These tools will no longer be maintained as of December 31, 2024. Archived website can be found here. PubMed4Hh GitHub repository can be found here. Contact NLM Customer Service if you have questions.


BIOMARKERS

Molecular Biopsy of Human Tumors

- a resource for Precision Medicine *

142 related articles for article (PubMed ID: 12666176)

  • 1. 1H-NMR studies on a potent and selective antagonist at human melanocortin receptor 4 (hMC-4R).
    Victoria Silva Elipe M; Mosley RT; Bednarek MA; Arison BH
    Biopolymers; 2003 Apr; 68(4):512-27. PubMed ID: 12666176
    [TBL] [Abstract][Full Text] [Related]  

  • 2. Analogs of MTII, lactam derivatives of alpha-melanotropin, modified at the N-terminus, and their selectivity at human melanocortin receptors 3, 4, and 5.
    Bednarek MA; Macneil T; Kalyani RN; Tang R; Van der Ploeg LH; Weinberg DH
    Biochem Biophys Res Commun; 1999 Jul; 261(1):209-13. PubMed ID: 10405347
    [TBL] [Abstract][Full Text] [Related]  

  • 3. Solution structures of cyclic melanocortin agonists and antagonists by NMR.
    Ying J; Kövér KE; Gu X; Han G; Trivedi DB; Kavarana MJ; Hruby VJ
    Biopolymers; 2003; 71(6):696-716. PubMed ID: 14991679
    [TBL] [Abstract][Full Text] [Related]  

  • 4. Analogs of lactam derivatives of alpha-melanotropin with basic and acidic residues.
    Bednarek MA; MacNeil T; Kalyani RN; Tang R; Van der Ploeg LH; Weinberg DH
    Biochem Biophys Res Commun; 2000 May; 272(1):23-8. PubMed ID: 10872798
    [TBL] [Abstract][Full Text] [Related]  

  • 5. Structure-activity relationships of novel cyclic alpha-MSH/beta-MSH hybrid analogues that lead to potent and selective ligands for the human MC3R and human MC5R.
    Balse-Srinivasan P; Grieco P; Cai M; Trivedi D; Hruby VJ
    J Med Chem; 2003 Aug; 46(17):3728-33. PubMed ID: 12904077
    [TBL] [Abstract][Full Text] [Related]  

  • 6. Design of novel chimeric melanotropin-deltorphin analogues. Discovery of the first potent human melanocortin 1 receptor antagonist.
    Han G; Quillan JM; Carlson K; Sadée W; Hruby VJ
    J Med Chem; 2003 Feb; 46(5):810-9. PubMed ID: 12593660
    [TBL] [Abstract][Full Text] [Related]  

  • 7. Further pharmacological characterization of the selective melanocortin 4 receptor antagonist HS014: comparison with SHU9119.
    Schiöth HB; Muceniece R; Mutulis F; Bouifrouri AA; Mutule I; Wikberg JE
    Neuropeptides; 1999 Jun; 33(3):191-6. PubMed ID: 10657491
    [TBL] [Abstract][Full Text] [Related]  

  • 8. Structure-activity relationships of gamma-MSH analogues at the human melanocortin MC3, MC4, and MC5 receptors. Discovery of highly selective hMC3R, hMC4R, and hMC5R analogues.
    Balse-Srinivasan P; Grieco P; Cai M; Trivedi D; Hruby VJ
    J Med Chem; 2003 Nov; 46(23):4965-73. PubMed ID: 14584947
    [TBL] [Abstract][Full Text] [Related]  

  • 9. Accelerating sensory recovery after sciatic nerve crush: non-selective versus melanocortin MC4 receptor-selective peptides.
    Nijenhuis WA; Wanders N; Kruijtzer JA; Liskamp RM; Gispen WH; Adan RA
    Eur J Pharmacol; 2004 Jul; 495(2-3):145-52. PubMed ID: 15249163
    [TBL] [Abstract][Full Text] [Related]  

  • 10. Cyclic analogs of alpha-melanocyte-stimulating hormone (alphaMSH) with high agonist potency and selectivity at human melanocortin receptor 1b.
    Bednarek MA; MacNeil T; Tang R; Fong TM; Cabello MA; Maroto M; Teran A
    Peptides; 2008 Jun; 29(6):1010-7. PubMed ID: 18378043
    [TBL] [Abstract][Full Text] [Related]  

