116 related articles for article (PubMed ID: 12941292)
1. Novel bisubstrate analog inhibitors of serotonin N-acetyltransferase: the importance of being neutral.
Zheng W; Cole PA
Bioorg Chem; 2003 Oct; 31(5):398-411. PubMed ID: 12941292
[TBL] [Abstract][Full Text] [Related]
2. X-ray crystallographic studies of serotonin N-acetyltransferase catalysis and inhibition.
Wolf E; De Angelis J; Khalil EM; Cole PA; Burley SK
J Mol Biol; 2002 Mar; 317(2):215-24. PubMed ID: 11902838
[TBL] [Abstract][Full Text] [Related]
3. Design, synthesis and in vitro evaluation of novel derivatives as serotonin N-acetyltransferase inhibitors.
Beaurain N; Mésangeau C; Chavatte P; Ferry G; Audinot V; Boutin JA; Delagrange P; Bennejean C; Yous S
J Enzyme Inhib Med Chem; 2002 Dec; 17(6):409-14. PubMed ID: 12683677
[TBL] [Abstract][Full Text] [Related]
4. Mechanistic studies on the alkyltransferase activity of serotonin N-acetyltransferase.
Zheng W; Scheibner KA; Ho AK; Cole PA
Chem Biol; 2001 Apr; 8(4):379-89. PubMed ID: 11325593
[TBL] [Abstract][Full Text] [Related]
5. Bisubstrate ketone analogues as serotonin N-acetyltransferase inhibitors.
Kim CM; Cole PA
J Med Chem; 2001 Jul; 44(15):2479-85. PubMed ID: 11448230
[TBL] [Abstract][Full Text] [Related]
6. Investigation of the roles of catalytic residues in serotonin N-acetyltransferase.
Scheibner KA; De Angelis J; Burley SK; Cole PA
J Biol Chem; 2002 May; 277(20):18118-26. PubMed ID: 11884405
[TBL] [Abstract][Full Text] [Related]
7. Serotonin N-acetyltransferase: mechanism and inhibition.
Zheng W; Cole PA
Curr Med Chem; 2002 Jun; 9(12):1187-99. PubMed ID: 12052171
[TBL] [Abstract][Full Text] [Related]
8. Design, synthesis and in vitro evaluation of novel benzo[b]thiophene derivatives as serotonin N-acetyltransferase (AANAT) inhibitors.
Mesangeau C; Yous S; Chavatte P; Ferry G; Audinot V; Boutin JA; Delagrange P; Bennejean C; Renard P; Lesieur D
J Enzyme Inhib Med Chem; 2003 Apr; 18(2):119-25. PubMed ID: 12943195
[TBL] [Abstract][Full Text] [Related]
9. De novo discovery of serotonin N-acetyltransferase inhibitors.
Szewczuk LM; Saldanha SA; Ganguly S; Bowers EM; Javoroncov M; Karanam B; Culhane JC; Holbert MA; Klein DC; Abagyan R; Cole PA
J Med Chem; 2007 Nov; 50(22):5330-8. PubMed ID: 17924613
[TBL] [Abstract][Full Text] [Related]
10. New substrate analogues of human serotonin N-acetyltransferase produce in situ specific and potent inhibitors.
Ferry G; Ubeaud C; Mozo J; Péan C; Hennig P; Rodriguez M; Scoul C; Bonnaud A; Nosjean O; Galizzi JP; Delagrange P; Renard P; Volland JP; Yous S; Lesieur D; Boutin JA
Eur J Biochem; 2004 Jan; 271(2):418-28. PubMed ID: 14717709
[TBL] [Abstract][Full Text] [Related]
11. Indoleamine analogs as probes of the substrate selectivity and catalytic mechanism of serotonin N-acetyltransferase.
Khalil EM; De Angelis J; Cole PA
J Biol Chem; 1998 Nov; 273(46):30321-7. PubMed ID: 9804794
[TBL] [Abstract][Full Text] [Related]
12. The structural basis of ordered substrate binding by serotonin N-acetyltransferase: enzyme complex at 1.8 A resolution with a bisubstrate analog.
Hickman AB; Namboodiri MA; Klein DC; Dyda F
Cell; 1999 Apr; 97(3):361-9. PubMed ID: 10319816
[TBL] [Abstract][Full Text] [Related]
13. Characterization and regulation of a CHO cell line stably expressing human serotonin N-acetyltransferase (EC 2.3.1.87).
Ferry G; Mozo J; Ubeaud C; Berger S; Bertrand M; Try A; Beauverger P; Mesangeau C; Delagrange P; Boutin JA
Cell Mol Life Sci; 2002 Aug; 59(8):1395-405. PubMed ID: 12363042
[TBL] [Abstract][Full Text] [Related]
14. Synthesis and structure-activity relationships of truncated bisubstrate inhibitors of aminoglycoside 6'-N-acetyltransferases.
Gao F; Yan X; Shakya T; Baettig OM; Ait-Mohand-Brunet S; Berghuis AM; Wright GD; Auclair K
J Med Chem; 2006 Aug; 49(17):5273-81. PubMed ID: 16913716
[TBL] [Abstract][Full Text] [Related]
15. Mechanism-based inhibition of the melatonin rhythm enzyme: pharmacologic exploitation of active site functional plasticity.
Khalil EM; De Angelis J; Ishii M; Cole PA
Proc Natl Acad Sci U S A; 1999 Oct; 96(22):12418-23. PubMed ID: 10535937
[TBL] [Abstract][Full Text] [Related]
16. Crystal structure of a GCN5-related N-acetyltransferase: Serratia marcescens aminoglycoside 3-N-acetyltransferase.
Wolf E; Vassilev A; Makino Y; Sali A; Nakatani Y; Burley SK
Cell; 1998 Aug; 94(4):439-49. PubMed ID: 9727487
[TBL] [Abstract][Full Text] [Related]
17. Melatonin synthesis: arylalkylamine N-acetyltransferases in trout retina and pineal organ are different.
Benyassi A; Schwartz C; Coon SL; Klein DC; Falcón J
Neuroreport; 2000 Feb; 11(2):255-8. PubMed ID: 10674465
[TBL] [Abstract][Full Text] [Related]
18. Substrate specificity and inhibition studies of human serotonin N-acetyltransferase.
Ferry G; Loynel A; Kucharczyk N; Bertin S; Rodriguez M; Delagrange P; Galizzi JP; Jacoby E; Volland JP; Lesieur D; Renard P; Canet E; Fauchère JL; Boutin JA
J Biol Chem; 2000 Mar; 275(12):8794-805. PubMed ID: 10722724
[TBL] [Abstract][Full Text] [Related]
19. The arylalkylamine-N-acetyltransferase (AANAT) acetylates dopamine in the digestive tract of goldfish: a role in intestinal motility.
Nisembaum LG; Tinoco AB; Moure AL; Alonso Gómez AL; Delgado MJ; Valenciano AI
Neurochem Int; 2013 May; 62(6):873-80. PubMed ID: 23466408
[TBL] [Abstract][Full Text] [Related]
20. Serotonin metabolism in rat skin: characterization by liquid chromatography-mass spectrometry.
Semak I; Korik E; Naumova M; Wortsman J; Slominski A
Arch Biochem Biophys; 2004 Jan; 421(1):61-6. PubMed ID: 14678785
[TBL] [Abstract][Full Text] [Related]
[Next] [New Search]
