76 related articles for article (PubMed ID: 16621575)
1. Closing in on the AMPA receptor: synthesis and evaluation of 2-acetyl-1-(4'-chlorophenyl)-6-methoxy-7-[11C]methoxy-1,2,3,4-tetrahydroisoquinoline as a potential PET tracer.
Arstad E; Gitto R; Chimirri A; Caruso R; Constanti A; Turton D; Hume SP; Ahmad R; Pilowsky LS; Luthra SK
Bioorg Med Chem; 2006 Jul; 14(14):4712-7. PubMed ID: 16621575
[TBL] [Abstract][Full Text] [Related]
2. Synthesis of carbon-11 and fluorine-18 labeled N-acetyl-1-aryl-6,7-dimethoxy-1,2,3,4-tetrahydroisoquinoline derivatives as new potential PET AMPA receptor ligands.
Gao M; Kong D; Clearfield A; Zheng QH
Bioorg Med Chem Lett; 2006 Apr; 16(8):2229-33. PubMed ID: 16455250
[TBL] [Abstract][Full Text] [Related]
3. Towards NR2B receptor selective imaging agents for PET-synthesis and evaluation of N-[11C]-(2-methoxy)benzyl (E)-styrene-, 2-naphthyl- and 4-trifluoromethoxyphenylamidine.
Arstad E; Platzer S; Berthele A; Pilowsky LS; Luthra SK; Wester HJ; Henriksen G
Bioorg Med Chem; 2006 Sep; 14(18):6307-13. PubMed ID: 16777419
[TBL] [Abstract][Full Text] [Related]
4. Synthesis, resolution, stereochemistry, and molecular modeling of (R)- and (S)-2-acetyl-1-(4'-chlorophenyl)-6,7-dimethoxy-1,2,3,4-tetrahydroisoquinoline AMPAR antagonists.
Gitto R; Ficarra R; Stancanelli R; Guardo M; De Luca L; Barreca ML; Pagano B; Rotondo A; Bruno G; Russo E; De Sarro G; Chimirri A
Bioorg Med Chem; 2007 Aug; 15(16):5417-23. PubMed ID: 17566746
[TBL] [Abstract][Full Text] [Related]
5. In vitro and in vivo evaluation of [11C]MPEPy as a potential PET ligand for mGlu5 receptors.
Severance AJ; Parsey RV; Kumar JS; Underwood MD; Arango V; Majo VJ; Prabhakaran J; Simpson NR; Van Heertum RL; Mann JJ
Nucl Med Biol; 2006 Nov; 33(8):1021-7. PubMed ID: 17127176
[TBL] [Abstract][Full Text] [Related]
6. [2-11C]isopropyl-, [1-11C]ethyl-, and [11C]methyl-labeled phenoxyphenyl acetamide derivatives as positron emission tomography ligands for the peripheral benzodiazepine receptor: radiosynthesis, uptake, and in vivo binding in brain.
Zhang MR; Ogawa M; Maeda J; Ito T; Noguchi J; Kumata K; Okauchi T; Suhara T; Suzuki K
J Med Chem; 2006 May; 49(9):2735-42. PubMed ID: 16640334
[TBL] [Abstract][Full Text] [Related]
7. Discovery of a novel and highly potent noncompetitive AMPA receptor antagonist.
Gitto R; Barreca ML; De Luca L; De Sarro G; Ferreri G; Quartarone S; Russo E; Constanti A; Chimirri A
J Med Chem; 2003 Jan; 46(1):197-200. PubMed ID: 12502375
[TBL] [Abstract][Full Text] [Related]
8. Synthesis and in vivo evaluation of [11C]SN003 as a PET ligand for CRF1 receptors.
Kumar JS; Majo VJ; Sullivan GM; Prabhakaran J; Simpson NR; Van Heertum RL; Mann JJ; Parsey RV
Bioorg Med Chem; 2006 Jun; 14(12):4029-34. PubMed ID: 16529935
[TBL] [Abstract][Full Text] [Related]
9. Novel potent anticonvulsant agent containing a tetrahydroisoquinoline skeleton.
Gitto R; Caruso R; Pagano B; De Luca L; Citraro R; Russo E; De Sarro G; Chimirri A
J Med Chem; 2006 Sep; 49(18):5618-22. PubMed ID: 16942035
[TBL] [Abstract][Full Text] [Related]
10. Radiosynthesis and biodistribution of a histamine H3 receptor antagonist 4-[3-(4-piperidin-1-yl-but-1-ynyl)-[11C]benzyl]-morpholine: evaluation of a potential PET ligand.
