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4. Conformationally constrained o-tolylpiperazine camphorsulfonamide oxytocin antagonists. Structural modifications that provide high receptor affinity and suggest a bioactive conformation. Williams PD; Ball RG; Clineschmidt BV; Culberson JC; Erb JM; Freidinger RM; Pawluczyk JM; Perlow DS; Pettibone DJ; Veber DF Bioorg Med Chem; 1994 Sep; 2(9):971-85. PubMed ID: 7712132 [TBL] [Abstract][Full Text] [Related]
5. Progress in the development of oxytocin antagonists for use in preterm labor. Williams PD; Bock MG; Evans BE; Freidinger RM; Pettibone DJ Adv Exp Med Biol; 1998; 449():473-9. PubMed ID: 10026841 [TBL] [Abstract][Full Text] [Related]
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8. Isosteric substitution of Asn5 in antagonists of oxytocin and vasopressin leads to highly selective and potent oxytocin and V1a receptor antagonists: new approaches for the design of potential tocolytics for preterm labor. Chan WY; Wo NC; Cheng LL; Manning M J Pharmacol Exp Ther; 1996 May; 277(2):999-1003. PubMed ID: 8627583 [TBL] [Abstract][Full Text] [Related]
11. 2,5-diketopiperazines as potent, selective, and orally bioavailable oxytocin antagonists. 3. Synthesis, pharmacokinetics, and in vivo potency. Borthwick AD; Davies DE; Exall AM; Hatley RJ; Hughes JA; Irving WR; Livermore DG; Sollis SL; Nerozzi F; Valko KL; Allen MJ; Perren M; Shabbir SS; Woollard PM; Price MA J Med Chem; 2006 Jul; 49(14):4159-70. PubMed ID: 16821776 [TBL] [Abstract][Full Text] [Related]
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13. Oxytocin antagonists with changes in the Asn5 position shed light on hormone-oxytocin receptor interactions. Hill PS; Chan WY; Hruby VJ Int J Pept Protein Res; 1991 Jul; 38(1):32-7. PubMed ID: 1657804 [TBL] [Abstract][Full Text] [Related]
14. In vivo activity of the potent oxytocin antagonist on uterine activity in the rat. Ahn TG; Han SJ; Cho YS; An TH; Pak SC; Flouret G In Vivo; 2004; 18(6):763-6. PubMed ID: 15646817 [TBL] [Abstract][Full Text] [Related]
15. Advances in the design of selective antagonists, potential tocolytics, and radioiodinated ligands for oxytocin receptors. Manning M; Cheng LL; Klis WA; Stoev S; Przybylski J; Bankowski K; Sawyer WH; Barberis C; Chan WY Adv Exp Med Biol; 1995; 395():559-83. PubMed ID: 8714021 [TBL] [Abstract][Full Text] [Related]
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17. The role of oxytocin receptors and vasopressin V1a receptors in uterine contractions in rats: implications for tocolytic therapy with oxytocin antagonists. Chan WY; Wo NC; Manning M Am J Obstet Gynecol; 1996 Nov; 175(5):1331-5. PubMed ID: 8942510 [TBL] [Abstract][Full Text] [Related]