BIOMARKERS

Molecular Biopsy of Human Tumors

- a resource for Precision Medicine *

574 related articles for article (PubMed ID: 15358292)

  • 1. Design, synthesis, and pharmacological evaluation of some 2-[4-morpholino]-3-aryl-5-substituted thiophenes as novel anti-inflammatory agents: generation of a novel anti-inflammatory pharmacophore.
    Pillai AD; Rathod PD; Xavier FP; Vasu KK; Padh H; Sudarsanam V
    Bioorg Med Chem; 2004 Sep; 12(17):4667-71. PubMed ID: 15358292
    [TBL] [Abstract][Full Text] [Related]  

  • 2. Novel drug designing approach for dual inhibitors as anti-inflammatory agents: implication of pyridine template.
    Pillai AD; Rathod PD; P X F; Patel M; Nivsarkar M; Vasu KK; Padh H; Sudarsanam V
    Biochem Biophys Res Commun; 2003 Jan; 301(1):183-6. PubMed ID: 12535659
    [TBL] [Abstract][Full Text] [Related]  

  • 3. Tetra substituted thiophenes as anti-inflammatory agents: exploitation of analogue-based drug design.
    Pillai AD; Rathod PD; Xavier FP; Padh H; Sudarsanam V; K Vasu K
    Bioorg Med Chem; 2005 Dec; 13(24):6685-92. PubMed ID: 16125391
    [TBL] [Abstract][Full Text] [Related]  

  • 4. 2-Amino-5-thiazolyl motif: a novel scaffold for designing anti-inflammatory agents of diverse structures.
    Franklin PX; Pillai AD; Rathod PD; Yerande S; Nivsarkar M; Padh H; Vasu KK; Sudarsanam V
    Eur J Med Chem; 2008 Jan; 43(1):129-34. PubMed ID: 17467123
    [TBL] [Abstract][Full Text] [Related]  

  • 5. Syntheses of new tetrasubstituted thiophenes as novel anti-inflammatory agents.
    Molvi KI; Vasu KK; Yerande SG; Sudarsanam V; Haque N
    Eur J Med Chem; 2007 Aug; 42(8):1049-58. PubMed ID: 17336429
    [TBL] [Abstract][Full Text] [Related]  

  • 6. Synthesis and pharmacological evaluation of a novel series of 5-(substituted)aryl-3-(3-coumarinyl)-1-phenyl-2-pyrazolines as novel anti-inflammatory and analgesic agents.
    Khode S; Maddi V; Aragade P; Palkar M; Ronad PK; Mamledesai S; Thippeswamy AH; Satyanarayana D
    Eur J Med Chem; 2009 Apr; 44(4):1682-8. PubMed ID: 18986738
    [TBL] [Abstract][Full Text] [Related]  

  • 7. Design, synthesis and evaluation of novel 2-thiophen-5-yl-3H-quinazolin-4-one analogues as inhibitors of transcription factors NF-kappaB and AP-1 mediated transcriptional activation: Their possible utilization as anti-inflammatory and anti-cancer agents.
    Giri RS; Thaker HM; Giordano T; Williams J; Rogers D; Vasu KK; Sudarsanam V
    Bioorg Med Chem; 2010 Apr; 18(7):2796-808. PubMed ID: 20335039
    [TBL] [Abstract][Full Text] [Related]  

  • 8. Design, synthesis, and biological evaluation of 6-substituted-3-(4-methanesulfonylphenyl)-4-phenylpyran-2-ones: a novel class of diarylheterocyclic selective cyclooxygenase-2 inhibitors.
    Praveen Rao PN; Amini M; Li H; Habeeb AG; Knaus EE
    J Med Chem; 2003 Nov; 46(23):4872-82. PubMed ID: 14584938
    [TBL] [Abstract][Full Text] [Related]  

  • 9. Aroylpropionic acid based 2,5-disubstituted-1,3,4-oxadiazoles: synthesis and their anti-inflammatory and analgesic activities.
    Akhter M; Husain A; Azad B; Ajmal M
    Eur J Med Chem; 2009 Jun; 44(6):2372-8. PubMed ID: 18977556
    [TBL] [Abstract][Full Text] [Related]  

  • 10. QSAR studies on some thiophene analogs as anti-inflammatory agents: enhancement of activity by electronic parameters and its utilization for chemical lead optimization.
    Pillai AD; Rani S; Rathod PD; Xavier FP; Vasu KK; Padh H; Sudarsanam V
    Bioorg Med Chem; 2005 Feb; 13(4):1275-83. PubMed ID: 15670936
    [TBL] [Abstract][Full Text] [Related]  

