247 related articles for article (PubMed ID: 12857111)
1. Solid-phase parallel synthesis of 17alpha-substituted estradiol sulfamate and phenol libraries using the multidetachable sulfamate linker.
Ciobanu LC; Poirier D
J Comb Chem; 2003; 5(4):429-40. PubMed ID: 12857111
[TBL] [Abstract][Full Text] [Related]
2. Potent inhibition of steroid sulfatase activity by 3-O-sulfamate 17alpha-benzyl(or 4'-tert-butylbenzyl)estra-1,3,5(10)-trienes: combination of two substituents at positions C3 and c17alpha of estradiol.
Ciobanu LC; Boivin RP; Luu-The V; Labrie F; Poirier D
J Med Chem; 1999 Jun; 42(12):2280-6. PubMed ID: 10377235
[TBL] [Abstract][Full Text] [Related]
3. Structure-activity relationships of 17alpha-derivatives of estradiol as inhibitors of steroid sulfatase.
Boivin RP; Luu-The V; Lachance R; Labrie F; Poirier D
J Med Chem; 2000 Nov; 43(23):4465-78. PubMed ID: 11087571
[TBL] [Abstract][Full Text] [Related]
4. A multidetachable sulfamate linker successfully used in a solid-phase strategy to generate libraries of sulfamate and phenol derivatives.
Poirier D; Ciobanu LC; Bérubé M
Bioorg Med Chem Lett; 2002 Oct; 12(20):2833-8. PubMed ID: 12270157
[TBL] [Abstract][Full Text] [Related]
5. Steroidal and nonsteroidal sulfamates as potent inhibitors of steroid sulfatase.
Woo LW; Howarth NM; Purohit A; Hejaz HA; Reed MJ; Potter BV
J Med Chem; 1998 Mar; 41(7):1068-83. PubMed ID: 9544207
[TBL] [Abstract][Full Text] [Related]
6. 3Beta-sulfamate derivatives of C19 and C21 steroids bearing a t-butylbenzyl or a benzyl group: synthesis and evaluation as non-estrogenic and non-androgenic steroid sulfatase inhibitors.
Ciobanu LC; Boivin RP; Luu-The V; Poirier D
J Enzyme Inhib Med Chem; 2003 Feb; 18(1):15-26. PubMed ID: 12751816
[TBL] [Abstract][Full Text] [Related]
7. Nonsteroidal compounds designed to mimic potent steroid sulfatase inhibitors.
Ciobanu LC; Luu-The V; Poirier D
J Steroid Biochem Mol Biol; 2002 Mar; 80(3):339-53. PubMed ID: 11948019
[TBL] [Abstract][Full Text] [Related]
8. Preparation of 6beta-estradiol derivative libraries as bisubstrate inhibitors of 7beta-hydroxysteroid dehydrogenase type using the multidetachable sulfamate linker.
Bérubé M; Delagoutte F; Poirier D
Molecules; 2010 Mar; 15(3):1590-631. PubMed ID: 20336003
[TBL] [Abstract][Full Text] [Related]
9. Inhibition of estrone sulfate-induced uterine growth by potent nonestrogenic steroidal inhibitors of steroid sulfatase.
Ciobanu LC; Luu-The V; Martel C; Labrie F; Poirier D
Cancer Res; 2003 Oct; 63(19):6442-6. PubMed ID: 14559834
[TBL] [Abstract][Full Text] [Related]
10. Synthesis and biological activity of the superestrogen (E)-17-oximino-3-O-sulfamoyl-1,3,5(10)-estratriene: x-ray crystal structure of (E)-17-oximino-3-hydroxy-1,3,5(10)-estratriene.
Hejaz HA; Purohit A; Mahon MF; Reed MJ; Potter BV
J Med Chem; 1999 Aug; 42(16):3188-92. PubMed ID: 10447965
[TBL] [Abstract][Full Text] [Related]
11. Carbonic anhydrase inhibitors. Inhibition of cytosolic isozymes I and II and transmembrane, tumor-associated isozyme IX with sulfamates including EMATE also acting as steroid sulfatase inhibitors.
Winum JY; Vullo D; Casini A; Montero JL; Scozzafava A; Supuran CT
J Med Chem; 2003 May; 46(11):2197-204. PubMed ID: 12747791
[TBL] [Abstract][Full Text] [Related]
12. 2-Substituted 4-(thio)chromenone 6-O-sulfamates: potent inhibitors of human steroid sulfatase.
Nussbaumer P; Lehr P; Billich A
J Med Chem; 2002 Sep; 45(19):4310-20. PubMed ID: 12213072
[TBL] [Abstract][Full Text] [Related]
13. 2-phenylindole sulfamates: inhibitors of steroid sulfatase with antiproliferative activity in MCF-7 breast cancer cells.
Walter G; Liebl R; von Angerer E
J Steroid Biochem Mol Biol; 2004 Apr; 88(4-5):409-20. PubMed ID: 15145451
[TBL] [Abstract][Full Text] [Related]
14. In vivo activity of 4-methylcoumarin-7-O-sulfamate, a nonsteroidal, nonestrogenic steroid sulfatase inhibitor.
Purohit A; Woo LW; Singh A; Winterborn CJ; Potter BV; Reed MJ
Cancer Res; 1996 Nov; 56(21):4950-5. PubMed ID: 8895749
[TBL] [Abstract][Full Text] [Related]
15. First report of the investigation into the importance of pK(a) in the inhibition of estrone sulfatase by sulfamate containing compounds.
Ahmed S; James K; Patel CK
Biochem Biophys Res Commun; 2000 Jun; 272(2):583-5. PubMed ID: 10833455
[TBL] [Abstract][Full Text] [Related]
16. Scavestrogen sulfamates: correlation between estrone sulfatase inhibiting and antioxidant effects.
Römer W; Oettel M; Schwarz S
Can J Physiol Pharmacol; 1998 Feb; 76(2):99-109. PubMed ID: 9635147
[TBL] [Abstract][Full Text] [Related]
17. Structure-activity relationship determination within a group of substituted phenyl sulfamate based compounds against the enzyme oestrone sulfatase.
Patel CK; Galisson A; James K; Owen CP; Ahmed S
J Pharm Pharmacol; 2003 Feb; 55(2):211-8. PubMed ID: 12631414
[TBL] [Abstract][Full Text] [Related]
18. Development of novel steroid sulfatase inhibitors. I. Synthesis and biological evaluation of biphenyl-4-O-sulfamates.
Okada M; Nakagawa T; Iwashita S; Takegawa S; Fujii T; Koizumi N
J Steroid Biochem Mol Biol; 2003 Nov; 87(2-3):141-8. PubMed ID: 14672734
[TBL] [Abstract][Full Text] [Related]
19. 4,4'-Benzophenone-O,O'-disulfamate: a potent inhibitor of steroid sulfatase.
Nussbaumer P; Bilban M; Billich A
Bioorg Med Chem Lett; 2002 Aug; 12(16):2093-5. PubMed ID: 12127511
[TBL] [Abstract][Full Text] [Related]
20. 17Alpha-alkan (or alkyn) amide derivatives of estradiol as inhibitors of steroid-sulfatase activity.
Boivin RP; Labrie F; Poirier D
Steroids; 1999 Dec; 64(12):825-33. PubMed ID: 10576217
[TBL] [Abstract][Full Text] [Related]
[Next] [New Search]