182 related articles for article (PubMed ID: 15070776)
1. Quantitative analysis of the formation and diffusion of A1-adenosine receptor-antagonist complexes in single living cells.
Briddon SJ; Middleton RJ; Cordeaux Y; Flavin FM; Weinstein JA; George MW; Kellam B; Hill SJ
Proc Natl Acad Sci U S A; 2004 Mar; 101(13):4673-8. PubMed ID: 15070776
[TBL] [Abstract][Full Text] [Related]
2. Application of fluorescence correlation spectroscopy to the measurement of agonist binding to a G-protein coupled receptor at the single cell level.
Briddon SJ; Middleton RJ; Yates AS; George MW; Kellam B; Hill SJ
Faraday Discuss; 2004; 126():197-207; discussion 245-54. PubMed ID: 14992407
[TBL] [Abstract][Full Text] [Related]
3. Antagonist selective modulation of adenosine A1 and A3 receptor pharmacology by the food dye Brilliant Black BN: evidence for allosteric interactions.
May LT; Briddon SJ; Hill SJ
Mol Pharmacol; 2010 Apr; 77(4):678-86. PubMed ID: 20086038
[TBL] [Abstract][Full Text] [Related]
4. Influence of fluorophore and linker composition on the pharmacology of fluorescent adenosine A1 receptor ligands.
Baker JG; Middleton R; Adams L; May LT; Briddon SJ; Kellam B; Hill SJ
Br J Pharmacol; 2010 Feb; 159(4):772-86. PubMed ID: 20105183
[TBL] [Abstract][Full Text] [Related]
5. Agonist-occupied A3 adenosine receptors exist within heterogeneous complexes in membrane microdomains of individual living cells.
Cordeaux Y; Briddon SJ; Alexander SP; Kellam B; Hill SJ
FASEB J; 2008 Mar; 22(3):850-60. PubMed ID: 17959910
[TBL] [Abstract][Full Text] [Related]
6. A1 adenosine receptor inhibition of cyclic AMP formation and radioligand binding in the guinea-pig cerebral cortex.
Alexander SP; Curtis AR; Kendall DA; Hill SJ
Br J Pharmacol; 1994 Dec; 113(4):1501-7. PubMed ID: 7889308
[TBL] [Abstract][Full Text] [Related]
7. Kinetic analysis of antagonist-occupied adenosine-A3 receptors within membrane microdomains of individual cells provides evidence of receptor dimerization and allosterism.
Corriden R; Kilpatrick LE; Kellam B; Briddon SJ; Hill SJ
FASEB J; 2014 Oct; 28(10):4211-22. PubMed ID: 24970394
[TBL] [Abstract][Full Text] [Related]
8. [3H]xanthine amine congener of 1,3-dipropyl-8-phenylxanthine: an antagonist radioligand for adenosine receptors.
Jacobson KA; Ukena D; Kirk KL; Daly JW
Proc Natl Acad Sci U S A; 1986 Jun; 83(11):4089-93. PubMed ID: 3012550
[TBL] [Abstract][Full Text] [Related]
9. Determination of adenosine A1 receptor agonist and antagonist pharmacology using Saccharomyces cerevisiae: implications for ligand screening and functional selectivity.
Stewart GD; Valant C; Dowell SJ; Mijaljica D; Devenish RJ; Scammells PJ; Sexton PM; Christopoulos A
J Pharmacol Exp Ther; 2009 Oct; 331(1):277-86. PubMed ID: 19641164
[TBL] [Abstract][Full Text] [Related]
10. Allosteric interactions across native adenosine-A3 receptor homodimers: quantification using single-cell ligand-binding kinetics.
May LT; Bridge LJ; Stoddart LA; Briddon SJ; Hill SJ
FASEB J; 2011 Oct; 25(10):3465-76. PubMed ID: 21715680
[TBL] [Abstract][Full Text] [Related]
11. Mass spectrometry-based ligand binding assays on adenosine A1 and A2A receptors.
Massink A; Holzheimer M; Hölscher A; Louvel J; Guo D; Spijksma G; Hankemeier T; IJzerman AP
Purinergic Signal; 2015 Dec; 11(4):581-94. PubMed ID: 26482925
[TBL] [Abstract][Full Text] [Related]
12. New fluorescent adenosine A1-receptor agonists that allow quantification of ligand-receptor interactions in microdomains of single living cells.
Middleton RJ; Briddon SJ; Cordeaux Y; Yates AS; Dale CL; George MW; Baker JG; Hill SJ; Kellam B
J Med Chem; 2007 Feb; 50(4):782-93. PubMed ID: 17249651
[TBL] [Abstract][Full Text] [Related]
13. Comparative pharmacology of human adenosine receptor subtypes - characterization of stably transfected receptors in CHO cells.
Klotz KN; Hessling J; Hegler J; Owman C; Kull B; Fredholm BB; Lohse MJ
Naunyn Schmiedebergs Arch Pharmacol; 1998 Jan; 357(1):1-9. PubMed ID: 9459566
[TBL] [Abstract][Full Text] [Related]
14. Evidence of spare A1-adenosine receptors in guinea pig atrioventricular node.
Dennis D; Jacobson K; Belardinelli L
Am J Physiol; 1992 Mar; 262(3 Pt 2):H661-71. PubMed ID: 1558173
[TBL] [Abstract][Full Text] [Related]
15. Evaluation of 18F-CPFPX, a novel adenosine A1 receptor ligand: in vitro autoradiography and high-resolution small animal PET.
Bauer A; Holschbach MH; Cremer M; Weber S; Boy C; Shah NJ; Olsson RA; Halling H; Coenen HH; Zilles K
J Nucl Med; 2003 Oct; 44(10):1682-9. PubMed ID: 14530487
[TBL] [Abstract][Full Text] [Related]
16. GPCR ligand dendrimer (GLiDe) conjugates: adenosine receptor interactions of a series of multivalent xanthine antagonists.
Kecskés A; Tosh DK; Wei Q; Gao ZG; Jacobson KA
Bioconjug Chem; 2011 Jun; 22(6):1115-27. PubMed ID: 21539392
[TBL] [Abstract][Full Text] [Related]
17. Coupling of a transfected human brain A1 adenosine receptor in CHO-K1 cells to calcium mobilisation via a pertussis toxin-sensitive mechanism.
Iredale PA; Alexander SP; Hill SJ
Br J Pharmacol; 1994 Apr; 111(4):1252-6. PubMed ID: 8032613
[TBL] [Abstract][Full Text] [Related]
18. A comparison of the antagonist affinities for the Gi- and Gs-coupled states of the human adenosine A1-receptor.
Baker JG; Hill SJ
J Pharmacol Exp Ther; 2007 Jan; 320(1):218-28. PubMed ID: 17018691
[TBL] [Abstract][Full Text] [Related]
19. Comparison of effects of MgCl2 and Gpp(NH)p on antagonist and agonist radioligand binding to adenosine A1 receptors.
Finlayson K; Maemoto T; Butcher SP; Sharkey J; Olverman HJ
Acta Pharmacol Sin; 2003 Aug; 24(8):729-40. PubMed ID: 12904270
[TBL] [Abstract][Full Text] [Related]
20. Synthesis and Pharmacological Evaluation of Identified and Putative Metabolites of the A
Holschbach MH; Bier D; Sihver W; Schulze A; Neumaier B
ChemMedChem; 2017 May; 12(10):770-784. PubMed ID: 28217962
[TBL] [Abstract][Full Text] [Related]
[Next] [New Search]
