These tools will no longer be maintained as of December 31, 2024. Archived website can be found here. PubMed4Hh GitHub repository can be found here. Contact NLM Customer Service if you have questions.
2. Antitumor agents. 3. Design, synthesis, and biological evaluation of new pyridoisoquinolindione and dihydrothienoquinolindione derivatives with potent cytotoxic activity. Bolognese A; Correale G; Manfra M; Lavecchia A; Mazzoni O; Novellino E; La Colla P; Sanna G; Loddo R J Med Chem; 2004 Feb; 47(4):849-58. PubMed ID: 14761187 [TBL] [Abstract][Full Text] [Related]
3. Substitution at the F-ring N-imide of the indolocarbazole antitumor drug NB-506 increases the cytotoxicity, DNA binding, and topoisomerase I inhibition activities. Bailly C; Qu X; Chaires JB; Colson P; Houssier C; Ohkubo M; Nishimura S; Yoshinari T J Med Chem; 1999 Jul; 42(15):2927-35. PubMed ID: 10425102 [TBL] [Abstract][Full Text] [Related]
4. Synthesis and biological evaluation of amino-substituted benzo[f]pyrido[4,3-b] and pyrido[3,4-b]quinoxalines: a new class of antineoplastic agents. Nguyen CH; Fan E; Riou JF; Bissery MC; Vrignaud P; Lavelle F; Bisagni E Anticancer Drug Des; 1995 Jun; 10(4):277-97. PubMed ID: 7786395 [TBL] [Abstract][Full Text] [Related]
5. Novel antitumor agent family of 1H-benzo[c,d]indol-2-one with flexible basic side chains: synthesis and biological evaluation. Yin H; Xu Y; Qian X Bioorg Med Chem; 2007 Feb; 15(3):1356-62. PubMed ID: 17129733 [TBL] [Abstract][Full Text] [Related]
6. Synthesis and cytotoxic activity of a new potential DNA bisintercalator: 1,4-Bis{3-[N-(4-chlorobenzo[g]phthalazin-1-yl)aminopropyl]}piperazine. Galisteo J; Navarro P; Campayo L; Yunta MJ; Gómez-Contreras F; Villa-Pulgarin JA; Sierra BG; Mollinedo F; Gonzalez J; Garcia-España E Bioorg Med Chem; 2010 Jul; 18(14):5301-9. PubMed ID: 20538470 [TBL] [Abstract][Full Text] [Related]
7. N-fused imidazoles as novel anticancer agents that inhibit catalytic activity of topoisomerase IIα and induce apoptosis in G1/S phase. Baviskar AT; Madaan C; Preet R; Mohapatra P; Jain V; Agarwal A; Guchhait SK; Kundu CN; Banerjee UC; Bharatam PV J Med Chem; 2011 Jul; 54(14):5013-30. PubMed ID: 21644529 [TBL] [Abstract][Full Text] [Related]
8. Functionalized and [a]-anellated carbazoles as potential B-DNA ligands: experimental studies of DNA binding and molecular modeling of intercalation complexes. Pindur U; Marotto A; Schulze E; Fischer G Pharmazie; 2000 Oct; 55(10):727-32. PubMed ID: 11082831 [TBL] [Abstract][Full Text] [Related]
9. Novel DNA intercalators without basic side chains as efficient antitumor agents: design, synthesis and evaluation of benzo-[c,d]-indol-malononitrile derivatives. Li X; Wang Q; Qing Y; Lin Y; Zhang Y; Qian X; Cui J Bioorg Med Chem; 2010 May; 18(9):3279-84. PubMed ID: 20385497 [TBL] [Abstract][Full Text] [Related]
10. Novel imidazo[1,2-a]naphthyridinic systems (part 1): synthesis, antiproliferative and DNA-intercalating activities. Andaloussi M; Moreau E; Masurier N; Lacroix J; Gaudreault RC; Chezal JM; El Laghdach A; Canitrot D; Debiton E; Teulade JC; Chavignon O Eur J Med Chem; 2008 Nov; 43(11):2505-17. PubMed ID: 18403058 [TBL] [Abstract][Full Text] [Related]
