These tools will no longer be maintained as of December 31, 2024. Archived website can be found here. PubMed4Hh GitHub repository can be found here. Contact NLM Customer Service if you have questions.


BIOMARKERS

Molecular Biopsy of Human Tumors

- a resource for Precision Medicine *

164 related articles for article (PubMed ID: 16139501)

  • 1. Synthesis and evaluation of 18F-labeled dopamine D3 receptor ligands as potential PET imaging agents.
    Hocke C; Prante O; Löber S; Hübner H; Gmeiner P; Kuwert T
    Bioorg Med Chem Lett; 2005 Nov; 15(21):4819-23. PubMed ID: 16139501
    [TBL] [Abstract][Full Text] [Related]  

  • 2. 18F-Labeled FAUC 346 and BP 897 derivatives as subtype-selective potential PET radioligands for the dopamine D3 receptor.
    Hocke C; Prante O; Salama I; Hübner H; Löber S; Kuwert T; Gmeiner P
    ChemMedChem; 2008 May; 3(5):788-93. PubMed ID: 18306190
    [TBL] [Abstract][Full Text] [Related]  

  • 3. Fluorinated diaryl sulfides as serotonin transporter ligands: synthesis, structure-activity relationship study, and in vivo evaluation of fluorine-18-labeled compounds as PET imaging agents.
    Huang Y; Bae SA; Zhu Z; Guo N; Roth BL; Laruelle M
    J Med Chem; 2005 Apr; 48(7):2559-70. PubMed ID: 15801845
    [TBL] [Abstract][Full Text] [Related]  

  • 4. Structure-selectivity investigations of D2-like receptor ligands by CoMFA and CoMSIA guiding the discovery of D3 selective PET radioligands.
    Salama I; Hocke C; Utz W; Prante O; Boeckler F; Hübner H; Kuwert T; Gmeiner P
    J Med Chem; 2007 Feb; 50(3):489-500. PubMed ID: 17266201
    [TBL] [Abstract][Full Text] [Related]  

  • 5. Synthesis, biological evaluation and radiolabelling by 18F-fluoroarylation of a dopamine D3-selective ligand as prospective imaging probe for PET.
    Höfling SB; Maschauer S; Hübner H; Gmeiner P; Wester HJ; Prante O; Heinrich MR
    Bioorg Med Chem Lett; 2010 Dec; 20(23):6933-7. PubMed ID: 21030255
    [TBL] [Abstract][Full Text] [Related]  

  • 6. Synthesis and radioiodination of selective ligands for the dopamine D3 receptor subtype.
    Hocke C; Prante O; Löber S; Hübner H; Gmeiner P; Kuwert T
    Bioorg Med Chem Lett; 2004 Aug; 14(15):3963-6. PubMed ID: 15225707
    [TBL] [Abstract][Full Text] [Related]  

  • 7. Synthesis and in vitro evaluation of 18F labeled tyrosine derivatives as potential positron emission tomography (PET) imaging agents.
    Wang L; Qu W; Lieberman B; Ploessl K; Kung HF
    Bioorg Med Chem Lett; 2010 Jun; 20(12):3482-5. PubMed ID: 20529679
    [TBL] [Abstract][Full Text] [Related]  

  • 8. 5-substituted derivatives of 6-halogeno-3-((2-(S)-azetidinyl)methoxy)pyridine and 6-halogeno-3-((2-(S)-pyrrolidinyl)methoxy)pyridine with low picomolar affinity for alpha4beta2 nicotinic acetylcholine receptor and wide range of lipophilicity: potential probes for imaging with positron emission tomography.
    Zhang Y; Pavlova OA; Chefer SI; Hall AW; Kurian V; Brown LL; Kimes AS; Mukhin AG; Horti AG
    J Med Chem; 2004 May; 47(10):2453-65. PubMed ID: 15115389
    [TBL] [Abstract][Full Text] [Related]  

  • 9. Fluorine-18 click radiosynthesis and preclinical evaluation of a new 18F-labeled folic acid derivative.
    Ross TL; Honer M; Lam PY; Mindt TL; Groehn V; Schibli R; Schubiger PA; Ametamey SM
    Bioconjug Chem; 2008 Dec; 19(12):2462-70. PubMed ID: 19053298
    [TBL] [Abstract][Full Text] [Related]  

  • 10. [18F]FEAC and [18F]FEDAC: Two novel positron emission tomography ligands for peripheral-type benzodiazepine receptor in the brain.
    Yanamoto K; Kumata K; Yamasaki T; Odawara C; Kawamura K; Yui J; Hatori A; Suzuki K; Zhang MR
    Bioorg Med Chem Lett; 2009 Mar; 19(6):1707-10. PubMed ID: 19217778
    [TBL] [Abstract][Full Text] [Related]  

