195 related articles for article (PubMed ID: 12182657)
1. Diastereoselective synthesis of new psi[(E)-CH=CMe]- and psi[(Z)-CH=CMe]-type alkene dipeptide isosteres by organocopper reagents and application to conformationally restricted cyclic RGD peptidomimetics.
Oishi S; Kamano T; Niida A; Odagaki Y; Hamanaka N; Yamamoto M; Ajito K; Tamamura H; Otaka A; Fujii N
J Org Chem; 2002 Aug; 67(17):6162-73. PubMed ID: 12182657
[TBL] [Abstract][Full Text] [Related]
2. Regio- and stereoselective synthesis of (E)-alkene trans-Xaa-Pro dipeptide mimetics utilizing organocopper-mediated anti-S(N)2' reactions.
Otaka A; Katagiri F; Kinoshita T; Odagaki Y; Oishi S; Tamamura H; Hamanaka N; Fujii N
J Org Chem; 2002 Aug; 67(17):6152-61. PubMed ID: 12182656
[TBL] [Abstract][Full Text] [Related]
3. Diastereoselective synthesis of psi[(E)-CH=CMe]- and psi[(Z)-CH=CMe]-type dipeptide isosteres by organocopper-mediated anti-S(N)2' reaction.
Oishi S; Kamano T; Niida A; Odagaki Y; Tamamura H; Otaka A; Hamanaka N; Fujii N
Org Lett; 2002 Apr; 4(7):1051-4. PubMed ID: 11922780
[TBL] [Abstract][Full Text] [Related]
4. [Structure-activity relationship studies on cyclic RGD peptides utilizing novel alkene dipeptide isosteres].
Oishi S
Yakugaku Zasshi; 2004 May; 124(5):269-77. PubMed ID: 15118239
[TBL] [Abstract][Full Text] [Related]
5. Diastereoselective synthesis of psi[(E)-CMe=CH]- and psi[(E)-CMe=CMe]- type dipeptide isosteres based on organocopper-mediated anti-S(N)2' reaction.
Oishi S; Niida A; Kamano T; Odagaki Y; Tamamura H; Otaka A; Hamanaka N; Fujii N
Org Lett; 2002 Apr; 4(7):1055-8. PubMed ID: 11922781
[TBL] [Abstract][Full Text] [Related]
6. Stereoselective synthesis of (Z)-alkene-containing proline dipeptide mimetics.
Sasaki Y; Niida A; Tsuji T; Shigenaga A; Fujii N; Otaka A
J Org Chem; 2006 Jun; 71(13):4969-79. PubMed ID: 16776529
[TBL] [Abstract][Full Text] [Related]
7. Serine-cis-proline and serine-trans-proline isosteres: stereoselective synthesis of (Z)- and (E)-alkene mimics by Still-Wittig and Ireland-Claisen rearrangements.
Wang XJ; Hart SA; Xu B; Mason MD; Goodell JR; Etzkorn FA
J Org Chem; 2003 Mar; 68(6):2343-9. PubMed ID: 12636401
[TBL] [Abstract][Full Text] [Related]
8. SmI2-mediated reduction of gamma,gamma-difluoro-alpha,beta-enoates with application to the synthesis of functionalized (Z)-fluoroalkene-type dipeptide isosteres.
Otaka A; Watanabe J; Yukimasa A; Sasaki Y; Watanabe H; Kinoshita T; Oishi S; Tamamura H; Fujii N
J Org Chem; 2004 Mar; 69(5):1634-45. PubMed ID: 14987023
[TBL] [Abstract][Full Text] [Related]
9. Unequivocal synthesis of (Z)-alkene and (E)-fluoroalkene dipeptide isosteres to probe structural requirements of the peptide transporter PEPT1.
Niida A; Tomita K; Mizumoto M; Tanigaki H; Terada T; Oishi S; Otaka A; Inui K; Fujii N
Org Lett; 2006 Feb; 8(4):613-6. PubMed ID: 16468724
[TBL] [Abstract][Full Text] [Related]
10. Remote Stereoinduction in the Organocuprate-Mediated Allylic Alkylation of Allylic gem-Dichlorides: Highly Diastereoselective Synthesis of (Z)-Chloroalkene Dipeptide Isosteres.
