These tools will no longer be maintained as of December 31, 2024. Archived website can be found here. PubMed4Hh GitHub repository can be found here. Contact NLM Customer Service if you have questions.


BIOMARKERS

Molecular Biopsy of Human Tumors

- a resource for Precision Medicine *

200 related articles for article (PubMed ID: 16392821)

  • 41. Allosteric modulators and selective agonists of muscarinic receptors.
    Holzgrabe U; De Amici M; Mohr K
    J Mol Neurosci; 2006; 30(1-2):165-8. PubMed ID: 17192667
    [TBL] [Abstract][Full Text] [Related]  

  • 42. Synthesis and pharmacological characterization of chiral pyrrolidinylfuran derivatives: the discovery of new functionally selective muscarinic agonists.
    Scapecchi S; Nesi M; Matucci R; Bellucci C; Buccioni M; Dei S; Guandalini L; Manetti D; Martini E; Marucci G; Romanelli MN; Teodori E; Cirilli R
    J Med Chem; 2008 Jul; 51(13):3905-12. PubMed ID: 18543900
    [TBL] [Abstract][Full Text] [Related]  

  • 43. Muscarinic antagonists with multiple stereocenters: Synthesis, affinity profile and functional activity of isomeric 1-methyl-2-(2,2-alkylaryl-1,3-oxathiolan-5-yl)pyrrolidine sulfoxide derivatives.
    Dei S; Bellucci C; Buccioni M; Ferraroni M; Guandalini L; Manetti D; Marucci G; Matucci R; Nesi M; Romanelli MN; Scapecchi S; Teodori E
    Bioorg Med Chem; 2008 May; 16(10):5490-500. PubMed ID: 18455407
    [TBL] [Abstract][Full Text] [Related]  

  • 44. Bis(ammonio)alkane-type agonists of muscarinic acetylcholine receptors: synthesis, in vitro functional characterization, and in vivo evaluation of their analgesic activity.
    Matera C; Flammini L; Quadri M; Vivo V; Ballabeni V; Holzgrabe U; Mohr K; De Amici M; Barocelli E; Bertoni S; Dallanoce C
    Eur J Med Chem; 2014 Mar; 75():222-32. PubMed ID: 24534538
    [TBL] [Abstract][Full Text] [Related]  

  • 45. Regulation of glutamate release from primary afferents and interneurons in the spinal cord by muscarinic receptor subtypes.
    Zhang HM; Chen SR; Pan HL
    J Neurophysiol; 2007 Jan; 97(1):102-9. PubMed ID: 17050831
    [TBL] [Abstract][Full Text] [Related]  

  • 46. Potentiation by alcuronium of the antimuscarinic effect of N-methylscopolamine in guinea pig left atria.
    Maass A; Kostenis E; Mohr K
    Eur J Pharmacol; 1995 Jan; 272(1):103-6. PubMed ID: 7713140
    [TBL] [Abstract][Full Text] [Related]  

  • 47. Determination of dissociation constants and relative efficacies of oxotremorine analogs at muscarinic receptors in the guinea-pig ileum by pharmacological procedures.
    Ringdahl B
    J Pharmacol Exp Ther; 1984 Apr; 229(1):199-206. PubMed ID: 6707935
    [TBL] [Abstract][Full Text] [Related]  

  • 48. Novel M(1) allosteric ligands: a patent review.
    Kuduk SD; Beshore DC
    Expert Opin Ther Pat; 2012 Dec; 22(12):1385-98. PubMed ID: 23092292
    [TBL] [Abstract][Full Text] [Related]  

  • 49. An optical dynamic mass redistribution assay reveals biased signaling of dualsteric GPCR activators.
    Kebig A; Kostenis E; Mohr K; Mohr-Andrä M
    J Recept Signal Transduct Res; 2009; 29(3-4):140-5. PubMed ID: 19586284
    [TBL] [Abstract][Full Text] [Related]  

  • 50. Impact of species variability and 'probe-dependence' on the detection and in vivo validation of allosteric modulation at the M4 muscarinic acetylcholine receptor.
    Suratman S; Leach K; Sexton P; Felder C; Loiacono R; Christopoulos A
    Br J Pharmacol; 2011 Apr; 162(7):1659-70. PubMed ID: 21198541
    [TBL] [Abstract][Full Text] [Related]  

