These tools will no longer be maintained as of December 31, 2024. Archived website can be found here. PubMed4Hh GitHub repository can be found here. Contact NLM Customer Service if you have questions.


BIOMARKERS

Molecular Biopsy of Human Tumors

- a resource for Precision Medicine *

93 related articles for article (PubMed ID: 12818667)

  • 1. Novel tetrahydropyran-based peptidomimetics from a bioisosteric transformation of a tripeptide. Evidence of their activity at melanocortin receptors.
    Mazur AW; Kulesza A; Mishra RK; Cross-Doersen D; Russell AF; Ebetino FH
    Bioorg Med Chem; 2003 Jul; 11(14):3053-63. PubMed ID: 12818667
    [TBL] [Abstract][Full Text] [Related]  

  • 2. Synthesis of 2,4,5-trisubstituted tetrahydropyrans as peptidomimetic scaffolds for melanocortin receptor ligands.
    Kulesza A; Ebetino FH; Mishra RK; Cross-Doersen D; Mazur AW
    Org Lett; 2003 Apr; 5(8):1163-6. PubMed ID: 12688709
    [TBL] [Abstract][Full Text] [Related]  

  • 3. Structure-activity relationships of the melanocortin tetrapeptide Ac-His-DPhe-Arg-Trp-NH(2) at the mouse melanocortin receptors: part 2 modifications at the Phe position.
    Holder JR; Bauzo RM; Xiang Z; Haskell-Luevano C
    J Med Chem; 2002 Jul; 45(14):3073-81. PubMed ID: 12086493
    [TBL] [Abstract][Full Text] [Related]  

  • 4. Design of cyclic peptides with biological activities from biologically active peptides: the case of peptide modulators of melanocortin receptors.
    Hruby VJ
    Biopolymers; 2016 Nov; 106(6):884-888. PubMed ID: 27486849
    [TBL] [Abstract][Full Text] [Related]  

  • 5. Structure-activity relationships of the melanocortin tetrapeptide Ac-His-D-Phe-Arg-Trp-NH2 at the mouse melanocortin receptors. 4. Modifications at the Trp position.
    Holder JR; Xiang Z; Bauzo RM; Haskell-Luevano C
    J Med Chem; 2002 Dec; 45(26):5736-44. PubMed ID: 12477357
    [TBL] [Abstract][Full Text] [Related]  

  • 6. Design of novel chimeric melanotropin-deltorphin analogues. Discovery of the first potent human melanocortin 1 receptor antagonist.
    Han G; Quillan JM; Carlson K; Sadée W; Hruby VJ
    J Med Chem; 2003 Feb; 46(5):810-9. PubMed ID: 12593660
    [TBL] [Abstract][Full Text] [Related]  

  • 7. Chimeric NDP-MSH and MTII melanocortin peptides with agouti-related protein (AGRP) Arg-Phe-Phe amino acids possess agonist melanocortin receptor activity.
    Joseph CG; Wilczynski A; Holder JR; Xiang Z; Bauzo RM; Scott JW; Haskell-Luevano C
    Peptides; 2003 Dec; 24(12):1899-908. PubMed ID: 15127941
    [TBL] [Abstract][Full Text] [Related]  

  • 8. Structure-activity relationships of the melanocortin tetrapeptide Ac-His-DPhe-Arg-Trp-NH(2) at the mouse melanocortin receptors. 1. Modifications at the His position.
    Holder JR; Bauzo RM; Xiang Z; Haskell-Luevano C
    J Med Chem; 2002 Jun; 45(13):2801-10. PubMed ID: 12061882
    [TBL] [Abstract][Full Text] [Related]  

  • 9. Identification of putative agouti-related protein(87-132)-melanocortin-4 receptor interactions by homology molecular modeling and validation using chimeric peptide ligands.
    Wilczynski A; Wang XS; Joseph CG; Xiang Z; Bauzo RM; Scott JW; Sorensen NB; Shaw AM; Millard WJ; Richards NG; Haskell-Luevano C
    J Med Chem; 2004 Apr; 47(9):2194-207. PubMed ID: 15084118
    [TBL] [Abstract][Full Text] [Related]  

  • 10. Aza-scanning of the potent melanocortin receptor agonist Ac-His-D-Phe-Arg-Trp-NH.
    Boeglin D; Xiang Z; Sorenson NB; Wood MS; Haskell-Luevano C; Lubell WD
    Chem Biol Drug Des; 2006 Apr; 67(4):275-83. PubMed ID: 16629825
    [TBL] [Abstract][Full Text] [Related]  

