166 related articles for article (PubMed ID: 14565305)
21. Characterization of the activation pathway of phosphoramidate triester prodrugs of stavudine and zidovudine.
Saboulard D; Naesens L; Cahard D; Salgado A; Pathirana R; Velazquez S; McGuigan C; De Clercq E; Balzarini J
Mol Pharmacol; 1999 Oct; 56(4):693-704. PubMed ID: 10496951
[TBL] [Abstract][Full Text] [Related]
22. Synthesis and anti-retroviral activity of O,O'-bis(3'-azido-2',3'-dideoxythymidin-5'-yl) phosphoramidate derivatives.
Kers I; Stawiński J; Girardet JL; Imbach JL; Périgaud C; Gosselin G; Aubertin AM
Nucleosides Nucleotides; 1999 Oct; 18(10):2317-25. PubMed ID: 10616733
[TBL] [Abstract][Full Text] [Related]
23. New 3'-azido-3'-deoxythymidin-5'-yl O-(omega-hydroxyalkyl) carbonate prodrugs: synthesis and anti-HIV evaluation.
Vlieghe P; Bihel F; Clerc T; Pannecouque C; Witvrouw M; De Clercq E; Salles JP; Chermann JC; Kraus JL
J Med Chem; 2001 Mar; 44(5):777-86. PubMed ID: 11262088
[TBL] [Abstract][Full Text] [Related]
24. Synthesis and anti-HIV activity of steroidal prodrugs of 3'-azido-3'-deoxythymidine (AZT).
Balagopala MI; Ollapally AP; Lee HJ
Cell Mol Biol (Noisy-le-grand); 1995; 41 Suppl 1():S1-7. PubMed ID: 8574137
[TBL] [Abstract][Full Text] [Related]
25. Synthesis of zidovudine prodrugs with broad-spectrum chemotherapeutic properties for the effective treatment of HIV/AIDS.
Sriram D; Srichakravarthy N; Bal TR; Yogeeswari P
Biomed Pharmacother; 2005 Sep; 59(8):452-5. PubMed ID: 16154314
[TBL] [Abstract][Full Text] [Related]
26. S-acyl-2-thioethyl aryl phosphotriester derivatives of AZT: synthesis, antiviral activity, and stability study.
Peyrottes S; Coussot G; Lefebvre I; Imbach JL; Gosselin G; Aubertin AM; Périgaud C
J Med Chem; 2003 Feb; 46(5):782-93. PubMed ID: 12593658
[TBL] [Abstract][Full Text] [Related]
27. Phosphoramidate and phosphate prodrugs of (-)-beta-D-(2R,4R)-dioxolane-thymine: synthesis, anti-HIV activity and stability studies.
Liang Y; Narayanasamy J; Schinazi RF; Chu CK
Bioorg Med Chem; 2006 Apr; 14(7):2178-89. PubMed ID: 16314108
[TBL] [Abstract][Full Text] [Related]
28. Brain targeting of anti-HIV nucleosides: synthesis and in vitro and in vivo studies of dihydropyridine derivatives of 3'-azido-2',3'-dideoxyuridine and 3'-azido-3'-deoxythymidine.
Chu CK; Bhadti VS; Doshi KJ; Etse JT; Gallo JM; Boudinot FD; Schinazi RF
J Med Chem; 1990 Aug; 33(8):2188-92. PubMed ID: 2374145
[TBL] [Abstract][Full Text] [Related]
29. Synthesis and in vitro activity of long-chain 5'-O-[(alkoxycarbonyl)phosphinyl]-3'-azido-3'-deoxythymidines against wild-type and AZT- and foscarnet-resistant strains of HIV-1.
Rosowsky A; Fu H; Pai N; Mellors J; Richman DD; Hostetler KY
J Med Chem; 1997 Aug; 40(16):2482-90. PubMed ID: 9258355
[TBL] [Abstract][Full Text] [Related]
30. AZT and AZT-monophosphate prodrugs incorporating HIV-protease substrate fragment: synthesis and evaluation as specific drug delivery systems.
