79 related articles for article (PubMed ID: 15863297)
21. Studies toward the discovery of the next generation of antidepressants. Part 6: Dual 5-HT1A receptor and serotonin transporter affinity within a class of arylpiperazinyl-cyclohexyl indole derivatives.
Zhou D; Zhou P; Evrard DA; Meagher K; Webb M; Harrison BL; Huryn DM; Golembieski J; Hornby GA; Schechter LE; Smith DL; Andree TH; Mewshaw RE
Bioorg Med Chem; 2008 Jul; 16(14):6707-23. PubMed ID: 18571421
[TBL] [Abstract][Full Text] [Related]
22. Structure-activity relationships of chiral selective norepinephrine reuptake inhibitors (sNRI) with increased oxidative stability.
Hudson S; Kiankarimi M; Eccles W; Dwight W; Mostofi YS; Genicot MJ; Fleck BA; Gogas K; Aparicio A; Wang H; Wen J; Wade WS
Bioorg Med Chem Lett; 2008 Aug; 18(16):4491-4. PubMed ID: 18672364
[TBL] [Abstract][Full Text] [Related]
23. Structure-activity relationships of the cycloalkanol ethylamine scaffold: discovery of selective norepinephrine reuptake inhibitors.
Mahaney PE; Gavrin LK; Trybulski EJ; Stack GP; Vu TA; Cohn ST; Ye F; Belardi JK; Santilli AA; Sabatucci JP; Leiter J; Johnston GH; Bray JA; Burroughs KD; Cosmi SA; Leventhal L; Koury EJ; Zhang Y; Mugford CA; Ho DM; Rosenzweig-Lipson SJ; Platt B; Smith VA; Deecher DC
J Med Chem; 2008 Jul; 51(13):4038-49. PubMed ID: 18557608
[TBL] [Abstract][Full Text] [Related]
24. Fragment based design of new H4 receptor-ligands with anti-inflammatory properties in vivo.
Smits RA; Lim HD; Hanzer A; Zuiderveld OP; Guaita E; Adami M; Coruzzi G; Leurs R; de Esch IJ
J Med Chem; 2008 Apr; 51(8):2457-67. PubMed ID: 18357976
[TBL] [Abstract][Full Text] [Related]
25. New benzomorphan derivatives of MPCB as MOP and KOP receptor ligands.
Pasquinucci L; Iadanza M; Marrazzo A; Prezzavento O; Ronsisvalle S; Scoto GM; Parenti C; De Luca L; Ronsisvalle G
Pharmazie; 2007 Nov; 62(11):813-24. PubMed ID: 18065096
[TBL] [Abstract][Full Text] [Related]
26. Conformationally constrained CCK8 analogues obtained from a rationally designed peptide library as ligands for cholecystokinin type B receptor.
De Luca S; Saviano M; Della Moglie R; Digilio G; Bracco C; Aloj L; Tarallo L; Pedone C; Morelli G
ChemMedChem; 2006 Sep; 1(9):997-1006. PubMed ID: 16915602
[TBL] [Abstract][Full Text] [Related]
27. The effects of norepinephrine transporter inactivation on locomotor activity in mice.
Mitchell HA; Ahern TH; Liles LC; Javors MA; Weinshenker D
Biol Psychiatry; 2006 Nov; 60(10):1046-52. PubMed ID: 16893531
[TBL] [Abstract][Full Text] [Related]
28. Novel trans-2-aryl-cyclopropylamine analogues as potent and selective dipeptidyl peptidase IV inhibitors.
Tsai TY; Hsu T; Chen CT; Cheng JH; Yeh TK; Chen X; Huang CY; Chang CN; Yeh KC; Hsieh SH; Chien CH; Chang YW; Huang CH; Huang YW; Huang CL; Wu SH; Wang MH; Lu CT; Chao YS; Jiaang WT
Bioorg Med Chem; 2009 Mar; 17(6):2388-99. PubMed ID: 19261480
[TBL] [Abstract][Full Text] [Related]
29. Synthesis and monoamine transporter affinity of 3-aryl substituted trop-2-enes.
Krunic A; Mariappan SV; Reith ME; Dunn WJ
Bioorg Med Chem Lett; 2005 Dec; 15(24):5488-93. PubMed ID: 16202585
[TBL] [Abstract][Full Text] [Related]
