BIOMARKERS

Molecular Biopsy of Human Tumors

- a resource for Precision Medicine *

122 related articles for article (PubMed ID: 15341944)

  • 1. Synthesis and evaluation of 2-amino-8-alkoxy quinolines as MCHr1 antagonists. Part 3.
    Souers AJ; Wodka D; Gao J; Lewis JC; Vasudevan A; Brodjian S; Dayton B; Ogiela CA; Fry D; Hernandez LE; Marsh KC; Collins CA; Kym PR
    Bioorg Med Chem Lett; 2004 Oct; 14(19):4883-6. PubMed ID: 15341944
    [TBL] [Abstract][Full Text] [Related]  

  • 2. Synthesis and evaluation of 2-amino-8-alkoxy quinolines as MCHr1 antagonists. Part 2.
    Vasudevan A; Wodka D; Verzal MK; Souers AJ; Gao J; Brodjian S; Fry D; Dayton B; Marsh KC; Hernandez LE; Ogiela CA; Collins CA; Kym PR
    Bioorg Med Chem Lett; 2004 Oct; 14(19):4879-82. PubMed ID: 15341943
    [TBL] [Abstract][Full Text] [Related]  

  • 3. Synthesis and evaluation of 2-amino-8-alkoxy quinolines as MCHr1 antagonists. Part 1.
    Souers AJ; Wodka D; Gao J; Lewis JC; Vasudevan A; Gentles R; Brodjian S; Dayton B; Ogiela CA; Fry D; Hernandez LE; Marsh KC; Collins CA; Kym PR
    Bioorg Med Chem Lett; 2004 Oct; 14(19):4873-7. PubMed ID: 15341942
    [TBL] [Abstract][Full Text] [Related]  

  • 4. Identification of aminopiperidine benzamides as MCHr1 antagonists.
    Vasudevan A; Verzal MK; Wodka D; Souers AJ; Blackburn C; Che JL; Lai S; Brodjian S; Falls DH; Dayton BD; Govek E; Daniels T; Geddes B; Marsh KC; Hernandez LE; Collins CA; Kym PR
    Bioorg Med Chem Lett; 2005 Jul; 15(14):3412-6. PubMed ID: 15950463
    [TBL] [Abstract][Full Text] [Related]  

  • 5. Constrained 7-fluorocarboxychromone-4-aminopiperidine based Melanin-concentrating hormone receptor 1 antagonists: the effects of chirality on substituted indan-1-ylamines.
    Souers AJ; Iyengar RR; Judd AS; Beno DW; Gao J; Zhao G; Brune ME; Napier JJ; Mulhern MM; Lynch JK; Freeman JC; Wodka D; Chen CJ; Falls HD; Brodjian S; Dayton BD; Diaz GJ; Bush EN; Shapiro R; Droz BA; Knourek-Segel V; Hernandez LE; Marsh KC; Reilly RM; Sham HL; Collins CA; Kym PR
    Bioorg Med Chem Lett; 2007 Feb; 17(4):884-9. PubMed ID: 17188866
    [TBL] [Abstract][Full Text] [Related]  

  • 6. Synthesis and evaluation of urea-based indazoles as melanin-concentrating hormone receptor 1 antagonists for the treatment of obesity.
    Souers AJ; Gao J; Wodka D; Judd AS; Mulhern MM; Napier JJ; Brune ME; Bush EN; Brodjian SJ; Dayton BD; Shapiro R; Hernandez LE; Marsh KC; Sham HL; Collins CA; Kym PR
    Bioorg Med Chem Lett; 2005 Jun; 15(11):2752-7. PubMed ID: 15911251
    [TBL] [Abstract][Full Text] [Related]  

  • 7. Identification of 2-(4-benzyloxyphenyl)-N- [1-(2-pyrrolidin-1-yl-ethyl)-1H-indazol-6-yl]acetamide, an orally efficacious melanin-concentrating hormone receptor 1 antagonist for the treatment of obesity.
    Souers AJ; Gao J; Brune M; Bush E; Wodka D; Vasudevan A; Judd AS; Mulhern M; Brodjian S; Dayton B; Shapiro R; Hernandez LE; Marsh KC; Sham HL; Collins CA; Kym PR
    J Med Chem; 2005 Mar; 48(5):1318-21. PubMed ID: 15743174
    [TBL] [Abstract][Full Text] [Related]  

