BIOMARKERS

Molecular Biopsy of Human Tumors

- a resource for Precision Medicine *

102 related articles for article (PubMed ID: 1342833)

  • 1. Competitive parabolic inhibition of bovine trypsin by bis-benzamidines.
    Junqueira RG; Silva E; Mares-Guia M
    Braz J Med Biol Res; 1992; 25(9):873-87. PubMed ID: 1342833
    [TBL] [Abstract][Full Text] [Related]  

  • 2. A plausible identification of the secondary binding site in trypsin and trypsinogen.
    Andrade MH; Silva E; Mares-Guia M
    Braz J Med Biol Res; 1990; 23(12):1223-31. PubMed ID: 2136554
    [TBL] [Abstract][Full Text] [Related]  

  • 3. Tyrosine 151 is part of the substrate activation binding site of bovine trypsin. Identification by covalent labeling with p-diazoniumbenzamidine and kinetic characterization of Tyr-151-(p-benzamidino)-azo-beta-trypsin.
    Oliveira MG; Rogana E; Rosa JC; Reinhold BB; Andrade MH; Greene LJ; Mares-Guia M
    J Biol Chem; 1993 Dec; 268(36):26893-903. PubMed ID: 8262923
    [TBL] [Abstract][Full Text] [Related]  

  • 4. Structural binding evidence of the trypanocidal drugs berenil and pentacarinate active principles to a serine protease model.
    Perilo CS; Pereira MT; Santoro MM; Nagem RA
    Int J Biol Macromol; 2010 Jun; 46(5):502-11. PubMed ID: 20356563
    [TBL] [Abstract][Full Text] [Related]  

  • 5. Kinetic characterization of rat tissue kallikrein using N alpha-substituted arginine 4-nitroanilides and N alpha-benzoyl-L-arginine ethyl ester as substrates.
    Sousa MO; Rodrigues CV; Pena HB; Alvarenga MG; Machado-Coelho GL; Santoro MM; Juliano MA; Juliano L; Figueiredo AF
    Braz J Med Biol Res; 1996 Mar; 29(3):327-34. PubMed ID: 8736125
    [TBL] [Abstract][Full Text] [Related]  

  • 6. Thermodynamic evaluation and modeling of proton and water exchange associated with benzamidine and berenil binding to beta-trypsin.
    Pereira MT; Silva-Alves JM; Martins-José A; Lopes JC; Santoro MM
    Braz J Med Biol Res; 2005 Nov; 38(11):1593-601. PubMed ID: 16258627
    [TBL] [Abstract][Full Text] [Related]  

  • 7. Zymogen activation: effect of peptides sequentially related to the bovine beta-trypsin N-terminus on Kazal inhibitor and benzamidine binding to bovine trypsinogen.
    Ascenzi P; Coletta M; Amiconi G; Bolognesi M; Guarneri M; Menegatti E
    J Mol Recognit; 1988 Jun; 1(3):130-7. PubMed ID: 3273224
    [TBL] [Abstract][Full Text] [Related]  

  • 8. Mammalian tissue trypsin-like enzymes: substrate specificity and inhibitory potency of substituted isocoumarin mechanism-based inhibitors, benzamidine derivatives, and arginine fluoroalkyl ketone transition-state inhibitors.
    Kam CM; Hernandez MA; Patil GS; Ueda T; Simmons WH; Braganza VJ; Powers JC
    Arch Biochem Biophys; 1995 Feb; 316(2):808-14. PubMed ID: 7864637
    [TBL] [Abstract][Full Text] [Related]  

  • 9. Inhibition of bovine beta-trypsin, human alpha-thrombin and porcine pancreatic beta-kallikrein-B by benzamidine and its bis-, tris- and tetra-derivatives: thermodynamic and molecular modeling study.
    Menegatti E; Ferroni R; Nastruzzi C; Bortolotti F; Scalia S; Amiconi G; Bolognesi M; Coletta M; Onesti S; Fruttero R
    Farmaco; 1991 Nov; 46(11):1297-310. PubMed ID: 1811616
    [TBL] [Abstract][Full Text] [Related]  

  • 10. Kinetic mechanism of the inhibition of human urinary kallikrein by basic pancreatic trypsin inhibitor.
    Miranda TL; Ramos CH; Freire RT; Souza EP; Rogana E; Santoro MM; Figueiredo AF
    Braz J Med Biol Res; 1995 May; 28(5):505-12. PubMed ID: 8555969
    [TBL] [Abstract][Full Text] [Related]  

