134 related articles for article (PubMed ID: 16508202)
1. Synthesis of (-)-epibatidine and its derivatives from chiral allene-1,3-dicarboxylate esters.
Kimura H; Fujiwara T; Katoh T; Nishide K; Kajimoto T; Node M
Chem Pharm Bull (Tokyo); 2006 Mar; 54(3):399-402. PubMed ID: 16508202
[TBL] [Abstract][Full Text] [Related]
2. Epibatidine analogues as selective ligands for the alpha(x)beta2-containing subtypes of nicotinic acetylcholine receptors.
Huang Y; Zhu Z; Xiao Y; Laruelle M
Bioorg Med Chem Lett; 2005 Oct; 15(19):4385-8. PubMed ID: 16039849
[TBL] [Abstract][Full Text] [Related]
3. Synthesis and structure-activity data of some new epibatidine analogues.
Seerden JP; Tulp MT; Scheeren HW; Kruse CG
Bioorg Med Chem; 1998 Nov; 6(11):2103-10. PubMed ID: 9881100
[TBL] [Abstract][Full Text] [Related]
4. Epibatidine structure-activity relationships.
Carroll FI
Bioorg Med Chem Lett; 2004 Apr; 14(8):1889-96. PubMed ID: 15050621
[TBL] [Abstract][Full Text] [Related]
5. Stereoselective syntheses of (+/-)-epibatidine analogues.
Kim YH; Won DY; Oh CY; Lee KY; Lee YS; Woo NT; Park YH; Park HJ; Ham WH
Arch Pharm Res; 2002 Feb; 25(1):45-8. PubMed ID: 11885690
[TBL] [Abstract][Full Text] [Related]
6. Synthesis and nicotinic acetylcholine receptor binding properties of bridged and fused ring analogues of epibatidine.
Carroll FI; Robinson TP; Brieaddy LE; Atkinson RN; Mascarella SW; Damaj MI; Martin BR; Navarro HA
J Med Chem; 2007 Dec; 50(25):6383-91. PubMed ID: 17994682
[TBL] [Abstract][Full Text] [Related]
7. Syntheses and biological properties of cysteine-reactive epibatidine derivatives.
Che C; Petit G; Kotzyba-Hibert F; Bertrand S; Bertrand D; Grutter T; Goeldner M
Bioorg Med Chem Lett; 2003 Mar; 13(6):1001-4. PubMed ID: 12643898
[TBL] [Abstract][Full Text] [Related]
8. Synthesis and pharmacological characterization of exo-2-(2'-chloro-5-pyridinyl)-7-(endo and exo)-aminobicyclo[2.2.1]heptanes as novel epibatidine analogues.
Carroll FI; Brieaddy LE; Navarro HA; Damaj MI; Martin BR
J Med Chem; 2005 Nov; 48(23):7491-5. PubMed ID: 16279810
[TBL] [Abstract][Full Text] [Related]
9. Synthesis of (-)-epibatidine.
Evans DA; Scheidt KA; Downey CW
Org Lett; 2001 Sep; 3(19):3009-12. PubMed ID: 11554830
[TBL] [Abstract][Full Text] [Related]
10. An alternative improved synthesis of (-)-norferruginine, a potent nAChR agonist.
Wegge T; Schwarz S; Seitz G
Pharmazie; 2000 Oct; 55(10):779-80. PubMed ID: 11082844
[No Abstract] [Full Text] [Related]
11. Synthesis and pharmacological characterization of bivalent ligands of epibatidine at neuronal nicotinic acetylcholine receptors.
Wei ZL; Xiao Y; Kellar KJ; Kozikowski AP
Bioorg Med Chem Lett; 2004 Apr; 14(8):1855-8. PubMed ID: 15050615
[TBL] [Abstract][Full Text] [Related]
12. Syntheses of (+/-)-homoepibatidine analogues.
Kim YH; Oh CY; Lee KY; Lee YS; Jung YH; Park HJ; Ham WH
Arch Pharm Res; 2002 Feb; 25(1):49-52. PubMed ID: 11885691
[TBL] [Abstract][Full Text] [Related]
13. Synthesis and electrophysiological studies of a novel epibatidine analogue.
Spang JE; Patt JT; Bertrand S; Bertrand D; Westera G; Schubiger PA
J Recept Signal Transduct Res; 1999; 19(1-4):521-31. PubMed ID: 10071782
[TBL] [Abstract][Full Text] [Related]
14. Synthesis and binding studies of epibatidine analogues as ligands for the nicotinic acetylcholine receptors.
Mu L; Drandarov K; Bisson WH; Schibig A; Wirz C; Schubiger PA; Westera G
Eur J Med Chem; 2006 May; 41(5):640-50. PubMed ID: 16545497
[TBL] [Abstract][Full Text] [Related]
15. Synthesis of heterocyclic analogues of epibatidine via 7-azabicyclo[2.2.1]hept-2-yl radical intermediates. 1. Intermolecular reactions.
Gómez-Sánchez E; Soriano E; Marco-Contelles J
J Org Chem; 2008 Sep; 73(17):6784-92. PubMed ID: 18656981
[TBL] [Abstract][Full Text] [Related]
16. Novel pyridyl ring C5 substituted analogues of epibatidine and 3-(1-methyl-2(S)-pyrrolidinylmethoxy)pyridine (A-84543) as highly selective agents for neuronal nicotinic acetylcholine receptors containing beta2 subunits.
Wei ZL; Xiao Y; Yuan H; Baydyuk M; Petukhov PA; Musachio JL; Kellar KJ; Kozikowski AP
J Med Chem; 2005 Mar; 48(6):1721-4. PubMed ID: 15771418
[TBL] [Abstract][Full Text] [Related]
17. Synthesis, nicotinic acetylcholine receptor binding, and antinociceptive properties of 3'-substituted deschloroepibatidine analogues. Novel nicotinic antagonists.
Carroll FI; Ma W; Yokota Y; Lee JR; Brieaddy LE; Navarro HA; Damaj MI; Martin BR
J Med Chem; 2005 Feb; 48(4):1221-8. PubMed ID: 15715488
[TBL] [Abstract][Full Text] [Related]
18. Stereoselective synthesis of (+/-)-epibatidine analog:(+/-)-2beta-(2-chloro-5-pyridinyl)-8-azabicyclo[3.2.1] octane.
Kim YH; Won DY; Oh CY; Woo NT; Park YH; Jeong JH; Ham WH
Arch Pharm Res; 1999 Jun; 22(3):300-1. PubMed ID: 10403134
[TBL] [Abstract][Full Text] [Related]
19. Structure-activity studies of diazabicyclo[3.3.0]octane-substituted pyrazines and pyridines as potent α4β2 nicotinic acetylcholine receptor ligands.
Scanio MJ; Shi L; Bunnelle WH; Anderson DJ; Helfrich RJ; Malysz J; Thorin-Hagene KK; Van Handel CE; Marsh KC; Lee CH; Gopalakrishnan M
J Med Chem; 2011 Nov; 54(21):7678-92. PubMed ID: 21962147
[TBL] [Abstract][Full Text] [Related]
20. 7-substituted 2-azabicyclo[2.2.1]heptanes as key intermediates for the synthesis of novel epibatidine analogues; synthesis of syn-and anti-isoepiboxidine.
Malpass JR; White R
J Org Chem; 2004 Aug; 69(16):5328-34. PubMed ID: 15287778
[TBL] [Abstract][Full Text] [Related]
[Next] [New Search]
