339 related articles for article (PubMed ID: 15027875)
1. Novel endoperoxide antimalarials: synthesis, heme binding, and antimalarial activity.
Taylor DK; Avery TD; Greatrex BW; Tiekink ER; Macreadie IG; Macreadie PI; Humphries AD; Kalkanidis M; Fox EN; Klonis N; Tilley L
J Med Chem; 2004 Mar; 47(7):1833-9. PubMed ID: 15027875
[TBL] [Abstract][Full Text] [Related]
2. Synthesis and antimalarial activity of cyclic peroxides, 1,2,4,5, 7-pentoxocanes and 1,2,4,5-tetroxanes.
Kim HS; Shibata Y; Wataya Y; Tsuchiya K; Masuyama A; Nojima M
J Med Chem; 1999 Jul; 42(14):2604-9. PubMed ID: 10411480
[TBL] [Abstract][Full Text] [Related]
3. Comparison of the reactivity of antimalarial 1,2,4,5-tetraoxanes with 1,2,4-trioxolanes in the presence of ferrous iron salts, heme, and ferrous iron salts/phosphatidylcholine.
Bousejra-El Garah F; Wong MH; Amewu RK; Muangnoicharoen S; Maggs JL; Stigliani JL; Park BK; Chadwick J; Ward SA; O'Neill PM
J Med Chem; 2011 Oct; 54(19):6443-55. PubMed ID: 21888440
[TBL] [Abstract][Full Text] [Related]
4. Alkylation of natural endoperoxide G3-factor. Synthesis and antimalarial activity studies.
Najjar F; Gorrichon L; Baltas M; André-Barrès C; Vial H
Org Biomol Chem; 2005 May; 3(9):1612-4. PubMed ID: 15858637
[TBL] [Abstract][Full Text] [Related]
5. Synthesis and antimalarial activity of dihydroperoxides and tetraoxanes conjugated with bis(benzyl)acetone derivatives.
Franco LL; de Almeida MV; E Silva LF; Vieira PP; Pohlit AM; Valle MS
Chem Biol Drug Des; 2012 May; 79(5):790-7. PubMed ID: 22284812
[TBL] [Abstract][Full Text] [Related]
6. Synthesis and antiplasmodial activity of streptocyanine/peroxide and streptocyanine/4-aminoquinoline hybrid dyes.
Maether MP; Bernat V; Maturano M; André-Barrès C; Ladeira S; Valentin A; Vial H; Payrastre C
Org Biomol Chem; 2011 Nov; 9(21):7400-10. PubMed ID: 21897970
[TBL] [Abstract][Full Text] [Related]
7. Synthesis and antimalarial activity of side chain modified 4-aminoquinoline derivatives.
Solomon VR; Haq W; Srivastava K; Puri SK; Katti SB
J Med Chem; 2007 Jan; 50(2):394-8. PubMed ID: 17228883
[TBL] [Abstract][Full Text] [Related]
8. Synthesis and antiplasmodial activity of bicyclic dioxanes as simplified dihydroplakortin analogues.
Gemma S; Kunjir S; Coccone SS; Brindisi M; Moretti V; Brogi S; Novellino E; Basilico N; Parapini S; Taramelli D; Campiani G; Butini S
J Med Chem; 2011 Aug; 54(16):5949-53. PubMed ID: 21761935
[TBL] [Abstract][Full Text] [Related]
9. The structure-activity relationship of the antimalarial ozonide arterolane (OZ277).
Dong Y; Wittlin S; Sriraghavan K; Chollet J; Charman SA; Charman WN; Scheurer C; Urwyler H; Santo Tomas J; Snyder C; Creek DJ; Morizzi J; Koltun M; Matile H; Wang X; Padmanilayam M; Tang Y; Dorn A; Brun R; Vennerstrom JL
J Med Chem; 2010 Jan; 53(1):481-91. PubMed ID: 19924861
[TBL] [Abstract][Full Text] [Related]
10. Aminocyclopropanes as precursors of endoperoxides with antimalarial activity.
Madelaine C; Buriez O; Crousse B; Florent I; Grellier P; Retailleau P; Six Y
Org Biomol Chem; 2010 Dec; 8(24):5591-601. PubMed ID: 20938514
[TBL] [Abstract][Full Text] [Related]
11. Synthesis and heme-binding correlation with antimalarial activity of 3,6-bis-(omega-N,N-diethylaminoamyloxy)-4,5-difluoroxanthone.
