87 related articles for article (PubMed ID: 1642642)
1. Inactivation of brain cortex muscarinic receptors by 4-diphenylacetoxy-1-(2-chloroethyl) piperidine mustard.
Waelbroeck M; Renzetti AR; Tastenoy M; Barlow RB; Christophe J
Biochem Pharmacol; 1992 Jul; 44(2):285-90. PubMed ID: 1642642
[TBL] [Abstract][Full Text] [Related]
2. Conversion of N-(2-chloroethyl)-4-piperidinyl diphenylacetate (4-DAMP mustard) to an aziridinium ion and its interaction with muscarinic receptors in various tissues.
Thomas EA; Hsu HH; Griffin MT; Hunter AL; Luong T; Ehlert FJ
Mol Pharmacol; 1992 Apr; 41(4):718-26. PubMed ID: 1569923
[TBL] [Abstract][Full Text] [Related]
3. The interaction of 4-DAMP mustard with subtypes of the muscarinic receptor.
Ehlert FJ
Life Sci; 1996; 58(22):1971-8. PubMed ID: 8637426
[TBL] [Abstract][Full Text] [Related]
4. The quaternary transformation products of N-(3-chloropropyl)-4-piperidinyl diphenylacetate and N-(2-chloroethyl)-4-piperidinyl diphenylacetate (4-DAMP mustard) have differential affinity for subtypes of the muscarinic receptor.
Ehlert FJ; Oliff HS; Griffin MT
J Pharmacol Exp Ther; 1996 Feb; 276(2):405-10. PubMed ID: 8632303
[TBL] [Abstract][Full Text] [Related]
5. The use of 4-diphenylacetoxy-N-(2-chloroethyl)-piperidine (4-DAMP mustard) for estimating the apparent affinities of some agonists acting at muscarinic receptors in guinea-pig ileum.
Barlow RB; McMillen LS; Veale MA
Br J Pharmacol; 1991 Mar; 102(3):657-62. PubMed ID: 1364835
[TBL] [Abstract][Full Text] [Related]
6. Phenoxybenzamine and benextramine, but not 4-diphenylacetoxy-N-[2-chloroethyl]piperidine hydrochloride, display irreversible noncompetitive antagonism at G protein-coupled receptors.
Bodenstein J; Venter DP; Brink CB
J Pharmacol Exp Ther; 2005 Aug; 314(2):891-905. PubMed ID: 15857948
[TBL] [Abstract][Full Text] [Related]
7. Selective inactivation of muscarinic M2 and M3 receptors in guinea-pig ileum and atria in vitro.
Eglen RM; Harris GC
Br J Pharmacol; 1993 Aug; 109(4):946-52. PubMed ID: 8401947
[TBL] [Abstract][Full Text] [Related]
8. The use of irreversible ligands to inactivate receptor subtypes: 4-DAMP mustard and muscarinic receptors in smooth muscle.
Ehlert FJ; Griffin MT
Life Sci; 1998; 62(17-18):1659-64. PubMed ID: 9585153
[TBL] [Abstract][Full Text] [Related]
9. Irreversible effects of 4-DAMP mustard on muscarinic receptors in vivo.
Thomas EA; Ehlert FJ
Proc West Pharmacol Soc; 1992; 35():233-7. PubMed ID: 1502231
[No Abstract] [Full Text] [Related]
10. Functional role for the M2 muscarinic receptor in smooth muscle of guinea pig ileum.
Thomas EA; Baker SA; Ehlert FJ
Mol Pharmacol; 1993 Jul; 44(1):102-10. PubMed ID: 8393516
[TBL] [Abstract][Full Text] [Related]
11. Pharmacological profiles for rat cortical M1 and M2 muscarinic receptors using selective antagonists: comparison with N1E-115 muscarinic receptors.
McKinney M; Anderson DJ; Vella-Rountree L; Connolly T; Miller JH
J Pharmacol Exp Ther; 1991 Jun; 257(3):1121-9. PubMed ID: 1646322
[TBL] [Abstract][Full Text] [Related]
12. Characterization of muscarinic receptors in the human bladder mucosa: direct quantification of subtypes using 4-DAMP mustard.
Yoshida A; Seki M; Nasrin S; Otsuka A; Ozono S; Takeda M; Masuyama K; Araki I; Ehlert FJ; Yamada S
Urology; 2011 Sep; 78(3):721.e7-721.e12. PubMed ID: 21777958
[TBL] [Abstract][Full Text] [Related]
13. Functional and direct binding studies using subtype selective muscarinic receptor antagonists.
Kunysz EL; Michel AD; Whiting RL
Br J Pharmacol; 1988 Mar; 93(3):491-500. PubMed ID: 2897216
[TBL] [Abstract][Full Text] [Related]
14. Kinetics of activation and in vivo muscarinic receptor binding of N-(2-bromoethyl)-4-piperidinyl diphenylacetate: an analog of 4-DAMP mustard.
Griffin MT; Thomas EA; Ehlert FJ
J Pharmacol Exp Ther; 1993 Jul; 266(1):301-5. PubMed ID: 8331565
[TBL] [Abstract][Full Text] [Related]
15. Muscarinic M2 receptor-mediated contraction in the guinea pig Taenia caeci: possible involvement of protein kinase C.
Shen A; Mitchelson F
Biochem Pharmacol; 1998 Dec; 56(11):1529-37. PubMed ID: 9827588
[TBL] [Abstract][Full Text] [Related]
16. On the involvement of multiple muscarinic receptor subtypes in the activation of phosphoinositide metabolism in rat cerebral cortex.
Forray C; el-Fakahany EE
Mol Pharmacol; 1990 Jun; 37(6):893-902. PubMed ID: 2163015
[TBL] [Abstract][Full Text] [Related]
17. Some differential effects of 4-diphenylacetoxy-N-(2-chloroethyl)-piperidine hydrochloride on guinea-pig atria and ileum.
Barlow RB; Shepherd MK; Veale MA
J Pharm Pharmacol; 1990 Jun; 42(6):412-8. PubMed ID: 1979621
[TBL] [Abstract][Full Text] [Related]
18. Selective inactivation of muscarinic receptor subtypes.
Eglen RM; Reddy H; Watson N
Int J Biochem; 1994 Dec; 26(12):1357-68. PubMed ID: 7890115
[TBL] [Abstract][Full Text] [Related]
19. Propylbenzilylcholine mustard is selective for rat heart muscarinic receptors having a low affinity for agonists.
Christophe J; De Neef P; Robberecht P; Waelbroeck M
Br J Pharmacol; 1986 May; 88(1):63-70. PubMed ID: 3708224
[TBL] [Abstract][Full Text] [Related]
20. The role of M2 muscarinic receptor subtypes in mediating contraction of the pig bladder base after cyclic adenosine monophosphate elevation and/or selective M3 inactivation.
Yamanishi T; Chapple CR; Yasuda K; Chess-Williams R
J Urol; 2002 Jan; 167(1):397-401. PubMed ID: 11743363
[TBL] [Abstract][Full Text] [Related]
[Next] [New Search]
