BIOMARKERS

Molecular Biopsy of Human Tumors

- a resource for Precision Medicine *

25 related articles for article (PubMed ID: 16380259)

  • 1. Synthesis of selective PAK4 inhibitors for lung metastasis of lung cancer and melanoma cells.
    Song P; Zhao F; Li D; Qu J; Yao M; Su Y; Wang H; Zhou M; Wang Y; Gao Y; Li F; Zhao D; Zhang F; Rao Y; Xia M; Li H; Wang J; Cheng M
    Acta Pharm Sin B; 2022 Jun; 12(6):2905-2922. PubMed ID: 35755272
    [TBL] [Abstract][Full Text] [Related]  

  • 2. Three-Dimensional Interactions Analysis of the Anticancer Target c-Src Kinase with Its Inhibitors.
    Jha V; Macchia M; Tuccinardi T; Poli G
    Cancers (Basel); 2020 Aug; 12(8):. PubMed ID: 32824733
    [TBL] [Abstract][Full Text] [Related]  

  • 3. Insights into the EGFR SAR of N-phenylquinazolin-4-amine-derivatives using quantum mechanical pairwise-interaction energies.
    Simeon S; Jongkon N; Chotpatiwetchkul W; Gleeson MP
    J Comput Aided Mol Des; 2019 Aug; 33(8):745-757. PubMed ID: 31494804
    [TBL] [Abstract][Full Text] [Related]  

  • 4. Design, Synthesis and Biological Evaluation of Isoxazole-Based CK1 Inhibitors Modified with Chiral Pyrrolidine Scaffolds.
    Luxenburger A; Schmidt D; Ianes C; Pichlo C; Krüger M; von Drathen T; Brunstein E; Gainsford GJ; Baumann U; Knippschild U; Peifer C
    Molecules; 2019 Mar; 24(5):. PubMed ID: 30832206
    [TBL] [Abstract][Full Text] [Related]  

  • 5. Role of the Fyn-PKCδ signaling in SE-induced neuroinflammation and epileptogenesis in experimental models of temporal lobe epilepsy.
    Sharma S; Carlson S; Puttachary S; Sarkar S; Showman L; Putra M; Kanthasamy AG; Thippeswamy T
    Neurobiol Dis; 2018 Feb; 110():102-121. PubMed ID: 29197620
    [TBL] [Abstract][Full Text] [Related]  

  • 6. Chemical characteristics, synthetic methods, and biological potential of quinazoline and quinazolinone derivatives.
    Asif M
    Int J Med Chem; 2014; 2014():395637. PubMed ID: 25692041
    [TBL] [Abstract][Full Text] [Related]  

  • 7. Discovery of AZD8931, an Equipotent, Reversible Inhibitor of Signaling by EGFR, HER2, and HER3 Receptors.
    Barlaam B; Anderton J; Ballard P; Bradbury RH; Hennequin LF; Hickinson DM; Kettle JG; Kirk G; Klinowska T; Lambert-van der Brempt C; Trigwell C; Vincent J; Ogilvie D
    ACS Med Chem Lett; 2013 Aug; 4(8):742-6. PubMed ID: 24900741
    [TBL] [Abstract][Full Text] [Related]  

  • 8. Synthesis of quinazolines as tyrosine kinase inhibitors.
    Srivastava SK; Kumar V; Agarwal SK; Mukherjee R; Burman AC
    Anticancer Agents Med Chem; 2009 Mar; 9(3):246-75. PubMed ID: 19275520
    [TBL] [Abstract][Full Text] [Related]  

  • 9. Specific inhibition of epidermal growth factor receptor tyrosine kinase by 4-anilinoquinazolines.
    Wakeling AE; Barker AJ; Davies DH; Brown DS; Green LR; Cartlidge SA; Woodburn JR
    Breast Cancer Res Treat; 1996; 38(1):67-73. PubMed ID: 8825124
    [TBL] [Abstract][Full Text] [Related]  