Liotard JF; Mehiri M; Di Giorgio A; Boggetto N; Reboud-Ravaux M; Aubertin AM; Condom R; Patino N
Antivir Chem Chemother; 2006; 17(4):193-213. PubMed ID: 17066898
[TBL] [Abstract][Full Text] [Related]
31. Synthesis and anti-HIV evaluation of new acyclic phosphonate nucleotide analogues and their bis(SATE) derivatives.
Li H; Hong JH
Nucleosides Nucleotides Nucleic Acids; 2010 Aug; 29(8):581-90. PubMed ID: 20661812
[TBL] [Abstract][Full Text] [Related]
32. SATE (aryl) phosphotriester series. I. Synthesis and biological evaluation.
Peyrottes S; Gosselin G; Aubertin AM; Périgaud C
Nucleosides Nucleotides Nucleic Acids; 2003; 22(5-8):903-5. PubMed ID: 14565307
[TBL] [Abstract][Full Text] [Related]
33. S-Acyl-2-thioethyl aryl phosphotriester derivatives as mononucleotide prodrugs.
Schlienger N; Peyrottes S; Kassem T; Imbach JL; Gosselin G; Aubertin AM; Périgaud C
J Med Chem; 2000 Nov; 43(23):4570-4. PubMed ID: 11087582
[TBL] [Abstract][Full Text] [Related]
34. New 3'-azido-3'-deoxythymidin-5'-yl O-(4-hydroxyalkyl or -alkenyl or -alkylepoxide) carbonate prodrugs: synthesis and anti-HIV evaluation.
Vlieghe P; Clerc T; Pannecouque C; Witvrouw M; De Clercq E; Salles JP; Kraus JL
J Med Chem; 2001 Aug; 44(18):3014-21. PubMed ID: 11520210
[TBL] [Abstract][Full Text] [Related]
35. Design and synthesis of novel SATE derivatives of acyclic isocytosine and 9-deazaadenine C-nucleosides.
Liu LJ; Hong JH
Nucleosides Nucleotides Nucleic Acids; 2010 Mar; 29(3):257-66. PubMed ID: 20408056
[TBL] [Abstract][Full Text] [Related]
36. Synthesis and anti-HIV activity of beta-D-3'-azido-2',3'-unsaturated nucleosides and beta-D-3'-azido-3'-deoxyribofuranosylnucleosides.
Gadthula S; Chu CK; Schinazi RF
Nucleosides Nucleotides Nucleic Acids; 2005; 24(10-12):1707-27. PubMed ID: 16438043
[TBL] [Abstract][Full Text] [Related]
37. One-pot synthesis of an AZT boranophosphate conjugated with tyrosine: a potential prodrug candidate.
Li P; Shaw BR
Nucleosides Nucleotides Nucleic Acids; 2003; 22(5-8):699-701. PubMed ID: 14565257
[TBL] [Abstract][Full Text] [Related]
38. Self-assembled drug delivery systems. Part 4. In vitro/in vivo studies of the self-assemblies of cholesteryl-phosphonyl zidovudine.
Jin Y; Xing L; Tian Y; Li M; Gao C; Du L; Dong J; Chen H
Int J Pharm; 2009 Oct; 381(1):40-8. PubMed ID: 19646518
[TBL] [Abstract][Full Text] [Related]
39. Synthesis, anti-HIV activity, and resistance profiles of ribose modified nucleoside phosphonates.
Mackman RL; Boojamra CG; Prasad V; Zhang L; Lin KY; Petrakovsky O; Babusis D; Chen J; Douglas J; Grant D; Hui HC; Kim CU; Markevitch DY; Vela J; Ray A; Cihlar T
Bioorg Med Chem Lett; 2007 Dec; 17(24):6785-9. PubMed ID: 18029175
[TBL] [Abstract][Full Text] [Related]
40. Anti-HIV therapy with AZT prodrugs: AZT phosphonate derivatives, current state and prospects.
Khandazhinskaya A; Matyugina E; Shirokova E
Expert Opin Drug Metab Toxicol; 2010 Jun; 6(6):701-14. PubMed ID: 20380483
[TBL] [Abstract][Full Text] [Related]
[Previous] [Next] [New Search]
