166 related articles for article (PubMed ID: 16641315)
21. Characterization of the subtype selectivity of the allosteric modulator heptane-1,7-bis-(dimethyl-3'-phthalimidopropyl) ammonium bromide (C7/3-phth) at cloned muscarinic acetylcholine receptors.
Christopoulos A; Sorman JL; Mitchelson F; El-Fakahany EE
Biochem Pharmacol; 1999 Jan; 57(2):171-9. PubMed ID: 9890565
[TBL] [Abstract][Full Text] [Related]
22. Subtype selectivity of the positive allosteric action of alcuronium at cloned M1-M5 muscarinic acetylcholine receptors.
Jakubík J; Bacáková L; el-Fakahany EE; Tucek S
J Pharmacol Exp Ther; 1995 Sep; 274(3):1077-83. PubMed ID: 7562472
[TBL] [Abstract][Full Text] [Related]
23. Cooperative interactions at M2 muscarinic acetylcholine receptors: structure/activity relationships in stepwise shortened bispyridinium- and bis(ammonio)alkane-type allosteric modulators.
Gilsbach R; Grossmüller M; Alptüzün V; Erciyas E; Tränkle C; Holzgrabe U; Mohr K
Neurochem Res; 2003 Apr; 28(3-4):667-73. PubMed ID: 12675159
[TBL] [Abstract][Full Text] [Related]
24. Allosteric interactions at muscarinic cholinoceptors.
Christopoulos A; Lanzafame A; Mitchelson F
Clin Exp Pharmacol Physiol; 1998; 25(3-4):185-94. PubMed ID: 9590567
[TBL] [Abstract][Full Text] [Related]
25. M2 Subtype preferring dibenzodiazepinone-type muscarinic receptor ligands: Effect of chemical homo-dimerization on orthosteric (and allosteric?) binding.
Keller M; Tränkle C; She X; Pegoli A; Bernhardt G; Buschauer A; Read RW
Bioorg Med Chem; 2015 Jul; 23(14):3970-90. PubMed ID: 25650309
[TBL] [Abstract][Full Text] [Related]
26. Site-directed mutagenesis reveals two epitopes involved in the subtype selectivity of the allosteric interactions of gallamine at muscarinic acetylcholine receptors.
Gnagey AL; Seidenberg M; Ellis J
Mol Pharmacol; 1999 Dec; 56(6):1245-53. PubMed ID: 10570052
[TBL] [Abstract][Full Text] [Related]
27. The allosteric site regulates the voltage sensitivity of muscarinic receptors.
Hoppe A; Marti-Solano M; Drabek M; Bünemann M; Kolb P; Rinne A
Cell Signal; 2018 Jan; 42():114-126. PubMed ID: 29056499
[TBL] [Abstract][Full Text] [Related]
28. The allosteric interaction of otenzepad (AF-DX 116) at muscarinic M2 receptors in guinea pig atria.
Lanzafame A; Christopoulos A; Mitchelson F
Eur J Pharmacol; 2001 Mar; 416(3):235-44. PubMed ID: 11290374
[TBL] [Abstract][Full Text] [Related]
29. Allosteric effects of four stereoisomers of a fused indole ring system with 3H-N-methylscopolamine and acetylcholine at M1-M4 muscarinic receptors.
Lazareno S; Birdsall B; Fukazawa T; Gharagozloo P; Hashimoto T; Kuwano H; Popham A; Sugimoto M; Birdsall NJ
Life Sci; 1999; 64(6-7):519-26. PubMed ID: 10069518
[TBL] [Abstract][Full Text] [Related]
30. Contribution of lateral substituents in symmetrical and non-symmetrical heptane-bisammonio compounds to the allosteric stabilization of N-methylscopolamine binding to muscarinic M2 receptors.