  • 11. Selective, high affinity peptide antagonists of alpha-melanotropin action at human melanocortin receptor 4: their synthesis and biological evaluation in vitro.
    Bednarek MA; MacNeil T; Kalyani RN; Tang R; Van der Ploeg LH; Weinberg DH
    J Med Chem; 2001 Oct; 44(22):3665-72. PubMed ID: 11606131
    [TBL] [Abstract][Full Text] [Related]  

  • 12. Design of cyclic peptides with agonist activity at melanocortin receptor-4.
    Odagami T; Tsuda Y; Kogami Y; Kouji H; Okada Y
    Bioorg Med Chem Lett; 2006 Jul; 16(14):3723-6. PubMed ID: 16678415
    [TBL] [Abstract][Full Text] [Related]  

  • 13. Identification of putative agouti-related protein(87-132)-melanocortin-4 receptor interactions by homology molecular modeling and validation using chimeric peptide ligands.
    Wilczynski A; Wang XS; Joseph CG; Xiang Z; Bauzo RM; Scott JW; Sorensen NB; Shaw AM; Millard WJ; Richards NG; Haskell-Luevano C
    J Med Chem; 2004 Apr; 47(9):2194-207. PubMed ID: 15084118
    [TBL] [Abstract][Full Text] [Related]  

  • 14. De novo design, synthesis, and pharmacology of alpha-melanocyte stimulating hormone analogues derived from somatostatin by a hybrid approach.
    Han G; Haskell-Luevano C; Kendall L; Bonner G; Hadley ME; Cone RD; Hruby VJ
    J Med Chem; 2004 Mar; 47(6):1514-26. PubMed ID: 14998337
    [TBL] [Abstract][Full Text] [Related]  

  • 15. Effect of the melanocortin receptor stimulation or inhibition on ethanol intake in alcohol-preferring rats.
    Polidori C; Geary N; Massi M
    Peptides; 2006 Jan; 27(1):144-9. PubMed ID: 16198024
    [TBL] [Abstract][Full Text] [Related]  

  • 16. Potent and selective agonists of human melanocortin receptor 5: cyclic analogues of alpha-melanocyte-stimulating hormone.
    Bednarek MA; MacNeil T; Tang R; Fong TM; Cabello MA; Maroto M; Teran A
    J Med Chem; 2007 May; 50(10):2520-6. PubMed ID: 17455928
    [TBL] [Abstract][Full Text] [Related]  

  • 17. Feeding and behavioural effects of central administration of the melanocortin 3/4-R antagonist SHU9119 in obese and lean Siberian hamsters.
    Schuhler S; Horan TL; Hastings MH; Mercer JG; Morgan PJ; Ebling FJ
    Behav Brain Res; 2004 Jul; 152(2):177-85. PubMed ID: 15196785
    [TBL] [Abstract][Full Text] [Related]  

  • 18. Melanocortin peptides affect the motivation to feed in rainbow trout (Oncorhynchus mykiss).
    Schjolden J; Schiöth HB; Larhammar D; Winberg S; Larson ET
    Gen Comp Endocrinol; 2009 Jan; 160(2):134-8. PubMed ID: 19027741
    [TBL] [Abstract][Full Text] [Related]  

  • 19. Potent and selective peptide agonists of alpha-melanotropin action at human melanocortin receptor 4: their synthesis and biological evaluation in vitro.
    Bednarek MA; MacNeil T; Tang R; Kalyani RN; Van der Ploeg LH; Weinberg DH
    Biochem Biophys Res Commun; 2001 Aug; 286(3):641-5. PubMed ID: 11511108
    [TBL] [Abstract][Full Text] [Related]  

  • 20. Discovery of a beta-MSH-derived MC-4R selective agonist.
    Mayer JP; Hsiung HM; Flora DB; Edwards P; Smith DP; Zhang XY; Gadski RA; Heiman ML; Hertel JL; Emmerson PJ; Husain S; O'brien TP; Kahl SD; Smiley DL; Zhang L; Dimarchi RD; Yan LZ
    J Med Chem; 2005 May; 48(9):3095-8. PubMed ID: 15857110
    [TBL] [Abstract][Full Text] [Related]  

    [Next]    [New Search]
    of 8.