  • 11. Design, synthesis and pharmacological evaluation of some novel 2-(4-nitrophenyl)-3-methylthio-3-(substituted)arylamino acrylamides as potential anti-inflammatory agents.
    Chhabria MT; Patel CK; Jani MH
    Pharmazie; 2005 Feb; 60(2):107-9. PubMed ID: 15739897
    [TBL] [Abstract][Full Text] [Related]  

  • 12. [Synthesis and anti-inflammatory activity of alpha-substituted p-(methanesulfonyl)phenylpropenamides].
    Ao GZ; Zhang YH; Ji H; Deng G
    Yao Xue Xue Bao; 2003 Sep; 38(9):671-6. PubMed ID: 14730916
    [TBL] [Abstract][Full Text] [Related]  

  • 13. Synthesis of 2-mercapto-3-substituted-5,6-dimethylthieno[2,3-d] pyrimidin-4(3H)-ones as new analgesic, anti-inflammatory agents.
    Alagarsamy V; Vijayakumar S; Raja Solomon V
    Biomed Pharmacother; 2007 Jun; 61(5):285-91. PubMed ID: 17391907
    [TBL] [Abstract][Full Text] [Related]  

  • 14. Design, synthesis, and SAR studies of some 5-aliphatic oximino esters of thiophene as potential anti-inflammatory leads: comparative biological activity profile of aliphatic oximes vs aromatic oximes.
    Pillai AD; Rathod PD; Franklin PX; Padh H; Vasu KK; Sudarsanam V
    Biochem Biophys Res Commun; 2004 May; 317(4):1067-74. PubMed ID: 15094377
    [TBL] [Abstract][Full Text] [Related]  

  • 15. Synthesis of celecoxib analogs that possess a N-hydroxypyrid-2(1H)one 5-lipoxygenase pharmacophore: biological evaluation as dual inhibitors of cyclooxygenases and 5-lipoxygenase with anti-inflammatory activity.
    Chowdhury MA; Abdellatif KR; Dong Y; Das D; Suresh MR; Knaus EE
    Bioorg Med Chem Lett; 2008 Dec; 18(23):6138-41. PubMed ID: 18945614
    [TBL] [Abstract][Full Text] [Related]  

  • 16. Design, synthesis and pharmacological screening of novel nitric oxide donors containing 1,5-diarylpyrazolin-3-one as nontoxic NSAIDs.
    Bhandari SV; Dangre SC; Bothara KG; Patil AA; Sarkate AP; Lokwani DK; Gore ST; Deshmane BJ; Raparti VT; Khachane CV
    Eur J Med Chem; 2009 Nov; 44(11):4622-36. PubMed ID: 19647903
    [TBL] [Abstract][Full Text] [Related]  

  • 17. Synthesis of 4-benzyl-1,3-thiazole derivatives as potential anti-inflammatory agents: an analogue-based drug design approach.
    Sharma RN; Xavier FP; Vasu KK; Chaturvedi SC; Pancholi SS
    J Enzyme Inhib Med Chem; 2009 Jun; 24(3):890-7. PubMed ID: 19469712
    [TBL] [Abstract][Full Text] [Related]  

  • 18. Design, synthesis, and structure-activity relationship studies of 3,4,6-triphenylpyran-2-ones as selective cyclooxygenase-2 inhibitors.
    Rao PN; Uddin MJ; Knaus EE
    J Med Chem; 2004 Jul; 47(16):3972-90. PubMed ID: 15267236
    [TBL] [Abstract][Full Text] [Related]  

  • 19. Design, synthesis, and anti-inflammatory evaluation of a series of novel amino acid-binding 1,5-diarylpyrazole derivatives.
    Li MH; Yin LL; Cai MJ; Zhang WY; Huang Y; Wang X; Zhu XZ; Shen JK
    Acta Pharmacol Sin; 2005 Jul; 26(7):865-72. PubMed ID: 15960895
    [TBL] [Abstract][Full Text] [Related]  

  • 20. Diarylspiro[2.4]heptenes as orally active, highly selective cyclooxygenase-2 inhibitors: synthesis and structure-activity relationships.
    Huang HC; Li JJ; Garland DJ; Chamberlain TS; Reinhard EJ; Manning RE; Seibert K; Koboldt CM; Gregory SA; Anderson GD; Veenhuizen AW; Zhang Y; Perkins WE; Burton EG; Cogburn JN; Isakson PC; Reitz DB
    J Med Chem; 1996 Jan; 39(1):253-66. PubMed ID: 8568815
    [TBL] [Abstract][Full Text] [Related]  

    [Next]    [New Search]
    of 29.