These tools will no longer be maintained as of December 31, 2024. Archived website can be found here. PubMed4Hh GitHub repository can be found here. Contact NLM Customer Service if you have questions.


BIOMARKERS

Molecular Biopsy of Human Tumors

- a resource for Precision Medicine *

127 related articles for article (PubMed ID: 14604650)

  • 1. Aza-THIP and related analogues of THIP as GABA C antagonists.
    Krehan D; Frølund B; Ebert B; Nielsen B; Krogsgaard-Larsen P; Johnston GA; Chebib M
    Bioorg Med Chem; 2003 Nov; 11(23):4891-6. PubMed ID: 14604650
    [TBL] [Abstract][Full Text] [Related]  

  • 2. trans-4-Amino-2-methylbut-2-enoic acid (2-MeTACA) and (+/-)-trans-2-aminomethylcyclopropanecarboxylic acid ((+/-)-TAMP) can differentiate rat rho3 from human rho1 and rho2 recombinant GABA(C) receptors.
    Vien J; Duke RK; Mewett KN; Johnston GA; Shingai R; Chebib M
    Br J Pharmacol; 2002 Feb; 135(4):883-90. PubMed ID: 11861315
    [TBL] [Abstract][Full Text] [Related]  

  • 3. Characterization of GABA(A) receptor ligands in the rat cortical wedge preparation: evidence for action at extrasynaptic receptors?
    Ebert B; i Storustovu S; Mortensen M; Frølund B
    Br J Pharmacol; 2002 Sep; 137(1):1-8. PubMed ID: 12183325
    [TBL] [Abstract][Full Text] [Related]  

  • 4. GABA(A) agonists and partial agonists: THIP (Gaboxadol) as a non-opioid analgesic and a novel type of hypnotic.
    Krogsgaard-Larsen P; Frølund B; Liljefors T; Ebert B
    Biochem Pharmacol; 2004 Oct; 68(8):1573-80. PubMed ID: 15451401
    [TBL] [Abstract][Full Text] [Related]  

  • 5. pH-dependent actions of THIP and ZAPA on an ionotropic Drosophila melanogaster GABA receptor.
    Matsuda K; Hosie AM; Buckingham SD; Squire MD; Baylis HA; Sattelle DB
    Brain Res; 1996 Nov; 739(1-2):335-8. PubMed ID: 8955956
    [TBL] [Abstract][Full Text] [Related]  

  • 6. GABA(A) receptor ligands and their therapeutic potentials.
    Frølund B; Ebert B; Kristiansen U; Liljefors T; Krogsgaard-Larsen P
    Curr Top Med Chem; 2002 Aug; 2(8):817-32. PubMed ID: 12171573
    [TBL] [Abstract][Full Text] [Related]  

  • 7. 4,5,6,7-Tetrahydroisothiazolo[5,4-c]pyridin-3-ol and related analogues of THIP. Synthesis and biological activity.
    Krogsgaard-Larsen P; Mikkelsen H; Jacobsen P; Falch E; Curtis DR; Peet MJ; Leah JD
    J Med Chem; 1983 Jun; 26(6):895-900. PubMed ID: 6304315
    [TBL] [Abstract][Full Text] [Related]  

  • 8. Characterization of bicuculline/baclofen-insensitive (rho-like) gamma-aminobutyric acid receptors expressed in Xenopus oocytes. II. Pharmacology of gamma-aminobutyric acidA and gamma-aminobutyric acidB receptor agonists and antagonists.
    Woodward RM; Polenzani L; Miledi R
    Mol Pharmacol; 1993 Apr; 43(4):609-25. PubMed ID: 8386310
    [TBL] [Abstract][Full Text] [Related]  

  • 9. Induction of low-affinity GABAA receptors by the GABA-agonist THIP (4,5,6,7-tetrahydroisoxazolo[5,4-c]pyridin-3-ol) in cultured rat cerebellar granule cells is prevented by inhibition of polyamine biosynthesis.
    Abraham JH; Seiler N; Schousboe A
    J Neurosci Res; 1994 Dec; 39(6):656-62. PubMed ID: 7897701
    [TBL] [Abstract][Full Text] [Related]  