Staudt M; Tränkle C; Mohr K; Holzgrabe U
Arch Pharm (Weinheim); 2003 Aug; 336(8):385-9. PubMed ID: 14502759
[TBL] [Abstract][Full Text] [Related]
31. Positive cooperativity of acetylcholine and other agonists with allosteric ligands on muscarinic acetylcholine receptors.
Jakubík J; Bacáková L; El-Fakahany EE; Tucek S
Mol Pharmacol; 1997 Jul; 52(1):172-9. PubMed ID: 9224827
[TBL] [Abstract][Full Text] [Related]
32. Characterization of methanthelinium binding and function at human M
Irmen M; Holze J; Bödefeld T; Tränkle C
Naunyn Schmiedebergs Arch Pharmacol; 2018 Oct; 391(10):1037-1052. PubMed ID: 29938305
[TBL] [Abstract][Full Text] [Related]
33. M2 receptor binding of the selective antagonist AF-DX 384: possible involvement of the common allosteric site.
Tränkle C; Andresen I; Lambrecht G; Mohr K
Mol Pharmacol; 1998 Feb; 53(2):304-12. PubMed ID: 9463489
[TBL] [Abstract][Full Text] [Related]
34. Muscarinic allosteric enhancers of ligand binding: pivotal pharmacophoric elements in hexamethonio-type agents.
Muth M; Sennwitz M; Mohr K; Holzgrabe U
J Med Chem; 2005 Mar; 48(6):2212-7. PubMed ID: 15771463
[TBL] [Abstract][Full Text] [Related]
35. Allosteric interactions of staurosporine and other indolocarbazoles with N-[methyl-(3)H]scopolamine and acetylcholine at muscarinic receptor subtypes: identification of a second allosteric site.
Lazareno S; Popham A; Birdsall NJ
Mol Pharmacol; 2000 Jul; 58(1):194-207. PubMed ID: 10860942
[TBL] [Abstract][Full Text] [Related]
36. Competitive and allosteric interactions of 6-chloro-5,10-dihydro-5-[(1-methyl-4-piperidinyl)acetyl]-11H-di benzo[b,e][1, 4]diazepine-11-one hydrochloride (UH-AH 37) at muscarinic receptors, via distinct epitopes.
Ellis J; Seidenberg M
Biochem Pharmacol; 1999 Jan; 57(2):181-6. PubMed ID: 9890566
[TBL] [Abstract][Full Text] [Related]
37. Subtype-selective positive cooperative interactions between brucine analogues and acetylcholine at muscarinic receptors: radioligand binding studies.
Lazareno S; Gharagozloo P; Kuonen D; Popham A; Birdsall NJ
Mol Pharmacol; 1998 Mar; 53(3):573-89. PubMed ID: 9495826
[TBL] [Abstract][Full Text] [Related]
38. Divergent modes of action among cationic allosteric modulators of muscarinic M2 receptors.
Tränkle C; Mohr K
Mol Pharmacol; 1997 Apr; 51(4):674-82. PubMed ID: 9106634
[TBL] [Abstract][Full Text] [Related]
39. Atypical muscarinic allosteric modulation: cooperativity between modulators and their atypical binding topology in muscarinic M2 and M2/M5 chimeric receptors.
Tränkle C; Dittmann A; Schulz U; Weyand O; Buller S; Jöhren K; Heller E; Birdsall NJ; Holzgrabe U; Ellis J; Höltje HD; Mohr K
Mol Pharmacol; 2005 Dec; 68(6):1597-610. PubMed ID: 16157694
[TBL] [Abstract][Full Text] [Related]
40. Influence of ligand choice on the apparent binding profile of gallamine to cardiac muscarinic receptors. Identification of three main types of gallamine-muscarinic receptor interactions.
Lee NH; el-Fakahany EE
J Pharmacol Exp Ther; 1988 Sep; 246(3):829-38. PubMed ID: 3418516
[TBL] [Abstract][Full Text] [Related]
[Previous] [Next] [New Search]