  • 10. Inhibitors of epidermal growth factor receptor tyrosine kinase: Novel C-5 substituted anilinoquinazolines designed to target the ribose pocket.
    Ballard P; Bradbury RH; Harris CS; Hennequin LF; Hickinson M; Johnson PD; Kettle JG; Klinowska T; Leach AG; Morgentin R; Pass M; Ogilvie DJ; Olivier A; Warin N; Williams EJ
    Bioorg Med Chem Lett; 2006 Mar; 16(6):1633-7. PubMed ID: 16380259
    [TBL] [Abstract][Full Text] [Related]  

  • 11. Enhancement of EGFR tyrosine kinase inhibition by C-C multiple bonds-containing anilinoquinazolines.
    Ban HS; Tanaka Y; Nabeyama W; Hatori M; Nakamura H
    Bioorg Med Chem; 2010 Jan; 18(2):870-9. PubMed ID: 19969465
    [TBL] [Abstract][Full Text] [Related]  

  • 12. Tyrosine kinase inhibitors. 11. Soluble analogues of pyrrolo- and pyrazoloquinazolines as epidermal growth factor receptor inhibitors: synthesis, biological evaluation, and modeling of the mode of binding.
    Palmer BD; Trumpp-Kallmeyer S; Fry DW; Nelson JM; Showalter HD; Denny WA
    J Med Chem; 1997 May; 40(10):1519-29. PubMed ID: 9154973
    [TBL] [Abstract][Full Text] [Related]  

  • 13. Tyrosine kinase inhibitors. 15. 4-(Phenylamino)quinazoline and 4-(phenylamino)pyrido[d]pyrimidine acrylamides as irreversible inhibitors of the ATP binding site of the epidermal growth factor receptor.
    Smaill JB; Palmer BD; Rewcastle GW; Denny WA; McNamara DJ; Dobrusin EM; Bridges AJ; Zhou H; Showalter HD; Winters RT; Leopold WR; Fry DW; Nelson JM; Slintak V; Elliot WL; Roberts BJ; Vincent PW; Patmore SJ
    J Med Chem; 1999 May; 42(10):1803-15. PubMed ID: 10346932
    [TBL] [Abstract][Full Text] [Related]  

  • 14. Neutral 5-substituted 4-indazolylaminoquinazolines as potent, orally active inhibitors of erbB2 receptor tyrosine kinase.
    Barlaam B; Acton DG; Ballard P; Bradbury RH; Cross D; Ducray R; Germain H; Hudson K; Klinowska T; Magnien F; Ogilvie DJ; Olivier A; Ross HS; Smith R; Trigwell CB; Vautier M; Wright L
    Bioorg Med Chem Lett; 2008 Mar; 18(6):1799-803. PubMed ID: 18313293
    [TBL] [Abstract][Full Text] [Related]  

  • 15. Tyrosine kinase inhibitors. 13. Structure-activity relationships for soluble 7-substituted 4-[(3-bromophenyl)amino]pyrido[4,3-d]pyrimidines designed as inhibitors of the tyrosine kinase activity of the epidermal growth factor receptor.
    Thompson AM; Murray DK; Elliott WL; Fry DW; Nelson JA; Showalter HD; Roberts BJ; Vincent PW; Denny WA
    J Med Chem; 1997 Nov; 40(24):3915-25. PubMed ID: 9397172
    [TBL] [Abstract][Full Text] [Related]  

  • 16.
    ; ; . PubMed ID:
    [No Abstract]   [Full Text] [Related]  

  • 17.
    ; ; . PubMed ID:
    [No Abstract]   [Full Text] [Related]  

  • 18.
    ; ; . PubMed ID:
    [No Abstract]   [Full Text] [Related]  

  • 19.
    ; ; . PubMed ID:
    [No Abstract]   [Full Text] [Related]  

  • 20.
    ; ; . PubMed ID:
    [No Abstract]   [Full Text] [Related]  

    [Next]    [New Search]
    of 2.