185 related articles for article (PubMed ID: 12443785)
1. Antitrypanosomal activities and cytotoxicity of 5-nitro-2-furancarbohydrazides.
Millet R; Maes L; Landry V; Sergheraert C; Davioud-Charvet E
Bioorg Med Chem Lett; 2002 Dec; 12(24):3601-4. PubMed ID: 12443785
[TBL] [Abstract][Full Text] [Related]
2. Antimalarial, antitrypanosomal, and antileishmanial activities and cytotoxicity of bis(9-amino-6-chloro-2-methoxyacridines): influence of the linker.
Girault S; Grellier P; Berecibar A; Maes L; Mouray E; Lemière P; Debreu MA; Davioud-Charvet E; Sergheraert C
J Med Chem; 2000 Jul; 43(14):2646-54. PubMed ID: 10893302
[TBL] [Abstract][Full Text] [Related]
3. Synthesis and in vitro evaluation of tropane halogenated-derivatives against malaria, sleeping sickness, Chagas disease and leishmaniasis.
Cretton S; Bartholomeusz TA; Mehl F; Allenbach Y; Matheeussen A; Cos P; Maes L; Christen P
Med Chem; 2014; 10(8):753-8. PubMed ID: 24813684
[TBL] [Abstract][Full Text] [Related]
4. Design, synthesis, and evaluation of inhibitors of trypanosomal and leishmanial dihydrofolate reductase.
Chowdhury SF; Villamor VB; Guerrero RH; Leal I; Brun R; Croft SL; Goodman JM; Maes L; Ruiz-Perez LM; Pacanowska DG; Gilbert IH
J Med Chem; 1999 Oct; 42(21):4300-12. PubMed ID: 10543874
[TBL] [Abstract][Full Text] [Related]
5. In vitro and in silico studies of polycondensed diazine systems as anti-parasitic agents.
Almerico AM; Tutone M; Guarcello A; Lauria A
Bioorg Med Chem Lett; 2012 Jan; 22(2):1000-4. PubMed ID: 22197138
[TBL] [Abstract][Full Text] [Related]
6. Synthesis and biological activity of nitro heterocycles analogous to megazol, a trypanocidal lead.
Chauvière G; Bouteille B; Enanga B; de Albuquerque C; Croft SL; Dumas M; Périé J
J Med Chem; 2003 Jan; 46(3):427-40. PubMed ID: 12540242
[TBL] [Abstract][Full Text] [Related]
7. Novel 3-nitro-1H-1,2,4-triazole-based piperazines and 2-amino-1,3-benzothiazoles as antichagasic agents.
Papadopoulou MV; Bloomer WD; Rosenzweig HS; Kaiser M; Chatelain E; Ioset JR
Bioorg Med Chem; 2013 Nov; 21(21):6600-7. PubMed ID: 24012457
[TBL] [Abstract][Full Text] [Related]
8. Synthesis and tripanocidal activity of ferrocenyl and benzyl diamines against Trypanosoma brucei and Trypanosoma cruzi.
Velásquez AM; Francisco AI; Kohatsu AA; Silva FA; Rodrigues DF; Teixeira RG; Chiari BG; de Almeida MG; Isaac VL; Vargas MD; Cicarelli RM
Bioorg Med Chem Lett; 2014 Apr; 24(7):1707-10. PubMed ID: 24630563
[TBL] [Abstract][Full Text] [Related]
9. Synthesis and evaluation of novel prenylated chalcone derivatives as anti-leishmanial and anti-trypanosomal compounds.
Passalacqua TG; Dutra LA; de Almeida L; Velásquez AM; Torres FA; Yamasaki PR; dos Santos MB; Regasini LO; Michels PA; Bolzani Vda S; Graminha MA
Bioorg Med Chem Lett; 2015 Aug; 25(16):3342-5. PubMed ID: 26055530
[TBL] [Abstract][Full Text] [Related]
10. Novel 3-nitro-1H-1,2,4-triazole-based amides and sulfonamides as potential antitrypanosomal agents.
Papadopoulou MV; Bloomer WD; Rosenzweig HS; Chatelain E; Kaiser M; Wilkinson SR; McKenzie C; Ioset JR
J Med Chem; 2012 Jun; 55(11):5554-65. PubMed ID: 22550999
[TBL] [Abstract][Full Text] [Related]
11. In vitro antiprotozoal and cytotoxic activity of 33 ethonopharmacologically selected medicinal plants from Democratic Republic of Congo.