30. Two- and three dimensional combinatorial chemistry from multicomponent Grignard reagents.
Bülow A; Sinning S; Wiborg O; Bols M
J Comb Chem; 2004; 6(4):509-19. PubMed ID: 15244412
[TBL] [Abstract][Full Text] [Related]
31. Ex vivo and in vivo evaluation of [18F]PR04.MZ in rodents: a selective dopamine transporter imaging agent.
Riss PJ; Debus F; Hummerich R; Schmidt U; Schloss P; Lueddens H; Roesch F
ChemMedChem; 2009 Sep; 4(9):1480-7. PubMed ID: 19588472
[TBL] [Abstract][Full Text] [Related]
32. Highly potent fluorescence-tagged nonimidazole histamine H3 receptor ligands.
Amon M; Ligneau X; Camelin JC; Berrebi-Bertrand I; Schwartz JC; Stark H
ChemMedChem; 2007 May; 2(5):708-16. PubMed ID: 17361979
[TBL] [Abstract][Full Text] [Related]
33. A medicinal-chemistry-guided approach to selective and druglike sigma 1 ligands.
Corbera J; Vaño D; Martínez D; Vela JM; Zamanillo D; Dordal A; Andreu F; Hernandez E; Perez R; Escriche M; Salgado L; Yeste S; Serafini MT; Pascual R; Alegre J; Calvet MC; Cano N; Carro M; Buschmann H; Holenz J
ChemMedChem; 2006 Jan; 1(1):140-54. PubMed ID: 16892345
[TBL] [Abstract][Full Text] [Related]
34. Synthesis and monoamine transporter affinity of 2beta-carbomethoxy-3beta-(4'-p-substituted phenyl)-piperidine analogs of cocaine.
Bois F; Baldwin RM; Kula NS; Baldessarini RJ; Al Tikriti M; Innis RB; Tamagnan GD
Bioorg Med Chem Lett; 2006 Oct; 16(19):5222-5. PubMed ID: 16908151
[TBL] [Abstract][Full Text] [Related]
35. Synthesis and pharmacological evaluation of novel conformationally constrained homologues of glutamic acid.
Conti P; Caligiuri A; Pinto A; Roda G; Tamborini L; Nielsen B; Madsen U; Frydenvang K; Colombo A; De Micheli C
Eur J Med Chem; 2007 Aug; 42(8):1059-68. PubMed ID: 17346858
[TBL] [Abstract][Full Text] [Related]
36. Tuning the acyclic ether moiety of anticancer agent AA005 with conformationally constrained fragments.
Liu HX; Shao F; Li GQ; Xun GL; Yao ZJ
Chemistry; 2008; 14(28):8632-9. PubMed ID: 18688824
[TBL] [Abstract][Full Text] [Related]
37. Cyclic MrIA: a stable and potent cyclic conotoxin with a novel topological fold that targets the norepinephrine transporter.
Lovelace ES; Armishaw CJ; Colgrave ML; Wahlstrom ME; Alewood PF; Daly NL; Craik DJ
J Med Chem; 2006 Nov; 49(22):6561-8. PubMed ID: 17064074
[TBL] [Abstract][Full Text] [Related]
38. Design, synthesis, and biological evaluation of potent c-Met inhibitors.
D'Angelo ND; Bellon SF; Booker SK; Cheng Y; Coxon A; Dominguez C; Fellows I; Hoffman D; Hungate R; Kaplan-Lefko P; Lee MR; Li C; Liu L; Rainbeau E; Reider PJ; Rex K; Siegmund A; Sun Y; Tasker AS; Xi N; Xu S; Yang Y; Zhang Y; Burgess TL; Dussault I; Kim TS
J Med Chem; 2008 Sep; 51(18):5766-79. PubMed ID: 18763753
[TBL] [Abstract][Full Text] [Related]
39. chi-Conopeptide pharmacophore development: toward a novel class of norepinephrine transporter inhibitor (Xen2174) for pain.
Brust A; Palant E; Croker DE; Colless B; Drinkwater R; Patterson B; Schroeder CI; Wilson D; Nielsen CK; Smith MT; Alewood D; Alewood PF; Lewis RJ
J Med Chem; 2009 Nov; 52(22):6991-7002. PubMed ID: 19860431
[TBL] [Abstract][Full Text] [Related]
40. Design, synthesis, and preliminary SAR study of 3- and 6-side-chain-extended tetrahydro-pyran analogues of cis- and trans-(6-benzhydryl-tetrahydropyran-3-yl)-benzylamine.
Zhang S; Zhen J; Reith ME; Dutta AK
Bioorg Med Chem; 2006 Jun; 14(11):3953-66. PubMed ID: 16481172
[TBL] [Abstract][Full Text] [Related]
[Previous] [Next] [New Search]