  • 11. Evaluation of 18F-labeled benzodioxine piperazine-based dopamine D4 receptor ligands: lipophilicity as a determinate of nonspecific binding.
    Kügler F; Sihver W; Ermert J; Hübner H; Gmeiner P; Prante O; Coenen HH
    J Med Chem; 2011 Dec; 54(24):8343-52. PubMed ID: 22039961
    [TBL] [Abstract][Full Text] [Related]  

  • 12. Development and evaluation of endothelin-A receptor (radio)ligands for positron emission tomography.
    Michel K; Büther K; Law MP; Wagner S; Schober O; Hermann S; Schäfers M; Riemann B; Höltke C; Kopka K
    J Med Chem; 2011 Feb; 54(4):939-48. PubMed ID: 21275367
    [TBL] [Abstract][Full Text] [Related]  

  • 13. Dopamine D3 receptor antagonists: the quest for a potentially selective PET ligand. Part 3: Radiosynthesis and in vivo studies.
    Bennacef I; Salinas CA; Bonasera TA; Gunn RN; Audrain H; Jakobsen S; Nabulsi N; Weinzimmer D; Carson RE; Huang Y; Holmes I; Micheli F; Heidbreder C; Gentile G; Rossi T; Laruelle M
    Bioorg Med Chem Lett; 2009 Sep; 19(17):5056-9. PubMed ID: 19635669
    [TBL] [Abstract][Full Text] [Related]  

  • 14. Design, synthesis, and binding affinities of potential positron emission tomography (PET) ligands with optimal lipophilicity for brain imaging of the dopamine D3 receptor. Part II.
    Leopoldo M; Lacivita E; De Giorgio P; Contino M; Berardi F; Perrone R
    Bioorg Med Chem; 2009 Jan; 17(2):758-66. PubMed ID: 19081257
    [TBL] [Abstract][Full Text] [Related]  

  • 15. Evaluation of [11C]hemicholinium-15 and [18F]hemicholinium-15 as new potential PET tracers for the high-affinity choline uptake system in the heart.
    Gao M; Miller MA; DeGrado TR; Mock BH; Lopshire JC; Rosenberger JG; Dusa C; Das MK; Groh WJ; Zipes DP; Hutchins GD; Zheng QH
    Bioorg Med Chem; 2007 Feb; 15(3):1289-97. PubMed ID: 17116396
    [TBL] [Abstract][Full Text] [Related]  

  • 16. Synthesis of an estrogen receptor beta-selective radioligand: 5-[18F]fluoro-(2R,3S)-2,3-bis(4-hydroxyphenyl)pentanenitrile and comparison of in vivo distribution with 16alpha-[18F]fluoro-17beta-estradiol.
    Yoo J; Dence CS; Sharp TL; Katzenellenbogen JA; Welch MJ
    J Med Chem; 2005 Oct; 48(20):6366-78. PubMed ID: 16190762
    [TBL] [Abstract][Full Text] [Related]  

  • 17. An improved synthesis of 4-[18F]-ADAM, a potent serotonin transporter imaging agent.
    Huang YY; Huang WS; Chu TC; Shiue CY
    Appl Radiat Isot; 2009 Jun; 67(6):1063-7. PubMed ID: 19339192
    [TBL] [Abstract][Full Text] [Related]  

  • 18. Fully automated synthesis of PET TSPO radioligands [11C]DAA1106 and [18F]FEDAA1106.
    Wang M; Gao M; Zheng QH
    Appl Radiat Isot; 2012 Jun; 70(6):965-73. PubMed ID: 22469868
    [TBL] [Abstract][Full Text] [Related]  

  • 19. Synthesis and evaluation of a 18F-labeled spirocyclic piperidine derivative as promising σ1 receptor imaging agent.
    Chen YY; Wang X; Zhang JM; Deuther-Conrad W; Zhang XJ; Huang Y; Li Y; Ye JJ; Cui MC; Steinbach J; Brust P; Liu BL; Jia HM
    Bioorg Med Chem; 2014 Oct; 22(19):5270-8. PubMed ID: 25189691
    [TBL] [Abstract][Full Text] [Related]  

  • 20. Synthesis of 4-(5-[18F]fluoromethyl-3-phenylisoxazol-4-yl)benzenesulfonamide, a new [18F]fluorinated analogue of valdecoxib, as a potential radiotracer for imaging cyclooxygenase-2 with positron emission tomography.
    Toyokuni T; Kumar JS; Walsh JC; Shapiro A; Talley JJ; Phelps ME; Herschman HR; Barrio JR; Satyamurthy N
    Bioorg Med Chem Lett; 2005 Nov; 15(21):4699-702. PubMed ID: 16153836
    [TBL] [Abstract][Full Text] [Related]  

    [Next]    [New Search]
    of 9.