Airaksinen AJ; Jablonowski JA; van der Mey M; Barbier AJ; Klok RP; Verbeek J; Schuit R; Herscheid JD; Leysen JE; Carruthers NI; Lammertsma AA; Windhorst AD
Nucl Med Biol; 2006 Aug; 33(6):801-10. PubMed ID: 16934699
[TBL] [Abstract][Full Text] [Related]
11. Synthetic approaches and bio-distribution studies of [11C]methyl-phenidate.
Patt M; Solbach C; Wüllner U; Blocher A; Stahlschmidt A; Gündisch D; Kovar KA; Machulla HJ
J Pharm Pharm Sci; 2007; 10(2):312s-320s. PubMed ID: 17718934
[TBL] [Abstract][Full Text] [Related]
12. Synthesis and preliminary biological evaluation of new carbon-11 labeled tetrahydroisoquinoline derivatives as SERM radioligands for PET imaging of ER expression in breast cancer.
Gao M; Wang M; Miller KD; Sledge GW; Zheng QH
Eur J Med Chem; 2008 Oct; 43(10):2211-9. PubMed ID: 18272256
[TBL] [Abstract][Full Text] [Related]
13. Human PET studies of metabotropic glutamate receptor subtype 5 with 11C-ABP688.
Ametamey SM; Treyer V; Streffer J; Wyss MT; Schmidt M; Blagoev M; Hintermann S; Auberson Y; Gasparini F; Fischer UC; Buck A
J Nucl Med; 2007 Feb; 48(2):247-52. PubMed ID: 17268022
[TBL] [Abstract][Full Text] [Related]
14. Measurement of glycine binding site of N-methyl-D-asparate receptors in living human brain using 4-acetoxy derivative of L-703,717, 4-acetoxy-7-chloro-3-[3-(4-[11c] methoxybenzyl) phenyl]-2(1H)-quinolone (AcL703) with positron emission tomography.
Matsumoto R; Haradahira T; Ito H; Fujimura Y; Seki C; Ikoma Y; Maeda J; Arakawa R; Takano A; Takahashi H; Higuchi M; Suzuki K; Fukui K; Suhara T
Synapse; 2007 Oct; 61(10):795-800. PubMed ID: 17598152
[TBL] [Abstract][Full Text] [Related]
15. Design, synthesis, and binding affinities of potential positron emission tomography (PET) ligands for visualization of brain dopamine D3 receptors.
Leopoldo M; Lacivita E; De Giorgio P; Colabufo NA; Niso M; Berardi F; Perrone R
J Med Chem; 2006 Jan; 49(1):358-65. PubMed ID: 16392820
[TBL] [Abstract][Full Text] [Related]
16. Effects of non-competitive AMPA receptor antagonists injected into some brain areas of WAG/Rij rats, an animal model of generalized absence epilepsy.
Citraro R; Russo E; Gratteri S; Di Paola ED; Ibbadu GF; Curinga C; Gitto R; Chimirri A; Donato G; De Sarro G
Neuropharmacology; 2006 Nov; 51(6):1058-67. PubMed ID: 16901515
[TBL] [Abstract][Full Text] [Related]
17. Evaluation of the novel 5-HT4 receptor PET ligand [11C]SB207145 in the Göttingen minipig.
Kornum BR; Lind NM; Gillings N; Marner L; Andersen F; Knudsen GM
J Cereb Blood Flow Metab; 2009 Jan; 29(1):186-96. PubMed ID: 18797470
[TBL] [Abstract][Full Text] [Related]
18. Synthesis and in vivo evaluation of fluorine-18 and iodine-123 labeled 2beta-carbo(2-fluoroethoxy)-3beta-(4'-((Z)-2-iodoethenyl)phenyl)nortropane as a candidate serotonin transporter imaging agent.
Plisson C; Stehouwer JS; Voll RJ; Howell L; Votaw JR; Owens MJ; Goodman MM
J Med Chem; 2007 Sep; 50(19):4553-60. PubMed ID: 17705359
[TBL] [Abstract][Full Text] [Related]
19. Determination of a potent non-competitive AMPA receptor antagonist in rat brain.
Rizzo M; Ventrice D; Casale F; De Sarro G; Gitto R; Chimirri A
J Chromatogr B Analyt Technol Biomed Life Sci; 2007 May; 850(1-2):161-7. PubMed ID: 17150419
[TBL] [Abstract][Full Text] [Related]
20. [11C]AZ10419369: a selective 5-HT1B receptor radioligand suitable for positron emission tomography (PET). Characterization in the primate brain.
Pierson ME; Andersson J; Nyberg S; McCarthy DJ; Finnema SJ; Varnäs K; Takano A; Karlsson P; Gulyás B; Medd AM; Lee CM; Powell ME; Heys JR; Potts W; Seneca N; Mrzljak L; Farde L; Halldin C
Neuroimage; 2008 Jul; 41(3):1075-85. PubMed ID: 18434202
[TBL] [Abstract][Full Text] [Related]
[Next] [New Search]
