125 related articles for article (PubMed ID: 15133253)
21. Beta-adrenoceptor subtype activities of trimetoquinol derivatives: biochemical studies on human beta-adrenoceptors expressed in chinese hamster ovary cells.
Konkar AA; Vansal SS; Shams G; Fraundorfer PF; Zheng WP; Nikulin VI; De Los Angeles J; Fertel RH; Miller DD; Feller DR
J Pharmacol Exp Ther; 1999 Nov; 291(2):875-83. PubMed ID: 10525112
[TBL] [Abstract][Full Text] [Related]
22. Agonist-directed trafficking of porcine alpha(2A)-adrenergic receptor signaling in Chinese hamster ovary cells: l-isoproterenol selectively activates G(s).
Brink CB; Wade SM; Neubig RR
J Pharmacol Exp Ther; 2000 Aug; 294(2):539-47. PubMed ID: 10900230
[TBL] [Abstract][Full Text] [Related]
23. The beta3-adrenoceptor agonist 4-[[(Hexylamino)carbonyl]amino]-N-[4-[2-[[(2S)-2-hydroxy-3-(4-hydroxyphenoxy)propyl]amino]ethyl]-phenyl]-benzenesulfonamide (L755507) and antagonist (S)-N-[4-[2-[[3-[3-(acetamidomethyl)phenoxy]-2-hydroxypropyl]amino]-ethyl]phenyl]benzenesulfonamide (L748337) activate different signaling pathways in Chinese hamster ovary-K1 cells stably expressing the human beta3-adrenoceptor.
Sato M; Hutchinson DS; Evans BA; Summers RJ
Mol Pharmacol; 2008 Nov; 74(5):1417-28. PubMed ID: 18684840
[TBL] [Abstract][Full Text] [Related]
24. Biochemical activities of trimetoquinol analogs at human beta(1)- and beta(3)-adrenergic receptors.
Konkar AA; Nikulin VI; De Los Angeles J; Hong SS; Fertel RH; Miller DD; Feller DR
Pharmacology; 2001 Jan; 62(1):45-55. PubMed ID: 11150922
[TBL] [Abstract][Full Text] [Related]
25. Beta 1- and beta 2-adrenergic receptors display subtype-selective coupling to Gs.
Green SA; Holt BD; Liggett SB
Mol Pharmacol; 1992 May; 41(5):889-93. PubMed ID: 1350321
[TBL] [Abstract][Full Text] [Related]
26. Agonist interactions with chimeric and mutant beta1- and beta3-adrenergic receptors: involvement of the seventh transmembrane region in conferring subtype specificity.
Granneman JG; Lahners KN; Zhai Y
Mol Pharmacol; 1998 May; 53(5):856-61. PubMed ID: 9584211
[TBL] [Abstract][Full Text] [Related]
27. Effects of (-)-RO363 at human atrial beta-adrenoceptor subtypes, the human cloned beta 3-adrenoceptor and rodent intestinal beta 3-adrenoceptors.
Molenaar P; Sarsero D; Arch JR; Kelly J; Henson SM; Kaumann AJ
Br J Pharmacol; 1997 Jan; 120(2):165-76. PubMed ID: 9117106
[TBL] [Abstract][Full Text] [Related]
28. 2-Amino-4-benzyl-4,5,6,7-tetrahydrothiazolo[5,4-c]pyridines: novel selective beta3-adrenoceptor agonists.
Zheng W; Nikulin VI; Konkar AA; Vansal SS; Shams G; Feller DR; Miller DD
J Med Chem; 1999 Jun; 42(12):2287-94. PubMed ID: 10377236
[TBL] [Abstract][Full Text] [Related]
29. L-750355, a human beta3-adrenoceptor agonist; in vitro pharmacology and profile of activity in vivo in the rhesus monkey.
Forrest MJ; Hom G; Bach T; Candelore MR; Cascieri MA; Strader C; Tota L; Fisher MH; Szumiloski J; Ok HO; Weber AE; Wyvratt M; Vicario P; Marko O; Deng L; Cioffe C; Hegarty-Friscino B; MacIntyre E
Eur J Pharmacol; 2000 Oct; 407(1-2):175-81. PubMed ID: 11050305
[TBL] [Abstract][Full Text] [Related]
30. Vibegron shows high selectivity and potent agonist activity for β3-adrenoceptors, irrespective of receptor density.
Yamamoto S; Kusabuka H; Matsuzawa A; Maruyama I; Yamazaki T
PLoS One; 2023; 18(9):e0290685. PubMed ID: 37656760
[TBL] [Abstract][Full Text] [Related]
31. Mouse beta 3a- and beta 3b-adrenoceptors expressed in Chinese hamster ovary cells display identical pharmacology but utilize distinct signalling pathways.
