BIOMARKERS

Molecular Biopsy of Human Tumors

- a resource for Precision Medicine *

281 related articles for article (PubMed ID: 12723946)

  • 1. Novel pyrazolo[3,4-d]pyrimidine-based inhibitors of Staphlococcus aureus DNA polymerase III: design, synthesis, and biological evaluation.
    Ali A; Taylor GE; Ellsworth K; Harris G; Painter R; Silver LL; Young K
    J Med Chem; 2003 May; 46(10):1824-30. PubMed ID: 12723946
    [TBL] [Abstract][Full Text] [Related]  

  • 2. 6-Anilinouracil-based inhibitors of Bacillus subtilis DNA polymerase III: antipolymerase and antimicrobial structure-activity relationships based on substitution at uracil N3.
    Tarantino PM; Zhi C; Gambino JJ; Wright GE; Brown NC
    J Med Chem; 1999 Jun; 42(11):2035-40. PubMed ID: 10354411
    [TBL] [Abstract][Full Text] [Related]  

  • 3. Design and synthesis of novel antibacterial agents with inhibitory activity against DNA polymerase III.
    Ali A; Aster SD; Graham DW; Patel GF; Taylor GE; Tolman RL; Painter RE; Silver LL; Young K; Ellsworth K; Geissler W; Harris GS
    Bioorg Med Chem Lett; 2001 Aug; 11(16):2185-8. PubMed ID: 11514166
    [TBL] [Abstract][Full Text] [Related]  

  • 4. Novel non-nucleobase inhibitors of Staphylococcus aureus DNA polymerase IIIC.
    Rose Y; Ciblat S; Reddy R; Belley AC; Dietrich E; Lehoux D; McKay GA; Poirier H; Far AR; Delorme D
    Bioorg Med Chem Lett; 2006 Feb; 16(4):891-6. PubMed ID: 16298129
    [TBL] [Abstract][Full Text] [Related]  

  • 5. Synthesis of substituted 6-anilinouracils and their inhibition of DNA polymerase IIIC and Gram-positive bacterial growth.
    Zhi C; Long ZY; Gambino J; Xu WC; Brown NC; Barnes M; Butler M; LaMarr W; Wright GE
    J Med Chem; 2003 Jun; 46(13):2731-9. PubMed ID: 12801236
    [TBL] [Abstract][Full Text] [Related]  

  • 6. Synthesis and antimycobacterial evaluation of various 6-substituted pyrazolo[3,4-d]pyrimidine derivatives.
    Trivedi A; Vaghasiya S; Dholariya B; Dodiya D; Shah V
    J Enzyme Inhib Med Chem; 2010 Dec; 25(6):893-9. PubMed ID: 21054238
    [TBL] [Abstract][Full Text] [Related]  

  • 7. Improved synthesis of antibacterial 3-substituted 6-anilinouracils.
    Svenstrup N; Kuhl A; Ehlert K; Häbich D
    Bioorg Med Chem Lett; 2008 Jun; 18(11):3215-8. PubMed ID: 18468893
    [TBL] [Abstract][Full Text] [Related]  

  • 8. Synthesis and antibacterial activity of 3-substituted-6-(3-ethyl-4-methylanilino)uracils.
    Zhi C; Long ZY; Manikowski A; Brown NC; Tarantino PM; Holm K; Dix EJ; Wright GE; Foster KA; Butler MM; LaMarr WA; Skow DJ; Motorina I; Lamothe S; Storer R
    J Med Chem; 2005 Nov; 48(22):7063-74. PubMed ID: 16250666
    [TBL] [Abstract][Full Text] [Related]  

  • 9. Design, synthesis, and biological evaluation of C9- and C2-substituted pyrazolo[4,3-e]-1,2,4-triazolo[1,5-c]pyrimidines as new A2A and A3 adenosine receptors antagonists.
    Baraldi PG; Fruttarolo F; Tabrizi MA; Preti D; Romagnoli R; El-Kashef H; Moorman A; Varani K; Gessi S; Merighi S; Borea PA
    J Med Chem; 2003 Mar; 46(7):1229-41. PubMed ID: 12646033
    [TBL] [Abstract][Full Text] [Related]  

  • 10. Synthesis of some novel pyrazolo[3,4-b]pyridine and pyrazolo[3,4-d]pyrimidine derivatives bearing 5,6-diphenyl-1,2,4-triazine moiety as potential antimicrobial agents.
    El-Sayed Ali T
    Eur J Med Chem; 2009 Nov; 44(11):4385-92. PubMed ID: 19586688
    [TBL] [Abstract][Full Text] [Related]  