Musuyu Muganza D; Fruth BI; Nzunzu Lami J; Mesia GK; Kambu OK; Tona GL; Cimanga Kanyanga R; Cos P; Maes L; Apers S; Pieters L
J Ethnopharmacol; 2012 May; 141(1):301-8. PubMed ID: 22394563
[TBL] [Abstract][Full Text] [Related]
12. Lipophilic conformationally constrained spiro carbocyclic 2,6-diketopiperazine-1-acetohydroxamic acid analogues as trypanocidal and leishmanicidal agents: An extended SAR study.
Zoidis G; Tsotinis A; Tsatsaroni A; Taylor MC; Kelly JM; Efstathiou A; Smirlis D; Fytas G
Chem Biol Drug Des; 2018 Feb; 91(2):408-421. PubMed ID: 28834291
[TBL] [Abstract][Full Text] [Related]
13. Antiprotozoal activity of major constituents from the bioactive fraction of Verbesina encelioides.
Ezzat SM; Salama MM; Mahrous EA; Maes L; Pan CH; Abdel-Sattar E
Nat Prod Res; 2017 Mar; 31(6):676-680. PubMed ID: 27154232
[TBL] [Abstract][Full Text] [Related]
14. Tractable Quinolone Hydrazides Exhibiting Sub-Micromolar and Broad Spectrum Antitrypanosomal Activities.
Chirwa KA; Francisco KR; Dube PS; Park H; Legoabe LJ; Teixeira TR; Caffrey CR; Beteck RM
ChemMedChem; 2024 May; 19(9):e202300667. PubMed ID: 38326914
[TBL] [Abstract][Full Text] [Related]
15. Thiazolidinone/thiazole based hybrids - New class of antitrypanosomal agents.
Kryshchyshyn A; Kaminskyy D; Karpenko O; Gzella A; Grellier P; Lesyk R
Eur J Med Chem; 2019 Jul; 174():292-308. PubMed ID: 31051403
[TBL] [Abstract][Full Text] [Related]
16. A Nature-Inspired Design Yields a New Class of Steroids Against Trypanosomatids.
Aguilera E; Perdomo C; Espindola A; Corvo I; Faral-Tello P; Robello C; Serna E; Benítez F; Riveros R; Torres S; Vera de Bilbao NI; Yaluff G; Alvarez G
Molecules; 2019 Oct; 24(20):. PubMed ID: 31652542
[TBL] [Abstract][Full Text] [Related]
17. 2- and 3-substituted 1,4-naphthoquinone derivatives as subversive substrates of trypanothione reductase and lipoamide dehydrogenase from Trypanosoma cruzi: synthesis and correlation between redox cycling activities and in vitro cytotoxicity.
Salmon-Chemin L; Buisine E; Yardley V; Kohler S; Debreu MA; Landry V; Sergheraert C; Croft SL; Krauth-Siegel RL; Davioud-Charvet E
J Med Chem; 2001 Feb; 44(4):548-65. PubMed ID: 11170645
[TBL] [Abstract][Full Text] [Related]
18. 1,4-Dihydroxy-2,3-dioxatricyclo[8.4.0.0(4,9)]tetradecane and derivatives with in vitro activity against Plasmodium falciparum, Trypanasoma b brucei, Trypanasoma cruzi, and Leishmaniasis infantum.
Howarth J; Wilson D
Bioorg Med Chem Lett; 2003 Jun; 13(12):2013-5. PubMed ID: 12781185
[TBL] [Abstract][Full Text] [Related]
19. Cytotoxicity of (2,2':6',2''-terpyridine)platinum(II) complexes to Leishmania donovani, Trypanosoma cruzi, and Trypanosoma brucei.
Lowe G; Droz AS; Vilaivan T; Weaver GW; Tweedale L; Pratt JM; Rock P; Yardley V; Croft SL
J Med Chem; 1999 Mar; 42(6):999-1006. PubMed ID: 10090783
[TBL] [Abstract][Full Text] [Related]
20. Synthesis, cytotoxicity, and antiplasmodial and antitrypanosomal activity of new neocryptolepine derivatives.
Jonckers TH; van Miert S; Cimanga K; Bailly C; Colson P; De Pauw-Gillet MC; van den Heuvel H; Claeys M; Lemière F; Esmans EL; Rozenski J; Quirijnen L; Maes L; Dommisse R; Lemière GL; Vlietinck A; Pieters L
J Med Chem; 2002 Aug; 45(16):3497-508. PubMed ID: 12139461
[TBL] [Abstract][Full Text] [Related]
[Next] [New Search]