These tools will no longer be maintained as of December 31, 2024. Archived website can be found here. PubMed4Hh GitHub repository can be found here. Contact NLM Customer Service if you have questions.


BIOMARKERS

Molecular Biopsy of Human Tumors

- a resource for Precision Medicine *

111 related articles for article (PubMed ID: 16002287)

  • 21. Discovery of 5-HT6 receptor ligands based on virtual HTS.
    Tasler S; Kraus J; Wuzik A; Müller O; Aschenbrenner A; Cubero E; Pascual R; Quintana-Ruiz JR; Dordal A; Mercè R; Codony X
    Bioorg Med Chem Lett; 2007 Nov; 17(22):6224-9. PubMed ID: 17892934
    [TBL] [Abstract][Full Text] [Related]  

  • 22. Pyrrolo[1,2-a][1,4]benzodiazepine: a novel class of non-azole anti-dermatophyte anti-fungal agents.
    Meerpoel L; Van Gestel J; Van Gerven F; Woestenborghs F; Marichal P; Sipido V; Terence G; Nash R; Corens D; Richards RD
    Bioorg Med Chem Lett; 2005 Jul; 15(14):3453-8. PubMed ID: 15950472
    [TBL] [Abstract][Full Text] [Related]  

  • 23. Synthesis, cannabinoid receptor affinity, and molecular modeling studies of substituted 1-aryl-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamides.
    Silvestri R; Cascio MG; La Regina G; Piscitelli F; Lavecchia A; Brizzi A; Pasquini S; Botta M; Novellino E; Di Marzo V; Corelli F
    J Med Chem; 2008 Mar; 51(6):1560-76. PubMed ID: 18293908
    [TBL] [Abstract][Full Text] [Related]  

  • 24. SAR studies on new bis-aryls 5-HT7 ligands: Synthesis and molecular modeling.
    Badarau E; Bugno R; Suzenet F; Bojarski AJ; Finaru AL; Guillaumet G
    Bioorg Med Chem; 2010 Mar; 18(5):1958-67. PubMed ID: 20138771
    [TBL] [Abstract][Full Text] [Related]  

  • 25. Benzimidazolone-based serotonin 5-HT1A or 5-HT7R ligands: synthesis and biological evaluation.
    Badarau E; Suzenet F; Bojarski AJ; Fînaru AL; Guillaumet G
    Bioorg Med Chem Lett; 2009 Mar; 19(6):1600-3. PubMed ID: 19237285
    [TBL] [Abstract][Full Text] [Related]  

  • 26. 1,2,3,4-tetrahydrocarbazoles as 5-HT6 serotonin receptor ligands.
    Chang-Fong J; Rangisetty JB; Dukat M; Setola V; Raffay T; Roth B; Glennon RA
    Bioorg Med Chem Lett; 2004 Apr; 14(8):1961-4. PubMed ID: 15050637
    [TBL] [Abstract][Full Text] [Related]  

  • 27. Structure-activity relationships of 1,5-biaryl pyrroles as EP1 receptor antagonists.
    Hall A; Atkinson S; Brown SH; Chessell IP; Chowdhury A; Clayton NM; Coleman T; Giblin GM; Gleave RJ; Hammond B; Healy MP; Johnson MR; Michel AD; Naylor A; Novelli R; Spalding DJ; Tang SP
    Bioorg Med Chem Lett; 2006 Jul; 16(14):3657-62. PubMed ID: 16697196
    [TBL] [Abstract][Full Text] [Related]  

  • 28. Preparation of piperazine derivatives as 5-HT7 receptor antagonists.
    Yoon J; Yoo EA; Kim JY; Pae AN; Rhim H; Park WK; Kong JY; Park Choo HY
    Bioorg Med Chem; 2008 May; 16(10):5405-12. PubMed ID: 18456500
    [TBL] [Abstract][Full Text] [Related]  

  • 29. Synthesis, cannabinoid receptor affinity, molecular modeling studies and in vivo pharmacological evaluation of new substituted 1-aryl-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamides. 2. Effect of the 3-carboxamide substituent on the affinity and selectivity profile.
    Silvestri R; Ligresti A; La Regina G; Piscitelli F; Gatti V; Brizzi A; Pasquini S; Lavecchia A; Allarà M; Fantini N; Carai MA; Novellino E; Colombo G; Di Marzo V; Corelli F
    Bioorg Med Chem; 2009 Aug; 17(15):5549-64. PubMed ID: 19595596
    [TBL] [Abstract][Full Text] [Related]  

  • 30. Cyclic guanidines as dual 5-HT5A/5-HT7 receptor ligands: optimising brain penetration.
    Peters JU; Lübbers T; Alanine A; Kolczewski S; Blasco F; Steward L
    Bioorg Med Chem Lett; 2008 Jan; 18(1):262-6. PubMed ID: 18023344
    [TBL] [Abstract][Full Text] [Related]  