Hutchinson DS; Bengtsson T; Evans BA; Summers RJ
Br J Pharmacol; 2002 Apr; 135(8):1903-14. PubMed ID: 11959793
[TBL] [Abstract][Full Text] [Related]
32. Molecular and functional characteristics of β3-adrenoceptors in late pregnant mouse uterus: a comparison with β2-adrenoceptors.
Parida S; Uttam Singh T; Ravi Prakash V; Mishra SK
Eur J Pharmacol; 2013 Jan; 700(1-3):74-9. PubMed ID: 23219791
[TBL] [Abstract][Full Text] [Related]
33. Stereoselectivity for interactions of agonists and antagonists at mouse, rat and human beta3-adrenoceptors.
Popp BD; Hutchinson DS; Evans BA; Summers RJ
Eur J Pharmacol; 2004 Jan; 484(2-3):323-31. PubMed ID: 14744619
[TBL] [Abstract][Full Text] [Related]
34. Site-directed mutagenesis of the human beta3-adrenoceptor--transmembrane residues involved in ligand binding and signal transduction.
Gros J; Manning BS; Pietri-Rouxel F; Guillaume JL; Drumare MF; Strosberg AD
Eur J Biochem; 1998 Feb; 251(3):590-6. PubMed ID: 9490030
[TBL] [Abstract][Full Text] [Related]
35. beta(1)-Adrenoceptors compensate for beta(3)-adrenoceptors in ileum from beta(3)-adrenoceptor knock-out mice.
Hutchinson DS; Evans BA; Summers RJ
Br J Pharmacol; 2001 Jan; 132(2):433-42. PubMed ID: 11159692
[TBL] [Abstract][Full Text] [Related]
36. Characterization of mexiletine as an antagonist of beta-adrenoceptor in Chinese hamster ovary cells expressing cloned human beta-adrenoceptors.
Sakamoto K; Karikomi Y; Kubota Y; Nakahara T; Ishii K
Biochem Pharmacol; 2004 Mar; 67(5):815-22. PubMed ID: 15104234
[TBL] [Abstract][Full Text] [Related]
37. Enhanced inhibition of L-type Ca2+ current by beta3-adrenergic stimulation in failing rat heart.
Zhang ZS; Cheng HJ; Onishi K; Ohte N; Wannenburg T; Cheng CP
J Pharmacol Exp Ther; 2005 Dec; 315(3):1203-11. PubMed ID: 16135702
[TBL] [Abstract][Full Text] [Related]
38. Discovery of a potent, orally bioavailable beta(3) adrenergic receptor agonist, (R)-N-[4-[2-[[2-hydroxy-2-(3-pyridinyl)ethyl]amino]ethyl]phenyl]-4-[4 -[4-(trifluoromethyl)phenyl]thiazol-2-yl]benzenesulfonamide.
Mathvink RJ; Tolman JS; Chitty D; Candelore MR; Cascieri MA; Colwell LF; Deng L; Feeney WP; Forrest MJ; Hom GJ; MacIntyre DE; Miller RR; Stearns RA; Tota L; Wyvratt MJ; Fisher MH; Weber AE
J Med Chem; 2000 Oct; 43(21):3832-6. PubMed ID: 11052788
[TBL] [Abstract][Full Text] [Related]
39. Novel (4-piperidin-1-yl)-phenyl sulfonamides as potent and selective human beta(3) agonists.
Hu B; Ellingboe J; Han S; Largis E; Lim K; Malamas M; Mulvey R; Niu C; Oliphant A; Pelletier J; Singanallore T; Sum FW; Tillett J; Wong V
Bioorg Med Chem; 2001 Aug; 9(8):2045-59. PubMed ID: 11504641
[TBL] [Abstract][Full Text] [Related]
40. Functional and molecular characterization of beta-adrenoceptors in the internal anal sphincter.
Rathi S; Kazerounian S; Banwait K; Schulz S; Waldman SA; Rattan S
J Pharmacol Exp Ther; 2003 May; 305(2):615-24. PubMed ID: 12606629
[TBL] [Abstract][Full Text] [Related]
[Previous] [Next] [New Search]