142 related articles for article (PubMed ID: 16481172)
21. Development of potent dopamine-norepinephrine uptake inhibitors (DNRIs) based on a (2S,4R,5R)-2-benzhydryl-5-((4-methoxybenzyl)amino)tetrahydro-2H-pyran-4-ol molecular template.
Santra S; Sharma H; Vedachalam S; Antonio T; Reith M; Dutta A
Bioorg Med Chem; 2015 Feb; 23(4):821-8. PubMed ID: 25593099
[TBL] [Abstract][Full Text] [Related]
22. Design and synthesis of a novel photoaffinity ligand for the dopamine and serotonin transporters based on 2beta-carbomethoxy-3beta-biphenyltropane.
Newman AH; Cha JH; Cao J; Kopajtic T; Katz JL; Parnas ML; Vaughan R; Lever JR
J Med Chem; 2006 Nov; 49(22):6621-5. PubMed ID: 17064081
[TBL] [Abstract][Full Text] [Related]
23. Synthesis of enantiomerically pure milnacipran analogs and inhibition of dopamine, serotonin, and norepinephrine transporters.
Roggen H; Kehler J; Stensbøl TB; Hansen T
Bioorg Med Chem Lett; 2007 May; 17(10):2834-7. PubMed ID: 17350257
[TBL] [Abstract][Full Text] [Related]
24. Synthesis and monoamine transporter binding properties of 2,3-diaryltropanes.
Kotturi SV; Jiang S; Chang AC; Abraham P; Navarro HA; Kuhar MJ; Carroll FI
J Med Chem; 2005 Nov; 48(23):7437-44. PubMed ID: 16279803
[TBL] [Abstract][Full Text] [Related]
25. Synthesis and pharmacological evaluation of 3-(3,4-dichlorophenyl)-1-indanamine derivatives as nonselective ligands for biogenic amine transporters.
Yu H; Kim IJ; Folk JE; Tian X; Rothman RB; Baumann MH; Dersch CM; Flippen-Anderson JL; Parrish D; Jacobson AE; Rice KC
J Med Chem; 2004 May; 47(10):2624-34. PubMed ID: 15115403
[TBL] [Abstract][Full Text] [Related]
26. Trishomocubane as a scaffold for the development of selective dopamine transporter (DAT) ligands.
Banister SD; Moussa IA; Beinat C; Reynolds AJ; Schiavini P; Jorgensen WT; Kassiou M
Bioorg Med Chem Lett; 2011 Jan; 21(1):38-41. PubMed ID: 21146989
[TBL] [Abstract][Full Text] [Related]
27. Synthesis and amine transporter affinities of novel phenyltropane derivatives as potential positron emission tomography (PET) imaging agents.
Peng X; Zhang A; Kula NS; Baldessarini RJ; Neumeyer JL
Bioorg Med Chem Lett; 2004 Nov; 14(22):5635-9. PubMed ID: 15482938
[TBL] [Abstract][Full Text] [Related]
28. Synthesis and monoamine transporter affinity of new 2beta-carbomethoxy-3beta-[aryl or heteroaryl]phenyltropanes.
Tamagnan G; Alagille D; Fu X; Kula NS; Baldessarini RJ; Innis RB; Baldwin RM
Bioorg Med Chem Lett; 2006 Jan; 16(1):217-20. PubMed ID: 16236497
[TBL] [Abstract][Full Text] [Related]
29. D-161, a novel pyran-based triple monoamine transporter blocker: behavioral pharmacological evidence for antidepressant-like action.
Dutta AK; Ghosh B; Biswas S; Reith ME
Eur J Pharmacol; 2008 Jul; 589(1-3):73-9. PubMed ID: 18561912
[TBL] [Abstract][Full Text] [Related]
30. Substrates and inhibitors display different sensitivity to expression level of the dopamine transporter in heterologously expressing cells.
Chen N; Reith ME
J Neurochem; 2007 Apr; 101(2):377-88. PubMed ID: 17250655
[TBL] [Abstract][Full Text] [Related]
31. Validation of a fluorescence-based high-throughput assay for the measurement of neurotransmitter transporter uptake activity.