  • 8. 6-Acylamino-2-amino-4-methylquinolines as potent melanin-concentrating hormone 1 receptor antagonists: structure-activity exploration of eastern and western parts.
    Ulven T; Little PB; Receveur JM; Frimurer TM; Rist O; Nørregaard PK; Högberg T
    Bioorg Med Chem Lett; 2006 Feb; 16(4):1070-5. PubMed ID: 16289819
    [TBL] [Abstract][Full Text] [Related]  

  • 9. Melanin-concentrating hormone receptor 1 antagonists. Synthesis and structure-activity relationships of novel 3-(aminomethyl)quinolines.
    Kamata M; Yamashita T; Imaeda T; Tanaka T; Masada S; Kamaura M; Kasai S; Hara R; Sasaki S; Takekawa S; Asami A; Kaisho T; Suzuki N; Ashina S; Ogino H; Nakano Y; Nagisa Y; Kato K; Kato K; Ishihara Y
    J Med Chem; 2012 Mar; 55(5):2353-66. PubMed ID: 22309223
    [TBL] [Abstract][Full Text] [Related]  

  • 10. Screening for cardiovascular safety: a structure-activity approach for guiding lead selection of melanin concentrating hormone receptor 1 antagonists.
    Kym PR; Souers AJ; Campbell TJ; Lynch JK; Judd AS; Iyengar R; Vasudevan A; Gao J; Freeman JC; Wodka D; Mulhern M; Zhao G; Wagaw SH; Napier JJ; Brodjian S; Dayton BD; Reilly RM; Segreti JA; Fryer RM; Preusser LC; Reinhart GA; Hernandez L; Marsh KC; Sham HL; Collins CA; Polakowski JS
    J Med Chem; 2006 Apr; 49(7):2339-52. PubMed ID: 16570930
    [TBL] [Abstract][Full Text] [Related]  

  • 11. Discovery of novel, orally available benzimidazoles as melanin concentrating hormone receptor 1 (MCHR1) antagonists.
    Sasmal PK; Sasmal S; Rao PT; Venkatesham B; Roshaiah M; Abbineni C; Khanna I; Jadhav VP; Suresh J; Talwar R; Muzeeb S; Receveur JM; Frimurer TM; Rist Ø; Elster L; Högberg T
    Bioorg Med Chem Lett; 2010 Sep; 20(18):5443-8. PubMed ID: 20724156
    [TBL] [Abstract][Full Text] [Related]  

  • 12. Discovery of imidazo[1,2-a]pyridines as potent MCH1R antagonists.
    Kishino H; Moriya M; Sakuraba S; Sakamoto T; Takahashi H; Suzuki T; Moriya R; Ito M; Iwaasa H; Takenaga N; Ishihara A; Kanatani A; Sato N; Fukami T
    Bioorg Med Chem Lett; 2009 Aug; 19(16):4589-93. PubMed ID: 19615899
    [TBL] [Abstract][Full Text] [Related]  

  • 13. Aminopiperidine indazoles as orally efficacious melanin concentrating hormone receptor-1 antagonists.
    Vasudevan A; Souers AJ; Freeman JC; Verzal MK; Gao J; Mulhern MM; Wodka D; Lynch JK; Engstrom KM; Wagaw SH; Brodjian S; Dayton B; Falls DH; Bush E; Brune M; Shapiro RD; Marsh KC; Hernandez LE; Collins CA; Kym PR
    Bioorg Med Chem Lett; 2005 Dec; 15(23):5293-7. PubMed ID: 16203136
    [TBL] [Abstract][Full Text] [Related]  

