gln-Phe hydroxy-ethylene dipeptide isostere.
Haug BE; Rich DH
Org Lett; 2004 Dec; 6(25):4783-6. PubMed ID: 15575685
[TBL] [Abstract][Full Text] [Related]
5. Design, synthesis, and evaluation of matrix metalloprotease inhibitors bearing cyclopropane-derived peptidomimetics as P1' and P2' replacements.
Reichelt A; Gaul C; Frey RR; Kennedy A; Martin SF
J Org Chem; 2002 Jun; 67(12):4062-75. PubMed ID: 12054939
[TBL] [Abstract][Full Text] [Related]
6. Synthesis of 2-amino-3-fluoroacrylic acid containing peptides.
Zhou H; van der Donk WA
Org Lett; 2001 Feb; 3(4):593-6. PubMed ID: 11178833
[TBL] [Abstract][Full Text] [Related]
7. Synthesis and modifications of phosphinic dipeptide analogues.
Mucha A
Molecules; 2012 Nov; 17(11):13530-68. PubMed ID: 23154272
[TBL] [Abstract][Full Text] [Related]
8. Late-Stage Diversification of Phosphinic Dehydroalanine Pseudopeptides Based on a Giese-Type Radical C-Alkylation Strategy.
Voreakos K; Devel L; Georgiadis D
Org Lett; 2019 Jun; 21(12):4397-4401. PubMed ID: 30933530
[TBL] [Abstract][Full Text] [Related]
9. Synthesis of novel N-phosphonoalkyl dipeptide inhibitors of human collagenase.
Bird J; De Mello RC; Harper GP; Hunter DJ; Karran EH; Markwell RE; Miles-Williams AJ; Rahman SS; Ward RW
J Med Chem; 1994 Jan; 37(1):158-69. PubMed ID: 8289190
[TBL] [Abstract][Full Text] [Related]
10. Diastereoselective synthesis of alpha,beta'-disubstituted aminomethyl(2-carboxyethyl)phosphinates as phosphinyl dipeptide isosteres.
Yamagishi T; Ichikawa H; Haruki T; Yokomatsu T
Org Lett; 2008 Oct; 10(19):4347-50. PubMed ID: 18781768
[TBL] [Abstract][Full Text] [Related]
11. Inhibition of stromelysin-1 (MMP-3) by P1'-biphenylylethyl carboxyalkyl dipeptides.
Esser CK; Bugianesi RL; Caldwell CG; Chapman KT; Durette PL; Girotra NN; Kopka IE; Lanza TJ; Levorse DA; MacCoss M; Owens KA; Ponpipom MM; Simeone JP; Harrison RK; Niedzwiecki L; Becker JW; Marcy AI; Axel MG; Christen AJ; McDonnell J; Moore VL; Olszewski JM; Saphos C; Visco DM; Hagmann WK
J Med Chem; 1997 Mar; 40(6):1026-40. PubMed ID: 9083493
[TBL] [Abstract][Full Text] [Related]
12. Diastereoselective solution and multipin-based combinatorial array synthesis of a novel class of potent phosphinic metalloprotease inhibitors.
Makaritis A; Georgiadis D; Dive V; Yiotakis A
Chemistry; 2003 May; 9(9):2079-94. PubMed ID: 12740857
[TBL] [Abstract][Full Text] [Related]
13. The most potent organophosphorus inhibitors of leucine aminopeptidase. Structure-based design, chemistry, and activity.
Grembecka J; Mucha A; Cierpicki T; Kafarski P
J Med Chem; 2003 Jun; 46(13):2641-55. PubMed ID: 12801228
[TBL] [Abstract][Full Text] [Related]
14. Synthesis of protected enantiopure (R) and (S)-α-trifluoromethylalanine containing dipeptide building blocks ready to use for solid phase peptide synthesis.
Devillers E; Pytkowicz J; Chelain E; Brigaud T
Amino Acids; 2016 Jun; 48(6):1457-68. PubMed ID: 26920748
[TBL] [Abstract][Full Text] [Related]
15. Ketomethylene analogues of phosphoryl dipeptides related to phosphoramidon: synthesis and inhibition of proteases.
Gómez-Monterrey I; González Muñiz R; Pérez-Martín C; López de Ceballos M; Del Río J; García-López MT
Arch Pharm (Weinheim); 1992 May; 325(5):261-5. PubMed ID: 1524467
[TBL] [Abstract][Full Text] [Related]
16. Synthesis and structural study of cyclic 5-aminovaleric acid-linked beta-Ala-beta-Ala dipeptides.
Mengel A; Reiser O; Aubé J
Bioorg Med Chem Lett; 2008 Nov; 18(22):5975-7. PubMed ID: 18682325
[TBL] [Abstract][Full Text] [Related]
17. Phosphinic peptide inhibitors of macrophage metalloelastase (MMP-12). Selectivity and mechanism of binding.
Schiødt CB; Buchardt J; Terp GE; Christensen U; Brink M; Berger Larsen Y; Meldal M; Foged NT
Curr Med Chem; 2001 Jul; 8(8):967-76. PubMed ID: 11375764
[TBL] [Abstract][Full Text] [Related]
18. Evaluation of P1'-diversified phosphinic peptides leads to the development of highly selective inhibitors of MMP-11.
Matziari M; Beau F; Cuniasse P; Dive V; Yiotakis A
J Med Chem; 2004 Jan; 47(2):325-36. PubMed ID: 14711305
[TBL] [Abstract][Full Text] [Related]
19. Practical Synthesis of Phosphinic Dipeptides by Tandem Esterification of Aminophosphinic and Acrylic Acids under Silylating Conditions.
Kokkala P; Voreakos K; Lelis A; Patiniotis K; Skoulikas N; Devel L; Ziotopoulou A; Kaloumenou E; Georgiadis D
Molecules; 2022 Feb; 27(4):. PubMed ID: 35209031
[TBL] [Abstract][Full Text] [Related]
20. Matrix metalloproteinase inhibitors: a structure-activity study.
Levy DE; Lapierre F; Liang W; Ye W; Lange CW; Li X; Grobelny D; Casabonne M; Tyrrell D; Holme K; Nadzan A; Galardy RE
J Med Chem; 1998 Jan; 41(2):199-223. PubMed ID: 9457244
[TBL] [Abstract][Full Text] [Related]
[Next] [New Search]