Jørgensen S; Nielsen EØ; Peters D; Dyhring T
J Neurosci Methods; 2008 Mar; 169(1):168-76. PubMed ID: 18222006
[TBL] [Abstract][Full Text] [Related]
32. Design, synthesis, and activity of novel cis- and trans-3,6-disubstituted pyran biomimetics of 3,6-disubstituted piperidine as potential ligands for the dopamine transporter.
Zhang S; Reith ME; Dutta AK
Bioorg Med Chem Lett; 2003 May; 13(9):1591-5. PubMed ID: 12699762
[TBL] [Abstract][Full Text] [Related]
33. Caulis Sinomenii extracts activate DA/NE transporter and inhibit 5HT transporter.
Zhao G; Bi C; Qin GW; Guo LH
Exp Biol Med (Maywood); 2009 Aug; 234(8):976-85. PubMed ID: 19491370
[TBL] [Abstract][Full Text] [Related]
34. Pharmacophore design and database searching for selective monoamine neurotransmitter transporter ligands.
Macdougall IJ; Griffith R
J Mol Graph Model; 2008 Apr; 26(7):1113-24. PubMed ID: 18023378
[TBL] [Abstract][Full Text] [Related]
35. Structure-activity relationships of substituted N-benzyl piperidines in the GBR series: Synthesis of 4-(2-(bis(4-fluorophenyl)methoxy)ethyl)-1-(2-trifluoromethylbenzyl)piperidine, an allosteric modulator of the serotonin transporter.
Boos TL; Greiner E; Calhoun WJ; Prisinzano TE; Nightingale B; Dersch CM; Rothman RB; Jacobson AE; Rice KC
Bioorg Med Chem; 2006 Jun; 14(11):3967-73. PubMed ID: 16563775
[TBL] [Abstract][Full Text] [Related]
36. Synthesis and in vivo evaluation of fluorine-18 and iodine-123 labeled 2beta-carbo(2-fluoroethoxy)-3beta-(4'-((Z)-2-iodoethenyl)phenyl)nortropane as a candidate serotonin transporter imaging agent.
Plisson C; Stehouwer JS; Voll RJ; Howell L; Votaw JR; Owens MJ; Goodman MM
J Med Chem; 2007 Sep; 50(19):4553-60. PubMed ID: 17705359
[TBL] [Abstract][Full Text] [Related]
37. Inhibitive effects of Fructus Psoraleae extract on dopamine transporter and noradrenaline transporter.
Zhao G; Li S; Qin GW; Fei J; Guo LH
J Ethnopharmacol; 2007 Jul; 112(3):498-506. PubMed ID: 17555897
[TBL] [Abstract][Full Text] [Related]
38. Synthesis and monoamine transporter affinity of 2beta-carbomethoxy-3beta-(4'-p-substituted phenyl)-piperidine analogs of cocaine.
Bois F; Baldwin RM; Kula NS; Baldessarini RJ; Al Tikriti M; Innis RB; Tamagnan GD
Bioorg Med Chem Lett; 2006 Oct; 16(19):5222-5. PubMed ID: 16908151
[TBL] [Abstract][Full Text] [Related]
39. Flexible and biomimetic analogs of triple uptake inhibitor 4-((((3S,6S)-6-benzhydryltetrahydro-2H-pyran-3-yl)amino)methyl)phenol: Synthesis, biological characterization, and development of a pharmacophore model.
Sharma H; Santra S; Debnath J; Antonio T; Reith M; Dutta A
Bioorg Med Chem; 2014 Jan; 22(1):311-24. PubMed ID: 24315194
[TBL] [Abstract][Full Text] [Related]
40. Further structure-activity relationship studies on 4-((((3S,6S)-6-benzhydryltetrahydro-2H-pyran-3-yl)amino)methyl)phenol: identification of compounds with triple uptake inhibitory activity as potential antidepressant agents.
Gopishetty B; Hazeldine S; Santra S; Johnson M; Modi G; Ali S; Zhen J; Reith M; Dutta A
J Med Chem; 2011 Apr; 54(8):2924-32. PubMed ID: 21446715
[TBL] [Abstract][Full Text] [Related]
[Previous] [Next] [New Search]