  • 31. Design of novel hexahydropyrazinoquinolines as potent and selective dopamine D3 receptor ligands with improved solubility.
    Chen J; Ding K; Levant B; Wang S
    Bioorg Med Chem Lett; 2006 Jan; 16(2):443-6. PubMed ID: 16290142
    [TBL] [Abstract][Full Text] [Related]  

  • 32. Identification of a series of benzoxazoles as potent 5-HT6 ligands.
    Liu KG; Lo JR; Comery TA; Zhang GM; Zhang JY; Kowal DM; Smith DL; Di L; Kerns EH; Schechter LE; Robichaud AJ
    Bioorg Med Chem Lett; 2009 Feb; 19(4):1115-7. PubMed ID: 19152787
    [TBL] [Abstract][Full Text] [Related]  

  • 33. 5-HT and benzodiazepine receptor ligands. III. Synthesis and receptor affinities of 1,2,4-triazolo[4',3':1,6]pyridazino[4,5-b]quinoline and 2,3-dihydro-9-phenyl-1H-pyrrolo[3,4-b]quinoline-1-one derivatives.
    Anzini M; Cappelli A; Vomero S; Botta M; Cagnotto A
    Farmaco; 1990 Nov; 45(11):1169-79. PubMed ID: 1965122
    [TBL] [Abstract][Full Text] [Related]  

  • 34. Substituted pyrazolo[3,4-b]pyridines as potent A1 adenosine antagonists: synthesis, biological evaluation, and development of an A1 bovine receptor model.
    Tuccinardi T; Schenone S; Bondavalli F; Brullo C; Bruno O; Mosti L; Zizzari AT; Tintori C; Manetti F; Ciampi O; Trincavelli ML; Martini C; Martinelli A; Botta M
    ChemMedChem; 2008 Jun; 3(6):898-913. PubMed ID: 18338422
    [TBL] [Abstract][Full Text] [Related]  

  • 35. (Phenylpiperazinyl-butyl)oxindoles as selective 5-HT7 receptor antagonists.
    Volk B; Barkóczy J; Hegedus E; Udvari S; Gacsályi I; Mezei T; Pallagi K; Kompagne H; Lévay G; Egyed A; Hársing LG; Spedding M; Simig G
    J Med Chem; 2008 Apr; 51(8):2522-32. PubMed ID: 18361484
    [TBL] [Abstract][Full Text] [Related]  

  • 36. Dihydropyrrole[2,3-d]pyridine derivatives as novel corticotropin-releasing factor-1 antagonists: mapping of the receptor binding pocket by in silico docking studies.
    Di Fabio R; Arban R; Bernasconi G; Braggio S; Blaney FE; Capelli AM; Castiglioni E; Donati D; Fazzolari E; Ratti E; Feriani A; Contini S; Gentile G; Ghirlanda D; Sabbatini FM; Andreotti D; Spada S; Marchioro C; Worby A; St-Denis Y
    J Med Chem; 2008 Nov; 51(22):7273-86. PubMed ID: 18975927
    [TBL] [Abstract][Full Text] [Related]  

  • 37. Discovery of a potent and selective 5-ht5A receptor antagonist by high-throughput chemistry.
    Corbett DF; Heightman TD; Moss SF; Bromidge SM; Coggon SA; Longley MJ; Roa AM; Williams JA; Thomas DR
    Bioorg Med Chem Lett; 2005 Sep; 15(18):4014-8. PubMed ID: 16002289
    [TBL] [Abstract][Full Text] [Related]  

  • 38. Synthesis and structure-activity relationships of thieno[2,3-b]pyrroles as antagonists of the GnRH receptor.
    Arnould JC; Delouvrié B; Boutron P; Dossetter AG; Foote KM; Hamon A; Hancox U; Harris CS; Hutton M; Lamorlette M; Matusiak Z
    Bioorg Med Chem Lett; 2007 Dec; 17(23):6448-54. PubMed ID: 17937987
    [TBL] [Abstract][Full Text] [Related]  

  • 39. Virtual screen for ligands of orphan G protein-coupled receptors.
    Bock JR; Gough DA
    J Chem Inf Model; 2005; 45(5):1402-14. PubMed ID: 16180917
    [TBL] [Abstract][Full Text] [Related]  

  • 40. Alpha-methyltryptamine sulfonamide derivatives as novel glucocorticoid receptor ligands.
    Marshall DR; Rodriguez G; Thomson DS; Nelson R; Capolina A
    Bioorg Med Chem Lett; 2007 Jan; 17(2):315-9. PubMed ID: 17118655
    [TBL] [Abstract][Full Text] [Related]  

    [Previous]   [Next]    [New Search]
    of 6.