  • 51. Exploring the mechanism of agonist efficacy: a relationship between efficacy and agonist dissociation rate at the muscarinic M3 receptor.
    Sykes DA; Dowling MR; Charlton SJ
    Mol Pharmacol; 2009 Sep; 76(3):543-51. PubMed ID: 19498041
    [TBL] [Abstract][Full Text] [Related]  

  • 52. 6H,13H-Pyrazino[1,2-a;4,5-a']diindole analogs: probing the pharmacophore for allosteric ligands of muscarinic M2 receptors.
    Zlotos DP; Tränkle C; Abdelrahman A; Gündisch D; Radacki K; Braunschweig H; Mohr K
    Bioorg Med Chem Lett; 2006 Mar; 16(6):1481-5. PubMed ID: 16387499
    [TBL] [Abstract][Full Text] [Related]  

  • 53. Developmental changes in presynaptic muscarinic modulation of excitatory and inhibitory neurotransmission in rat piriform cortex in vitro: relevance to epileptiform bursting susceptibility.
    Whalley BJ; Constanti A
    Neuroscience; 2006 Jul; 140(3):939-56. PubMed ID: 16616427
    [TBL] [Abstract][Full Text] [Related]  

  • 54. Characterization of aclidinium bromide, a novel inhaled muscarinic antagonist, with long duration of action and a favorable pharmacological profile.
    Gavaldà A; Miralpeix M; Ramos I; Otal R; Carreño C; Viñals M; Doménech T; Carcasona C; Reyes B; Vilella D; Gras J; Cortijo J; Morcillo E; Llenas J; Ryder H; Beleta J
    J Pharmacol Exp Ther; 2009 Nov; 331(2):740-51. PubMed ID: 19710368
    [TBL] [Abstract][Full Text] [Related]  

  • 55. Investigation of the interaction of a putative allosteric modulator, N-(2,3-diphenyl-1,2,4-thiadiazole-5-(2H)-ylidene) methanamine hydrobromide (SCH-202676), with M1 muscarinic acetylcholine receptors.
    Lanzafame A; Christopoulos A
    J Pharmacol Exp Ther; 2004 Mar; 308(3):830-7. PubMed ID: 14617684
    [TBL] [Abstract][Full Text] [Related]  

  • 56. Contrasting effects of allosteric and orthosteric agonists on m1 muscarinic acetylcholine receptor internalization and down-regulation.
    Thomas RL; Langmead CJ; Wood MD; Challiss RA
    J Pharmacol Exp Ther; 2009 Dec; 331(3):1086-95. PubMed ID: 19767446
    [TBL] [Abstract][Full Text] [Related]  

  • 57. The conformational and property space of acetylcholine bound to muscarinic receptors: an entropy component accounts for the subtype selectivity of acetylcholine.
    Vistoli G; Pedretti A; Testa B; Matucci R
    Arch Biochem Biophys; 2007 Aug; 464(1):112-21. PubMed ID: 17544360
    [TBL] [Abstract][Full Text] [Related]  

  • 58. Differential regulation of muscarinic M1 receptors by orthosteric and allosteric ligands.
    Davis CN; Bradley SR; Schiffer HH; Friberg M; Koch K; Tolf BR; Bonhaus DW; Lameh J
    BMC Pharmacol; 2009 Dec; 9():14. PubMed ID: 19951444
    [TBL] [Abstract][Full Text] [Related]  

  • 59. Orthosteric/allosteric bitopic ligands: going hybrid at GPCRs.
    Valant C; Sexton PM; Christopoulos A
    Mol Interv; 2009 Jun; 9(3):125-35. PubMed ID: 19592673
    [TBL] [Abstract][Full Text] [Related]  

  • 60. First gallamine-tacrine hybrid: design and characterization at cholinesterases and the M2 muscarinic receptor.
    Elsinghorst PW; Cieslik JS; Mohr K; Tränkle C; Gütschow M
    J Med Chem; 2007 Nov; 50(23):5685-95. PubMed ID: 17944454
    [TBL] [Abstract][Full Text] [Related]  

    [Previous]   [Next]    [New Search]
    of 10.