  • 10. Cytotoxic action of lindane in cerebellar granule neurons is mediated by interaction with inducible GABA(B) receptors.
    Vale C; Damgaard I; Suñol C; Rodríguez-Farré E; Schousboe A
    J Neurosci Res; 1998 May; 52(3):286-94. PubMed ID: 9590437
    [TBL] [Abstract][Full Text] [Related]  

  • 11. Evidence for inhibitory effect of the agonist gaboxadol at human alpha 1 beta 2 gamma 2S GABAA receptors.
    Smith M; Lindquist CE; Birnir B
    Eur J Pharmacol; 2003 Sep; 478(1):21-6. PubMed ID: 14555180
    [TBL] [Abstract][Full Text] [Related]  

  • 12. GABA(C) receptors as drug targets.
    Johnston GA; Chebib M; Hanrahan JR; Mewett KN
    Curr Drug Targets CNS Neurol Disord; 2003 Aug; 2(4):260-8. PubMed ID: 12871036
    [TBL] [Abstract][Full Text] [Related]  

  • 13. The effects of cyclopentane and cyclopentene analogues of GABA at recombinant GABA(C) receptors.
    Chebib M; Duke RK; Allan RD; Johnston GA
    Eur J Pharmacol; 2001 Nov; 430(2-3):185-92. PubMed ID: 11711030
    [TBL] [Abstract][Full Text] [Related]  

  • 14. Design and synthesis of a new series of 4-alkylated 3-isoxazolol GABA A antagonists.
    Frølund B; Tagmose L; Jørgensen AT; Kristiansen U; Stensbøl TB; Liljefors T; Krogsgaard-Larsen P
    Eur J Med Chem; 2003 Apr; 38(4):447-9. PubMed ID: 12750034
    [TBL] [Abstract][Full Text] [Related]  

  • 15. Activity of novel 4-PIOL analogues at human alpha 1 beta 2 gamma 2S GABA(A) receptors--correlation with hydrophobicity.
    Mortensen M; Frølund B; Jørgensen AT; Liljefors T; Krogsgaard-Larsen P; Ebert B
    Eur J Pharmacol; 2002 Sep; 451(2):125-32. PubMed ID: 12231381
    [TBL] [Abstract][Full Text] [Related]  

  • 16. Glycine antagonists structurally related to 4,5,6,7-tetrahydroisoxazolo [5,4-c]pyridin-3-ol inhibit binding of [3H]strychnine to rat brain membranes.
    Braestrup C; Nielsen M; Krogsgaard-Larsen P
    J Neurochem; 1986 Sep; 47(3):691-6. PubMed ID: 3016180
    [TBL] [Abstract][Full Text] [Related]  

  • 17. The binding of the GABA agonist [3H]THIP to rat brain synaptic membranes.
    Falch E; Krogsgaard-Larsen P
    J Neurochem; 1982 Apr; 38(4):1123-9. PubMed ID: 6278083
    [TBL] [Abstract][Full Text] [Related]  

  • 18. Effects of GABA(A) receptor partial agonists in primary cultures of cerebellar granule neurons and cerebral cortical neurons reflect different receptor subunit compositions.
    Hansen SL; Ebert B; Fjalland B; Kristiansen U
    Br J Pharmacol; 2001 Jun; 133(4):539-49. PubMed ID: 11399671
    [TBL] [Abstract][Full Text] [Related]  

  • 19. Pharmacology of GABA rho 1 and GABA alpha/beta receptors expressed in Xenopus oocytes and COS cells.
    Kusama T; Spivak CE; Whiting P; Dawson VL; Schaeffer JC; Uhl GR
    Br J Pharmacol; 1993 May; 109(1):200-6. PubMed ID: 8388298
    [TBL] [Abstract][Full Text] [Related]  

  • 20. Changes in extracellular K+ evoked by GABA, THIP and baclofen in the guinea-pig hippocampal slice.
    Barolet AW; Morris ME
    Exp Brain Res; 1991; 84(3):591-8. PubMed ID: 1650707
    [TBL] [Abstract][Full Text] [Related]  

    [Next]    [New Search]
    of 7.