BIOMARKERS

Molecular Biopsy of Human Tumors

- a resource for Precision Medicine *

119 related articles for article (PubMed ID: 12904075)

  • 1. A comparison of phosphonothioic acids with phosphonic acids as phosphatase inhibitors.
    Swierczek K; Pandey AS; Peters JW; Hengge AC
    J Med Chem; 2003 Aug; 46(17):3703-8. PubMed ID: 12904075
    [TBL] [Abstract][Full Text] [Related]  

  • 2. A nonhydrolyzable analogue of phosphotyrosine, and related aryloxymethano- and aryloxyethano-phosphonic acids as motifs for inhibition of phosphatases.
    Iyer S; Younker JM; Czyryca PG; Hengge AC
    Bioorg Med Chem Lett; 2004 Dec; 14(23):5931-5. PubMed ID: 15501071
    [TBL] [Abstract][Full Text] [Related]  

  • 3. Stereoselective inhibition of glutamate carboxypeptidase by chiral phosphonothioic acids.
    Lu H; Berkman CE
    Bioorg Med Chem; 2001 Feb; 9(2):395-402. PubMed ID: 11249132
    [TBL] [Abstract][Full Text] [Related]  

  • 4. Synthesis of [difluoro-(3-alkenylphenyl)-methyl]-phosphonic acids on non-crosslinked polystyrene and their evaluation as inhibitors of PTP1B.
    Hum G; Lee J; Taylor SD
    Bioorg Med Chem Lett; 2002 Dec; 12(23):3471-4. PubMed ID: 12419386
    [TBL] [Abstract][Full Text] [Related]  

  • 5. Mutation of Arg-166 of alkaline phosphatase alters the thio effect but not the transition state for phosphoryl transfer. Implications for the interpretation of thio effects in reactions of phosphatases.
    Holtz KM; Catrina IE; Hengge AC; Kantrowitz ER
    Biochemistry; 2000 Aug; 39(31):9451-8. PubMed ID: 10924140
    [TBL] [Abstract][Full Text] [Related]  

  • 6. Synthesis of tripeptides as potent Yersinia protein tyrosine phosphatase inhibitors.
    Lee K; Boovanahalli SK; Nam KY; Kang SU; Lee M; Phan J; Wu L; Waugh DS; Zhang ZY; No KT; Lee JJ; Burke TR
    Bioorg Med Chem Lett; 2005 Sep; 15(18):4037-42. PubMed ID: 16039123
    [TBL] [Abstract][Full Text] [Related]  

  • 7. Peptidic alpha-ketocarboxylic acids and sulfonamides as inhibitors of protein tyrosine phosphatases.
    Chen YT; Xie J; Seto CT
    J Org Chem; 2003 May; 68(10):4123-5. PubMed ID: 12737607
    [TBL] [Abstract][Full Text] [Related]  

  • 8. A targeted library of small-molecule, tyrosine, and dual-specificity phosphatase inhibitors derived from a rational core design and random side chain variation.
    Rice RL; Rusnak JM; Yokokawa F; Yokokawa S; Messner DJ; Boynton AL; Wipf P; Lazo JS
    Biochemistry; 1997 Dec; 36(50):15965-74. PubMed ID: 9398331
    [TBL] [Abstract][Full Text] [Related]  

  • 9. Discovery of protein phosphatase 2C inhibitors by virtual screening.
    Rogers JP; Beuscher AE; Flajolet M; McAvoy T; Nairn AC; Olson AJ; Greengard P
    J Med Chem; 2006 Mar; 49(5):1658-67. PubMed ID: 16509582
    [TBL] [Abstract][Full Text] [Related]  

  • 10. Structure based design of a series of potent and selective non peptidic PTP-1B inhibitors.
    Lau CK; Bayly CI; Gauthier JY; Li CS; Therien M; Asante-Appiah E; Cromlish W; Boie Y; Forghani F; Desmarais S; Wang Q; Skorey K; Waddleton D; Payette P; Ramachandran C; Kennedy BP; Scapin G
    Bioorg Med Chem Lett; 2004 Feb; 14(4):1043-8. PubMed ID: 15013020
    [TBL] [Abstract][Full Text] [Related]  

