These tools will no longer be maintained as of December 31, 2024. Archived website can be found here. PubMed4Hh GitHub repository can be found here. Contact NLM Customer Service if you have questions.
125 related articles for article (PubMed ID: 1515050)
1. N-substituted (aminomethyl)benzoate 21-esters of corticosteroids as water-soluble, solution-stable and biolabile prodrugs. Jensen E; Bundgaard H Acta Pharm Nord; 1992; 4(1):35-42. PubMed ID: 1515050 [TBL] [Abstract][Full Text] [Related]
2. Synthesis, enzymatic hydrolysis and physico-chemical properties of N-substituted 4-(aminomethyl)benzoate diester prodrugs of ganciclovir. Jensen E; Bundgaard H Acta Pharm Nord; 1991; 3(4):243-7. PubMed ID: 1781915 [TBL] [Abstract][Full Text] [Related]
3. Water-soluble, solution-stable, and biolabile N-substituted (aminomethyl)benzoate ester prodrugs of acyclovir. Bundgaard H; Jensen E; Falch E Pharm Res; 1991 Sep; 8(9):1087-93. PubMed ID: 1788153 [TBL] [Abstract][Full Text] [Related]
4. Kinetics of hydrolysis of indomethacin and indomethacin ester prodrugs in aqueous solution. Kahns AH; Jensen PB; Mørk N; Bundgaard H Acta Pharm Nord; 1989; 1(6):327-36. PubMed ID: 2624703 [TBL] [Abstract][Full Text] [Related]
5. Strategies in the design of solution-stable, water-soluble prodrugs I: a physical-organic approach to pro-moiety selection for 21-esters of corticosteroids. Anderson BD; Conradi RA; Knuth KE J Pharm Sci; 1985 Apr; 74(4):365-74. PubMed ID: 3998996 [TBL] [Abstract][Full Text] [Related]
6. Strategies in the design of solution-stable, water-soluble prodrugs III: influence of the pro-moiety on the bioconversion of 21-esters of corticosteroids. Anderson BD; Conradi RA; Spilman CH; Forbes AD J Pharm Sci; 1985 Apr; 74(4):382-7. PubMed ID: 3889274 [TBL] [Abstract][Full Text] [Related]
7. In vitro evaluation of quercetin-3-O-acyl esters as topical prodrugs. Montenegro L; Carbone C; Maniscalco C; Lambusta D; Nicolosi G; Ventura CA; Puglisi G Int J Pharm; 2007 May; 336(2):257-62. PubMed ID: 17257788 [TBL] [Abstract][Full Text] [Related]
8. Kinetics of the acid-catalyzed hydrolysis of acyclovir and an ester prodrug in aqueous solution. Jensen E; Bundgaard H Acta Pharm Nord; 1991; 3(3):147-50. PubMed ID: 1793509 [TBL] [Abstract][Full Text] [Related]
9. Development of water-soluble prodrugs of the HIV-1 protease inhibitor KNI-727: importance of the conversion time for higher gastrointestinal absorption of prodrugs based on spontaneous chemical cleavage. Sohma Y; Hayashi Y; Ito T; Matsumoto H; Kimura T; Kiso Y J Med Chem; 2003 Sep; 46(19):4124-35. PubMed ID: 12954064 [TBL] [Abstract][Full Text] [Related]
10. Strategies in the design of solution-stable, water-soluble prodrugs II: properties of micellar prodrugs of methylprednisolone. Anderson BD; Conradi RA; Knuth KE; Nail SL J Pharm Sci; 1985 Apr; 74(4):375-81. PubMed ID: 3998997 [TBL] [Abstract][Full Text] [Related]
11. Aminocarbonyloxymethyl ester prodrugs of flufenamic acid and diclofenac: suppressing the rearrangement pathway in aqueous media. Ribeiro L; Silva N; Iley J; Rautio J; Järvinen T; Mota-Filipe H; Moreira R; Mendes E Arch Pharm (Weinheim); 2007 Jan; 340(1):32-40. PubMed ID: 17206608 [TBL] [Abstract][Full Text] [Related]
12. Pre-formulation and chemical stability studies of penethamate, a benzylpenicillin ester prodrug, in aqueous vehicles. Jain R; Wu Z; Bork O; Tucker IG Drug Dev Ind Pharm; 2012 Jan; 38(1):55-63. PubMed ID: 21696334 [TBL] [Abstract][Full Text] [Related]
13. Synthesis and properties of N-nicotinoyl-2-(5-fluorouracil-1-yl)-D,L-glycine ester as a prodrug of 5-fluorouracil for rectal administration. Yang YW; Lee JS; Kim I; Jung YJ; Kim YM Eur J Pharm Biopharm; 2007 May; 66(2):260-7. PubMed ID: 17182232 [TBL] [Abstract][Full Text] [Related]
14. Synthesis, chemical and enzymatic hydrolysis, and bioavailability evaluation in rabbits of metronidazole amino acid ester prodrugs with enhanced water solubility. Mahfouz NM; Hassan MA J Pharm Pharmacol; 2001 Jun; 53(6):841-8. PubMed ID: 11428660 [TBL] [Abstract][Full Text] [Related]
15. Hydrolysis and rearrangement of phthalamic acid derivatives and assessment of their potential as prodrug forms for amines. Bundgaard H; Steffansen B Acta Pharm Nord; 1990; 2(5):333-42. PubMed ID: 2083038 [TBL] [Abstract][Full Text] [Related]
16. A water-soluble prodrug of cyclosporine A for ocular application: a stability study. Lallemand F; Perottet P; Felt-Baeyens O; Kloeti W; Philippoz F; Marfurt J; Besseghir K; Gurny R Eur J Pharm Sci; 2005 Sep; 26(1):124-9. PubMed ID: 15978789 [TBL] [Abstract][Full Text] [Related]
17. Prodrugs of thiabendazole with increased water-solubility. Nielsen LS; Bundgaard H; Falch E Acta Pharm Nord; 1992; 4(1):43-9. PubMed ID: 1515051 [TBL] [Abstract][Full Text] [Related]
18. Synthesis, characterization and stability of dendrimer prodrugs. Najlah M; Freeman S; Attwood D; D'Emanuele A Int J Pharm; 2006 Feb; 308(1-2):175-82. PubMed ID: 16384673 [TBL] [Abstract][Full Text] [Related]
19. Bioreversible quaternary N-acyloxymethyl derivatives of the tertiary amines bupivacaine and lidocaine--synthesis, aqueous solubility and stability in buffer, human plasma and simulated intestinal fluid. Nielsen AB; Buur A; Larsen C Eur J Pharm Sci; 2005 Apr; 24(5):433-40. PubMed ID: 15784333 [TBL] [Abstract][Full Text] [Related]
20. Dipeptide derivatives of AZT: synthesis, chemical stability, activation in human plasma, hPEPT1 affinity, and antiviral activity. Santos C; Morais J; Gouveia L; de Clercq E; Pannecouque C; Nielsen CU; Steffansen B; Moreira R; Gomes P ChemMedChem; 2008 Jun; 3(6):970-8. PubMed ID: 18389514 [TBL] [Abstract][Full Text] [Related] [Next] [New Search]