Dodean RA; Kelly JX; Peyton D; Gard GL; Riscoe MK; Winter RW
Bioorg Med Chem; 2008 Feb; 16(3):1174-83. PubMed ID: 18023189
[TBL] [Abstract][Full Text] [Related]
12. Influence of stereoisomer of dispiro-1,2,4,5-tetraoxanes on their binding mode with heme and on antimalarial activity: molecular docking studies.
Tonmunphean S; Wijitkosoom A; Tantirungrotechai Y
Bioorg Med Chem; 2004 May; 12(9):2005-12. PubMed ID: 15080904
[TBL] [Abstract][Full Text] [Related]
13. Endoperoxide carbonyl falcipain 2/3 inhibitor hybrids: toward combination chemotherapy of malaria through a single chemical entity.
Gibbons P; Verissimo E; Araujo NC; Barton V; Nixon GL; Amewu RK; Chadwick J; Stocks PA; Biagini GA; Srivastava A; Rosenthal PJ; Gut J; Guedes RC; Moreira R; Sharma R; Berry N; Cristiano ML; Shone AE; Ward SA; O'Neill PM
J Med Chem; 2010 Nov; 53(22):8202-6. PubMed ID: 20979352
[TBL] [Abstract][Full Text] [Related]
14. Plasmodium falciparum endoplasmic reticulum-resident calcium binding protein is a possible target of synthetic antimalarial endoperoxides, N-89 and N-251.
Morita M; Sanai H; Hiramoto A; Sato A; Hiraoka O; Sakura T; Kaneko O; Masuyama A; Nojima M; Wataya Y; Kim HS
J Proteome Res; 2012 Dec; 11(12):5704-11. PubMed ID: 23061985
[TBL] [Abstract][Full Text] [Related]
15. Glycosyl hydroperoxides: a new class of potential antimalarial agents.
Szechner B; Jaromin A; Parapini S; Basilico N; Grzeszczyk B; Furman B; Chmielewski M
Bioorg Med Chem; 2015 Jul; 23(13):3033-9. PubMed ID: 26022082
[TBL] [Abstract][Full Text] [Related]
16. Synthesis and evaluation of new antimalarial phenylurenyl chalcone derivatives.
Domínguez JN; León C; Rodrigues J; Gamboa de Domínguez N; Gut J; Rosenthal PJ
J Med Chem; 2005 May; 48(10):3654-8. PubMed ID: 15887974
[TBL] [Abstract][Full Text] [Related]
17. Synthesis of ring-substituted 4-aminoquinolines and evaluation of their antimalarial activities.
Madrid PB; Sherrill J; Liou AP; Weisman JL; Derisi JL; Guy RK
Bioorg Med Chem Lett; 2005 Feb; 15(4):1015-8. PubMed ID: 15686903
[TBL] [Abstract][Full Text] [Related]
18. Endoperoxide derivatives from marine organisms: 1,2-dioxanes of the plakortin family as novel antimalarial agents.
Fattorusso C; Campiani G; Catalanotti B; Persico M; Basilico N; Parapini S; Taramelli D; Campagnuolo C; Fattorusso E; Romano A; Taglialatela-Scafati O
J Med Chem; 2006 Nov; 49(24):7088-94. PubMed ID: 17125261
[TBL] [Abstract][Full Text] [Related]
19. Artemisinin and a series of novel endoperoxide antimalarials exert early effects on digestive vacuole morphology.
del Pilar Crespo M; Avery TD; Hanssen E; Fox E; Robinson TV; Valente P; Taylor DK; Tilley L
Antimicrob Agents Chemother; 2008 Jan; 52(1):98-109. PubMed ID: 17938190
[TBL] [Abstract][Full Text] [Related]
20. Synthesis, antimalarial activity, and molecular modeling of tebuquine analogues.
O'Neill PM; Willock DJ; Hawley SR; Bray PG; Storr RC; Ward SA; Park BK
J Med Chem; 1997 Feb; 40(4):437-48. PubMed ID: 9046333
[TBL] [Abstract][Full Text] [Related]
[Next] [New Search]
