These tools will no longer be maintained as of December 31, 2024. Archived website can be found here. PubMed4Hh GitHub repository can be found here. Contact NLM Customer Service if you have questions.
2. Substitution of aromatic and nonaromatic amino acids for the Phe3 residue in the delta-selective opioid peptide deltorphin I: effects on binding affinity and selectivity. Heyl DL; Schmitter SJ; Bouzit H; Johnson TW; Hepp AM; Kurtz KR; Mousigian C Int J Pept Protein Res; 1994 Nov; 44(5):420-6. PubMed ID: 7896499 [TBL] [Abstract][Full Text] [Related]
3. Design and synthesis of 1-aminocycloalkane-1-carboxylic acid-substituted deltorphin analogues: unique delta and mu opioid activity in modified peptides. Breveglieri A; Guerrini R; Salvadori S; Bianchi C; Bryant SD; Attila M; Lazarus LH J Med Chem; 1996 Feb; 39(3):773-80. PubMed ID: 8576920 [TBL] [Abstract][Full Text] [Related]
4. Differential stereochemical requirements of mu vs. delta opioid receptors for ligand binding and signal transduction: development of a class of potent and highly delta-selective peptide antagonists. Schiller PW; Nguyen TM; Weltrowska G; Wilkes BC; Marsden BJ; Lemieux C; Chung NN Proc Natl Acad Sci U S A; 1992 Dec; 89(24):11871-5. PubMed ID: 1334552 [TBL] [Abstract][Full Text] [Related]
5. Synthesis and activity profiles of novel cyclic opioid peptide monomers and dimers. Schiller PW; Nguyen TM; Lemieux C; Maziak LA J Med Chem; 1985 Dec; 28(12):1766-71. PubMed ID: 2999401 [TBL] [Abstract][Full Text] [Related]
6. Evolution of the Dmt-Tic pharmacophore: N-terminal methylated derivatives with extraordinary delta opioid antagonist activity. Salvadori S; Balboni G; Guerrini R; Tomatis R; Bianchi C; Bryant SD; Cooper PS; Lazarus LH J Med Chem; 1997 Sep; 40(19):3100-8. PubMed ID: 9301674 [TBL] [Abstract][Full Text] [Related]
7. Bioactivity of new mu and delta opioid peptides. Capasso A Med Chem; 2007 Sep; 3(5):480-7. PubMed ID: 17897075 [TBL] [Abstract][Full Text] [Related]
8. Structure-activity relationships of dermorphin analogues containing N-substituted amino acids in the 2-position of the peptide sequence. Schmidt R; Kálmán A; Chung NN; Lemieux C; Horváth C; Schiller PW Int J Pept Protein Res; 1995 Jul; 46(1):47-55. PubMed ID: 7558596 [TBL] [Abstract][Full Text] [Related]
9. Development of a model for the delta opioid receptor pharmacophore. 1. Conformationally restricted Tyr1 replacements in the cyclic delta receptor selective tetrapeptide Tyr-c[D-Cys-Phe-D-Pen]OH (JOM-13). Mosberg HI; Lomize AL; Wang C; Kroona H; Heyl DL; Sobczyk-Kojiro K; Ma W; Mousigian C; Porreca F J Med Chem; 1994 Dec; 37(25):4371-83. PubMed ID: 7996549 [TBL] [Abstract][Full Text] [Related]
10. Phe3-substituted analogues of deltorphin C. Spatial conformation and topography of the aromatic ring in peptide recognition by delta opioid receptors. Salvadori S; Bryant SD; Bianchi C; Balboni G; Scaranari V; Attila M; Lazarus LH J Med Chem; 1993 Nov; 36(24):3748-56. PubMed ID: 8254604 [TBL] [Abstract][Full Text] [Related]
12. Conformational restriction of the phenylalanine residue in a cyclic opioid peptide analogue: effects on receptor selectivity and stereospecificity. Schiller PW; Weltrowska G; Nguyen TM; Lemieux C; Chung NN; Marsden BJ; Wilkes BC J Med Chem; 1991 Oct; 34(10):3125-32. PubMed ID: 1656045 [TBL] [Abstract][Full Text] [Related]
13. Structural modifications of the N-terminal tetrapeptide segment of [D-Ala2]deltorphin I: effects on opioid receptor affinities and activities in vitro and on antinociceptive potency. Schmidt R; Menard D; Mrestani-Klaus C; Chung NN; Lemieux C; Schiller PW Peptides; 1997; 18(10):1615-21. PubMed ID: 9437724 [TBL] [Abstract][Full Text] [Related]
14. Synthesis, opioid receptor binding, and bioassay of naltrindole analogues substituted in the indolic benzene moiety. Ananthan S; Johnson CA; Carter RL; Clayton SD; Rice KC; Xu H; Davis P; Porreca F; Rothman RB J Med Chem; 1998 Jul; 41(15):2872-81. PubMed ID: 9667975 [TBL] [Abstract][Full Text] [Related]
15. Opioid antagonist properties of the highly delta-receptor-selective BOC-Tyr-Pro-Gly-Phe-Leu-Thr (OtBu) peptide and of its Phe1 and Mel1 analogues. Rónai AZ; Magyar A; Orosz G; Borsodi A; Benyhe S; Tóth G; Makó E; Kátay E; Babka E; Medzihradszky K Arch Int Pharmacodyn Ther; 1995; 330(3):361-9. PubMed ID: 8836454 [TBL] [Abstract][Full Text] [Related]
16. Helix-inducing alpha-aminoisobutyric acid in opioid mimetic deltorphin C analogues. Bryant SD; Guerrini R; Salvadori S; Bianchi C; Tomatis R; Attila M; Lazarus LH J Med Chem; 1997 Aug; 40(16):2579-87. PubMed ID: 9258365 [TBL] [Abstract][Full Text] [Related]
17. Delta opioidmimetic antagonists: prototypes for designing a new generation of ultraselective opioid peptides. Salvadori S; Attila M; Balboni G; Bianchi C; Bryant SD; Crescenzi O; Guerrini R; Picone D; Tancredi T; Temussi PA Mol Med; 1995 Sep; 1(6):678-89. PubMed ID: 8529134 [TBL] [Abstract][Full Text] [Related]
18. Development of a model for the delta opioid receptor pharmacophore. 2. Conformationally restricted Phe3 replacements in the cyclic delta receptor selective tetrapeptide Tyr-c[D-Cys-Phe-D-Pen]OH (JOM-13). Mosberg HI; Omnaas JR; Lomize A; Heyl DL; Nordan I; Mousigian C; Davis P; Porreca F J Med Chem; 1994 Dec; 37(25):4384-91. PubMed ID: 7996550 [TBL] [Abstract][Full Text] [Related]
19. Opioid activity of dermenkephalin analogues in the guinea-pig myenteric plexus and the hamster vas deferens. Sagan S; Corbett AD; Amiche M; Delfour A; Nicolas P; Kosterlitz HW Br J Pharmacol; 1991 Oct; 104(2):428-32. PubMed ID: 1665735 [TBL] [Abstract][Full Text] [Related]
20. Agonist and antagonist profiles of [D-Ala2,Glu4]deltorphin and its [Cys4]- and [Ser4]-substituted derivatives: further evidence of opioid delta receptor multiplicity. Horan PJ; Wild KD; Misicka A; Lipkowski A; Haaseth RC; Hruby VJ; Weber SJ; Davis TP; Yamamura HI; Porreca F J Pharmacol Exp Ther; 1993 May; 265(2):896-902. PubMed ID: 8388462 [TBL] [Abstract][Full Text] [Related] [Next] [New Search]