  • 11. Structure-activity relationships of the unique and potent agouti-related protein (AGRP)-melanocortin chimeric Tyr-c[beta-Asp-His-DPhe-Arg-Trp-Asn-Ala-Phe-Dpr]-Tyr-NH2 peptide template.
    Wilczynski A; Wilson KR; Scott JW; Edison AS; Haskell-Luevano C
    J Med Chem; 2005 Apr; 48(8):3060-75. PubMed ID: 15828845
    [TBL] [Abstract][Full Text] [Related]  

  • 12. N-terminal fatty acylated His-dPhe-Arg-Trp-NH(2) tetrapeptides: influence of fatty acid chain length on potency and selectivity at the mouse melanocortin receptors and human melanocytes.
    Todorovic A; Holder JR; Bauzo RM; Scott JW; Kavanagh R; Abdel-Malek Z; Haskell-Luevano C
    J Med Chem; 2005 May; 48(9):3328-36. PubMed ID: 15857138
    [TBL] [Abstract][Full Text] [Related]  

  • 13. Structure-activity relationships of the melanocortin tetrapeptide Ac-His-DPhe-Arg-Trp-NH2 at the mouse melanocortin receptors. Part 3: modifications at the Arg position.
    Holder JR; Xiang Z; Bauzo RM; Haskell-Luevano C
    Peptides; 2003 Jan; 24(1):73-82. PubMed ID: 12576087
    [TBL] [Abstract][Full Text] [Related]  

  • 14. Design of a new peptidomimetic agonist for the melanocortin receptors based on the solution structure of the peptide ligand, Ac-Nle-cyclo[Asp-Pro-DPhe-Arg-Trp-Lys]-NH(2).
    Fotsch C; Smith DM; Adams JA; Cheetham J; Croghan M; Doherty EM; Hale C; Jarosinski MA; Kelly MG; Norman MH; Tamayo NA; Xi N; Baumgartner JW
    Bioorg Med Chem Lett; 2003 Jul; 13(14):2337-40. PubMed ID: 12824029
    [TBL] [Abstract][Full Text] [Related]  

  • 15. Discovery of Novel Potent and Selective Agonists at the Melanocortin-3 Receptor.
    Carotenuto A; Merlino F; Cai M; Brancaccio D; Yousif AM; Novellino E; Hruby VJ; Grieco P
    J Med Chem; 2015 Dec; 58(24):9773-8. PubMed ID: 26599352
    [TBL] [Abstract][Full Text] [Related]  

  • 16. Melanocortin tetrapeptides modified at the N-terminus, His, Phe, Arg, and Trp positions.
    Holder J; Haskell-Luevano C
    Ann N Y Acad Sci; 2003 Jun; 994():36-48. PubMed ID: 12851296
    [TBL] [Abstract][Full Text] [Related]  

  • 17. Cyclization increases the antimicrobial activity and selectivity of arginine- and tryptophan-containing hexapeptides.
    Dathe M; Nikolenko H; Klose J; Bienert M
    Biochemistry; 2004 Jul; 43(28):9140-50. PubMed ID: 15248771
    [TBL] [Abstract][Full Text] [Related]  

  • 18. D-Amino acid scan of gamma-melanocyte-stimulating hormone: importance of Trp(8) on human MC3 receptor selectivity.
    Grieco P; Balse PM; Weinberg D; MacNeil T; Hruby VJ
    J Med Chem; 2000 Dec; 43(26):4998-5002. PubMed ID: 11150170
    [TBL] [Abstract][Full Text] [Related]  

  • 19. Structure⁻Activity Relationships of the Tetrapeptide Ac-His-Arg-(
    Schlasner KN; Ericson MD; Doering SR; Freeman KT; Weinrich M; Haskell-Luevano C
    Molecules; 2019 Apr; 24(8):. PubMed ID: 31013889
    [TBL] [Abstract][Full Text] [Related]  

  • 20. 1,2,3-Triazole Rings as a Disulfide Bond Mimetic in Chimeric AGRP-Melanocortin Peptides: Design, Synthesis, and Functional Characterization.
    Tala SR; Singh A; Lensing CJ; Schnell SM; Freeman KT; Rocca JR; Haskell-Luevano C
    ACS Chem Neurosci; 2018 May; 9(5):1001-1013. PubMed ID: 29257879
    [TBL] [Abstract][Full Text] [Related]  

    [Next]    [New Search]
    of 5.