Kobayakawa T; Narumi T; Tamamura H
Org Lett; 2015 May; 17(10):2302-5. PubMed ID: 25950639
[TBL] [Abstract][Full Text] [Related]
11. Stereocontrolled synthesis of psi[CH = CH] dipeptide isosteres.
Kempf DJ; Wang XC; Spanton SG
Int J Pept Protein Res; 1991 Sep; 38(3):237-41. PubMed ID: 1761370
[TBL] [Abstract][Full Text] [Related]
12. Trisubstituted (E)-alkene dipeptide isosteres as beta-turn promoters in the gramicidin S cyclodecapeptide scaffold.
Xiao J; Weisblum B; Wipf P
Org Lett; 2006 Oct; 8(21):4731-4. PubMed ID: 17020289
[TBL] [Abstract][Full Text] [Related]
13. Synthesis of the pro-gly dipeptide alkene isostere using olefin cross-metathesis.
Vasbinder MM; Miller SJ
J Org Chem; 2002 Aug; 67(17):6240-2. PubMed ID: 12182670
[TBL] [Abstract][Full Text] [Related]
14. Chloroalkene dipeptide isosteres as peptidomimetics.
Kobayakawa T; Tamamura H
Methods Enzymol; 2021; 656():191-239. PubMed ID: 34325787
[TBL] [Abstract][Full Text] [Related]
15. A novel one-pot reaction involving organocopper-mediated reduction/transmetalation/asymmetric alkylation, leading to the diastereoselective synthesis of functionalized (Z)-fluoroalkene dipeptide isosteres.
Narumi T; Niida A; Tomita K; Oishi S; Otaka A; Ohno H; Fujii N
Chem Commun (Camb); 2006 Dec; (45):4720-2. PubMed ID: 17109048
[TBL] [Abstract][Full Text] [Related]
16. Synthesis of Tic-D-Phe Psi[CH2-CH2] isostere and its use in the development of melanocortin receptor agonists.
Tian X; Chen X; Gan L; Hayes JC; Switzer AG; Solinsky MG; Ebetino FH; Wos JA; Pinney BB; Farmer JA; Crossdoersen D; Sheldon RJ
Bioorg Med Chem Lett; 2006 Mar; 16(6):1721-5. PubMed ID: 16376076
[TBL] [Abstract][Full Text] [Related]
17. Efficient synthesis of trifluoromethyl and related trisubstituted alkene dipeptide isosteres by palladium-catalyzed carbonylation of amino acid derived allylic carbonates.
Inokuchi E; Narumi T; Niida A; Kobayashi K; Tomita K; Oishi S; Ohno H; Fujii N
J Org Chem; 2008 May; 73(10):3942-5. PubMed ID: 18412390
[TBL] [Abstract][Full Text] [Related]
18. Enzymatic cyclisation of peptidomimetics with incorporated (E)-alkene dipeptide isosteres.
Garbe D; Sieber SA; Bandur NG; Koert U; Marahiel MA
Chembiochem; 2004 Jul; 5(7):1000-3. PubMed ID: 15239060
[No Abstract] [Full Text] [Related]
19. [Stereocontrolled synthesis of phosphinyl dipeptide isosteres using an asymmetric center at the phosphorus atom].
Yamagishi T
Yakugaku Zasshi; 2014; 134(9):915-24. PubMed ID: 25174361
[TBL] [Abstract][Full Text] [Related]
20. Amino acid-based synthesis of trifluoromethylalkene dipeptide isosteres by alcohol-assisted nucleophilic trifluoromethylation and organozinc-copper-mediated S(N)2' alkylation.
Kobayashi K; Narumi T; Oishi S; Ohno H; Fujii N
J Org Chem; 2009 Jun; 74(12):4626-9. PubMed ID: 19445465
[TBL] [Abstract][Full Text] [Related]
[Next] [New Search]