  • 11. Synthesis and biological evaluation of alpha,alpha-difluorobenzylphosphonic acid derivatives as small molecular inhibitors of protein-tyrosine phosphatase 1B.
    Yokomatsu T; Murano T; Umesue I; Soeda S; Shimeno H; Shibuya S
    Bioorg Med Chem Lett; 1999 Feb; 9(4):529-32. PubMed ID: 10098656
    [TBL] [Abstract][Full Text] [Related]  

  • 12. The most potent organophosphorus inhibitors of leucine aminopeptidase. Structure-based design, chemistry, and activity.
    Grembecka J; Mucha A; Cierpicki T; Kafarski P
    J Med Chem; 2003 Jun; 46(13):2641-55. PubMed ID: 12801228
    [TBL] [Abstract][Full Text] [Related]  

  • 13. Investigations of linker structure on the potency of a series of bidentate protein tyrosine phosphatase inhibitors.
    Xie J; Seto CT
    Bioorg Med Chem; 2005 Apr; 13(8):2981-91. PubMed ID: 15781408
    [TBL] [Abstract][Full Text] [Related]  

  • 14. Synthesis and characterization of a novel class of protein tyrosine phosphatase inhibitors.
    Ibrahimi OA; Wu L; Zhao K; Zhang ZY
    Bioorg Med Chem Lett; 2000 Mar; 10(5):457-60. PubMed ID: 10743947
    [TBL] [Abstract][Full Text] [Related]  

  • 15. [Calix[4]arene methylenebisphosphonic acids: the features of alkaline phosphatases inhibition].
    Muzychka OV; Tanchuk VIu; Vovk AI; Muravĭova IV; Cherenok SO; Kal'chenko VI; Kukhar VP
    Ukr Biokhim Zh (1999); 2007; 79(6):26-33. PubMed ID: 18712108
    [TBL] [Abstract][Full Text] [Related]  

  • 16. Inhibition of phosphatase activity by positively-charged cyclodextrins.
    Ghosh M; Sanders TC; Zhang R; Seto CT
    Org Lett; 1999 Dec; 1(12):1945-8. PubMed ID: 10836052
    [TBL] [Abstract][Full Text] [Related]  

  • 17. Is RK-682 a promiscuous enzyme inhibitor? Synthesis and in vitro evaluation of protein tyrosine phosphatase inhibition of racemic RK-682 and analogues.
    Carneiro VM; Trivella DB; Scorsato V; Beraldo VL; Dias MP; Sobreira TJ; Aparicio R; Pilli RA
    Eur J Med Chem; 2015 Jun; 97():42-54. PubMed ID: 25938987
    [TBL] [Abstract][Full Text] [Related]  

  • 18. Mechanistic studies of protein tyrosine phosphatases YopH and Cdc25A with m-nitrobenzyl phosphate.
    McCain DF; Grzyska PK; Wu L; Hengge AC; Zhang ZY
    Biochemistry; 2004 Jun; 43(25):8256-64. PubMed ID: 15209522
    [TBL] [Abstract][Full Text] [Related]  

  • 19. Synthesis and biological evaluation of cytostatin analogues.
    Bialy L; Waldmann H
    Chem Commun (Camb); 2003 Aug; (15):1872-3. PubMed ID: 12932009
    [TBL] [Abstract][Full Text] [Related]  

  • 20. Quinoxalinylurea derivatives as a novel class of JSP-1 inhibitors.
    Zhang L; Qiu B; Xiong B; Li X; Li J; Wang X; Li J; Shen J
    Bioorg Med Chem Lett; 2007 Apr; 17(8):2118-22. PubMed ID: 17303416
    [TBL] [Abstract][Full Text] [Related]  

    [Next]    [New Search]
    of 6.