  • 11. Inhibition of enzymes of polyamine back-conversion by pentamidine and berenil.
    Libby PR; Porter CW
    Biochem Pharmacol; 1992 Aug; 44(4):830-2. PubMed ID: 1510731
    [TBL] [Abstract][Full Text] [Related]  

  • 12. Benzamidine as a spectroscopic probe for the primary specificity subsite of trypsin-like serine proteinases. A case for BPTI binding to bovine beta-trypsin.
    Ascenzi P; Bolognesi M; Guarneri M; Menegatti E; Amiconi G
    Mol Cell Biochem; 1984 Sep; 64(2):139-44. PubMed ID: 6390168
    [TBL] [Abstract][Full Text] [Related]  

  • 13. Structural and functional analyses of benzamidine-based inhibitors in complex with trypsin: implications for the inhibition of factor Xa, tPA, and urokinase.
    Renatus M; Bode W; Huber R; Stürzebecher J; Stubbs MT
    J Med Chem; 1998 Dec; 41(27):5445-56. PubMed ID: 9876114
    [TBL] [Abstract][Full Text] [Related]  

  • 14. N-[2,2-dimethyl-3-(N-(4-cyanobenzoyl)amino)nonanoyl]-L-phenylalanine ethyl ester as a stable ester-type inhibitor of chymotrypsin-like serine proteases: structural requirements for potent inhibition of alpha-chymotrypsin.
    Iijima K; Katada J; Yasuda E; Uno I; Hayashi Y
    J Med Chem; 1999 Jan; 42(2):312-23. PubMed ID: 9925737
    [TBL] [Abstract][Full Text] [Related]  

  • 15. The substituent effect on complex formation between alpha-trypsin and para-substituted benzamidinium ions: a thermodynamic study.
    Rogana E; Penha-Silva N; Mares-Guia M
    Braz J Med Biol Res; 1989; 22(10):1177-90. PubMed ID: 2638191
    [TBL] [Abstract][Full Text] [Related]  

  • 16. Demonstration that 1-trans-epoxysuccinyl-L-leucylamido-(4-guanidino) butane (E-64) is one of the most effective low Mr inhibitors of trypsin-catalysed hydrolysis. Characterization by kinetic analysis and by energy minimization and molecular dynamics simulation of the E-64-beta-trypsin complex.
    Sreedharan SK; Verma C; Caves LS; Brocklehurst SM; Gharbia SE; Shah HN; Brocklehurst K
    Biochem J; 1996 Jun; 316 ( Pt 3)(Pt 3):777-86. PubMed ID: 8670152
    [TBL] [Abstract][Full Text] [Related]  

  • 17. In-depth study of tripeptide-based alpha-ketoheterocycles as inhibitors of thrombin. Effective utilization of the S1' subsite and its implications to structure-based drug design.
    Costanzo MJ; Almond HR; Hecker LR; Schott MR; Yabut SC; Zhang HC; Andrade-Gordon P; Corcoran TW; Giardino EC; Kauffman JA; Lewis JM; de Garavilla L; Haertlein BJ; Maryanoff BE
    J Med Chem; 2005 Mar; 48(6):1984-2008. PubMed ID: 15771442
    [TBL] [Abstract][Full Text] [Related]  

  • 18. Highly selective mechanism-based thrombin inhibitors: structures of thrombin and trypsin inhibited with rigid peptidyl aldehydes.
    Krishnan R; Zhang E; Hakansson K; Arni RK; Tulinsky A; Lim-Wilby MS; Levy OE; Semple JE; Brunck TK
    Biochemistry; 1998 Sep; 37(35):12094-103. PubMed ID: 9724521
    [TBL] [Abstract][Full Text] [Related]  

  • 19. [Interaction between alpha-2 macroglobulin and trypsin with synthetic trypsin inhibitors].
    Krebs G
    Biochimie; 1979; 61(4):559-65. PubMed ID: 90529
    [TBL] [Abstract][Full Text] [Related]  

  • 20. Kinetic study of the effect of heparin on the amidase activity of trypsin, plasmin and urokinase.
    Yomtova VM; Stambolieva NA; Blagoev BM
    Thromb Haemost; 1983 Jun; 49(3):199-203. PubMed ID: 6224310
    [TBL] [Abstract][Full Text] [Related]  

    [Next]    [New Search]
    of 6.