  • 14. 6-(4-chlorophenyl)-3-substituted-thieno[3,2-d]pyrimidin-4(3H)-one-based melanin-concentrating hormone receptor 1 antagonist.
    Tavares FX; Al-Barazanji KA; Bishop MJ; Britt CS; Carlton DL; Cooper JP; Feldman PL; Garrido DM; Goetz AS; Grizzle MK; Hertzog DL; Ignar DM; Lang DG; McIntyre MS; Ott RJ; Peat AJ; Zhou HQ
    J Med Chem; 2006 Nov; 49(24):7108-18. PubMed ID: 17125263
    [TBL] [Abstract][Full Text] [Related]  

  • 15. Building a MCHR1 homology model provides insight into the receptor-antagonist contacts that are important for the development of new anti-obesity agents.
    Cirauqui N; Schrey AK; Galiano S; Ceras J; Pérez-Silanes S; Aldana I; Monge A; Kühne R
    Bioorg Med Chem; 2010 Nov; 18(21):7365-79. PubMed ID: 20932767
    [TBL] [Abstract][Full Text] [Related]  

  • 16. Design and synthesis of substituted quinolines as novel and selective melanin concentrating hormone antagonists as anti-obesity agents.
    Warshakoon NC; Sheville J; Bhatt RT; Ji W; Mendez-Andino JL; Meyers KM; Kim N; Wos JA; Mitchell C; Paris JL; Pinney BB; Reizes O; Hu XE
    Bioorg Med Chem Lett; 2006 Oct; 16(19):5207-11. PubMed ID: 16870427
    [TBL] [Abstract][Full Text] [Related]  

  • 17. Discovery and characterization of aminopiperidinecoumarin melanin concentrating hormone receptor 1 antagonists.
    Kym PR; Iyengar R; Souers AJ; Lynch JK; Judd AS; Gao J; Freeman J; Mulhern M; Zhao G; Vasudevan A; Wodka D; Blackburn C; Brown J; Che JL; Cullis C; Lai SJ; LaMarche MJ; Marsilje T; Roses J; Sells T; Geddes B; Govek E; Patane M; Fry D; Dayton BD; Brodjian S; Falls D; Brune M; Bush E; Shapiro R; Knourek-Segel V; Fey T; McDowell C; Reinhart GA; Preusser LC; Marsh K; Hernandez L; Sham HL; Collins CA
    J Med Chem; 2005 Sep; 48(19):5888-91. PubMed ID: 16161992
    [TBL] [Abstract][Full Text] [Related]  

  • 18. Discovery of orally efficacious melanin-concentrating hormone receptor-1 antagonists as antiobesity agents. Synthesis, SAR, and biological evaluation of bicyclo[3.1.0]hexyl ureas.
    McBriar MD; Guzik H; Shapiro S; Paruchova J; Xu R; Palani A; Clader JW; Cox K; Greenlee WJ; Hawes BE; Kowalski TJ; O'neill K; Spar BD; Weig B; Weston DJ; Farley C; Cook J
    J Med Chem; 2006 Apr; 49(7):2294-310. PubMed ID: 16570926
    [TBL] [Abstract][Full Text] [Related]  

  • 19. Synthesis and anti-inflammatory activity evaluation of novel 7-alkoxy-1-amino-4,5-dihydro[1,2,4]triazole[4,3-a]quinolines.
    Sun XY; Wei CX; Chai KY; Piao HR; Quan ZS
    Arch Pharm (Weinheim); 2008 May; 341(5):288-93. PubMed ID: 18389515
    [TBL] [Abstract][Full Text] [Related]  

  • 20. Identification of ortho-amino benzamides and nicotinamides as MCHr1 antagonists.
    Vasudevan A; LaMarche MJ; Blackburn C; Che JL; Luchaco-Cullis CA; Lai S; Marsilje TH; Patane MA; Souers AJ; Wodka D; Geddes B; Chen S; Brodjian S; Falls DH; Dayton BD; Bush E; Brune M; Shapiro RD; Marsh KC; Hernandez LE; Sham HL; Collins CA; Kym PR
    Bioorg Med Chem Lett; 2005 Oct; 15(19):4174-9. PubMed ID: 16085414
    [TBL] [Abstract][Full Text] [Related]  

    [Next]    [New Search]
    of 7.