11. Design, synthesis, and biological evaluation of indenoisoquinoline topoisomerase I inhibitors featuring polyamine side chains on the lactam nitrogen. Nagarajan M; Xiao X; Antony S; Kohlhagen G; Pommier Y; Cushman M J Med Chem; 2003 Dec; 46(26):5712-24. PubMed ID: 14667224 [TBL] [Abstract][Full Text] [Related]
12. DNA binding to guide the development of tetrahydroindeno[1,2-b]pyrido[4,3,2-de]quinoline derivatives as cytotoxic agents. Catoen-Chackal S; Facompré M; Houssin R; Pommery N; Goossens JF; Colson P; Bailly C; Hénichart JP J Med Chem; 2004 Jul; 47(14):3665-73. PubMed ID: 15214793 [TBL] [Abstract][Full Text] [Related]
13. Highly stable phenanthridinium frameworks as a new class of tunable DNA binding agents with cytotoxic properties. Parenty AD; Smith LV; Guthrie KM; Long DL; Plumb J; Brown R; Cronin L J Med Chem; 2005 Jul; 48(14):4504-6. PubMed ID: 15999988 [TBL] [Abstract][Full Text] [Related]
14. Acenaphtho[1,2-b]pyrrole derivatives as new family of intercalators: various DNA binding geometry and interesting antitumor capacity. Zhang Z; Yang Y; Zhang D; Wang Y; Qian X; Liu F Bioorg Med Chem; 2006 Oct; 14(20):6962-70. PubMed ID: 16828559 [TBL] [Abstract][Full Text] [Related]
15. A novel ruthenium(II) arene based intercalator with potent anticancer activity. Ruiz J; Vicente C; de Haro C; Bautista D Dalton Trans; 2009 Jul; (26):5071-3. PubMed ID: 19562164 [TBL] [Abstract][Full Text] [Related]
16. Synthesis of mono- and bisdihydrodipyridopyrazines and assessment of their DNA binding and cytotoxic properties. Blanchard S; Rodriguez I; Tardy C; Baldeyrou B; Bailly C; Colson P; Houssier C; Léonce S; Kraus-Berthier L; Pfeiffer B; Renard P; Pierré A; Caubère P; Guillaumet G J Med Chem; 2004 Feb; 47(4):978-87. PubMed ID: 14761199 [TBL] [Abstract][Full Text] [Related]
17. 4-Hydroxymethyl-3-aminoacridine derivatives as a new family of anticancer agents. Charmantray F; Demeunynck M; Carrez D; Croisy A; Lansiaux A; Bailly C; Colson P J Med Chem; 2003 Mar; 46(6):967-77. PubMed ID: 12620073 [TBL] [Abstract][Full Text] [Related]
18. Design and synthesis of DNA-intercalating 9-fluoren-beta-O-glycosides as potential IFN-inducers, and antiviral and cytostatic agents. Alcaro S; Arena A; Neri S; Ottanà R; Ortuso F; Pavone B; Vigorita MG Bioorg Med Chem; 2004 Apr; 12(7):1781-91. PubMed ID: 15028268 [TBL] [Abstract][Full Text] [Related]
19. Design, synthesis and biological evaluation of new oligopyrrole carboxamides linked with tricyclic DNA-intercalators as potential DNA ligands or topoisomerase inhibitors. David-Cordonnier MH; Hildebrand MP; Baldeyrou B; Lansiaux A; Keuser C; Benzschawel K; Lemster T; Pindur U Eur J Med Chem; 2007 Jun; 42(6):752-71. PubMed ID: 17433851 [TBL] [Abstract][Full Text] [Related]
20. Amine-guanidine switch: a promising approach to improve DNA binding and antiproliferative activities. Ohara K; Smietana M; Restouin A; Mollard S; Borg JP; Collette Y; Vasseur JJ J Med Chem; 2007 Dec; 50(26):6465-75. PubMed ID: 18052116 [TBL] [Abstract][Full Text] [Related] [Next] [New Search]