  • 11. Substituted salicylanilides as inhibitors of two-component regulatory systems in bacteria.
    Macielag MJ; Demers JP; Fraga-Spano SA; Hlasta DJ; Johnson SG; Kanojia RM; Russell RK; Sui Z; Weidner-Wells MA; Werblood H; Foleno BD; Goldschmidt RM; Loeloff MJ; Webb GC; Barrett JF
    J Med Chem; 1998 Jul; 41(16):2939-45. PubMed ID: 9685233
    [TBL] [Abstract][Full Text] [Related]  

  • 12. Novel pyrazole derivatives as potent inhibitors of type II topoisomerases. Part 1: synthesis and preliminary SAR analysis.
    Gomez L; Hack MD; Wu J; Wiener JJ; Venkatesan H; Santillán A; Pippel DJ; Mani N; Morrow BJ; Motley ST; Shaw KJ; Wolin R; Grice CA; Jones TK
    Bioorg Med Chem Lett; 2007 May; 17(10):2723-7. PubMed ID: 17368897
    [TBL] [Abstract][Full Text] [Related]  

  • 13. Synthesis, isomerization, and antimicrobial evaluation of some pyrazolopyranotriazolopyrimidine derivatives.
    Shamroukh AH; Zaki ME; Morsy EM; Abdel-Motti FM; Abdel-Megeid FM
    Arch Pharm (Weinheim); 2007 Jul; 340(7):345-51. PubMed ID: 17610300
    [TBL] [Abstract][Full Text] [Related]  

  • 14. Synthesis, structure and antibacterial activity of novel 1-(5-substituted-3-substituted-4,5-dihydropyrazol-1-yl)ethanone oxime ester derivatives.
    Liu XH; Cui P; Song BA; Bhadury PS; Zhu HL; Wang SF
    Bioorg Med Chem; 2008 Apr; 16(7):4075-82. PubMed ID: 18262793
    [TBL] [Abstract][Full Text] [Related]  

  • 15. Synthesis of some novel pyrazolo[3,4-d]pyrimidine derivatives as potential antimicrobial agents.
    Holla BS; Mahalinga M; Karthikeyan MS; Akberali PM; Shetty NS
    Bioorg Med Chem; 2006 Mar; 14(6):2040-7. PubMed ID: 16310361
    [TBL] [Abstract][Full Text] [Related]  

  • 16. Biological characterization of novel inhibitors of the gram-positive DNA polymerase IIIC enzyme.
    Kuhl A; Svenstrup N; Ladel C; Otteneder M; Binas A; Schiffer G; Brands M; Lampe T; Ziegelbauer K; Rübsamen-Waigmann H; Haebich D; Ehlert K
    Antimicrob Agents Chemother; 2005 Mar; 49(3):987-95. PubMed ID: 15728893
    [TBL] [Abstract][Full Text] [Related]  

  • 17. Synthesis of 3-(1,3,4-thiadiazol-2-yl)pyrazolo[1,5-a] pyrimidine derivatives as potential antimicrobial agents.
    Auzzi G; Costanzo A; Bruni F; Clauser M; Guerrini G; Selleri S; Pecori Vettori L
    Farmaco; 1990 Nov; 45(11):1193-205. PubMed ID: 2128451
    [TBL] [Abstract][Full Text] [Related]  

  • 18. Synthesis and antibacterial activity of a novel series of potent DNA gyrase inhibitors. Pyrazole derivatives.
    Tanitame A; Oyamada Y; Ofuji K; Fujimoto M; Iwai N; Hiyama Y; Suzuki K; Ito H; Terauchi H; Kawasaki M; Nagai K; Wachi M; Yamagishi J
    J Med Chem; 2004 Jul; 47(14):3693-6. PubMed ID: 15214796
    [TBL] [Abstract][Full Text] [Related]  

  • 19. Inhibitors of DNA polymerase III as novel antimicrobial agents against gram-positive eubacteria.
    Tarantino PM; Zhi C; Wright GE; Brown NC
    Antimicrob Agents Chemother; 1999 Aug; 43(8):1982-7. PubMed ID: 10428923
    [TBL] [Abstract][Full Text] [Related]  

  • 20. Antibacterial and antifungal activities of new pyrazolo[3,4-d]pyridazin derivatives.
    Akbas E; Berber I
    Eur J Med Chem; 2005 Apr; 40(4):401-5. PubMed ID: 15804539
    [TBL] [Abstract][Full Text] [Related]  

    [Next]    [New Search]
    of 15.