309 related articles for article (PubMed ID: 16817895)
1. Inhibition of recombinant human maltase glucoamylase by salacinol and derivatives.
Rossi EJ; Sim L; Kuntz DA; Hahn D; Johnston BD; Ghavami A; Szczepina MG; Kumar NS; Sterchi EE; Nichols BL; Pinto BM; Rose DR
FEBS J; 2006 Jun; 273(12):2673-83. PubMed ID: 16817895
[TBL] [Abstract][Full Text] [Related]
2. New synthetic routes to chain-extended selenium, sulfur, and nitrogen analogues of the naturally occurring glucosidase inhibitor salacinol and their inhibitory activities against recombinant human maltase glucoamylase.
Liu H; Nasi R; Jayakanthan K; Sim L; Heipel H; Rose DR; Pinto BM
J Org Chem; 2007 Aug; 72(17):6562-72. PubMed ID: 17658854
[TBL] [Abstract][Full Text] [Related]
3. New glucosidase inhibitors from an ayurvedic herbal treatment for type 2 diabetes: structures and inhibition of human intestinal maltase-glucoamylase with compounds from Salacia reticulata.
Sim L; Jayakanthan K; Mohan S; Nasi R; Johnston BD; Pinto BM; Rose DR
Biochemistry; 2010 Jan; 49(3):443-51. PubMed ID: 20039683
[TBL] [Abstract][Full Text] [Related]
4. Mapping the intestinal alpha-glucogenic enzyme specificities of starch digesting maltase-glucoamylase and sucrase-isomaltase.
Jones K; Sim L; Mohan S; Kumarasamy J; Liu H; Avery S; Naim HY; Quezada-Calvillo R; Nichols BL; Pinto BM; Rose DR
Bioorg Med Chem; 2011 Jul; 19(13):3929-34. PubMed ID: 21669536
[TBL] [Abstract][Full Text] [Related]
5. Studies directed toward the stereochemical structure determination of the naturally occurring glucosidase inhibitor, kotalanol: synthesis and inhibitory activities against human maltase glucoamylase of seven-carbon, chain-extended homologues of salacinol.
Nasi R; Patrick BO; Sim L; Rose DR; Pinto BM
J Org Chem; 2008 Aug; 73(16):6172-81. PubMed ID: 18651773
[TBL] [Abstract][Full Text] [Related]
6. A new class of glucosidase inhibitor: analogues of the naturally occurring glucosidase inhibitor salacinol with different ring heteroatom substituents and acyclic chain extension.
Liu H; Sim L; Rose DR; Pinto BM
J Org Chem; 2006 Apr; 71(8):3007-13. PubMed ID: 16599595
[TBL] [Abstract][Full Text] [Related]
7. New chain-extended analogues of salacinol and blintol and their glycosidase inhibitory activities. Mapping the active-site requirements of human maltase glucoamylase.
Nasi R; Sim L; Rose DR; Pinto BM
J Org Chem; 2007 Jan; 72(1):180-6. PubMed ID: 17194097
[TBL] [Abstract][Full Text] [Related]
8. Synthesis of a salacinol analogue and its alpha-glucosidase inhibitory activity.
Shao Y; Osamu M; Kazuya Y; Yoshiharu M; Eriko Y; Toshie M; Genzoh T; Hisashi M; Masayuki Y; You QD
Yao Xue Xue Bao; 2006 Jul; 41(7):647-53. PubMed ID: 17007358
[TBL] [Abstract][Full Text] [Related]
9. Synthesis of phosphate derivatives related to the glycosidase inhibitor salacinol.
Bhat RG; Kumar NS; Pinto BM
Carbohydr Res; 2007 Sep; 342(12-13):1934-42. PubMed ID: 17572396
[TBL] [Abstract][Full Text] [Related]
10. Synthesis of 2-deoxy-2-fluoro and 1,2-ene derivatives of the naturally occurring glycosidase inhibitor, salacinol, and their inhibitory activities against recombinant human maltase glucoamylase.
Choubdar N; Sim L; Rose DR; Pinto BM
Carbohydr Res; 2008 Apr; 343(5):951-6. PubMed ID: 18295754
[TBL] [Abstract][Full Text] [Related]
11. Docking and SAR studies of salacinol derivatives as alpha-glucosidase inhibitors.
Nakamura S; Takahira K; Tanabe G; Morikawa T; Sakano M; Ninomiya K; Yoshikawa M; Muraoka O; Nakanishi I
Bioorg Med Chem Lett; 2010 Aug; 20(15):4420-3. PubMed ID: 20598536
[TBL] [Abstract][Full Text] [Related]
12. Naturally occurring sulfonium-ion glucosidase inhibitors and their derivatives: a promising class of potential antidiabetic agents.
Mohan S; Eskandari R; Pinto BM
Acc Chem Res; 2014 Jan; 47(1):211-25. PubMed ID: 23964564
[TBL] [Abstract][Full Text] [Related]
13. Probing the active-site requirements of human intestinal N-terminal maltase-glucoamylase: Synthesis and enzyme inhibitory activities of a six-membered ring nitrogen analogue of kotalanol and its de-O-sulfonated derivative.
Mohan S; Sim L; Rose DR; Pinto BM
Bioorg Med Chem; 2010 Nov; 18(22):7794-8. PubMed ID: 20970346
[TBL] [Abstract][Full Text] [Related]
14. Synthesis of D-lyxitol and D-ribitol analogues of the naturally occurring glycosidase inhibitor salacinol.
Kumar NS; Pinto BM
Carbohydr Res; 2005 Dec; 340(17):2612-9. PubMed ID: 16198322
[TBL] [Abstract][Full Text] [Related]
15. Synthesis of analogues of salacinol containing a carboxylate inner salt and their inhibitory activities against human maltase glucoamylase.
Chen W; Sim L; Rose DR; Pinto BM
Carbohydr Res; 2007 Sep; 342(12-13):1661-7. PubMed ID: 17597595
[TBL] [Abstract][Full Text] [Related]
16. Synthesis and biological evaluation of deoxy salacinols, the role of polar substituents in the side chain on the alpha-glucosidase inhibitory activity.
Muraoka O; Yoshikai K; Takahashi H; Minematsu T; Lu G; Tanabe G; Wang T; Matsuda H; Yoshikawa M
Bioorg Med Chem; 2006 Jan; 14(2):500-9. PubMed ID: 16198577
[TBL] [Abstract][Full Text] [Related]
17. In silico design, synthesis and evaluation of 3'-O-benzylated analogs of salacinol, a potent α-glucosidase inhibitor isolated from an Ayurvedic traditional medicine "Salacia".
Tanabe G; Nakamura S; Tsutsui N; Balakishan G; Xie W; Tsuchiya S; Akaki J; Morikawa T; Ninomiya K; Nakanishi I; Yoshikawa M; Muraoka O
Chem Commun (Camb); 2012 Sep; 48(69):8646-8. PubMed ID: 22820468
[TBL] [Abstract][Full Text] [Related]
18. Synthesis, enzymatic activity, and X-ray crystallography of an unusual class of amino acids.
Chen W; Kuntz DA; Hamlet T; Sim L; Rose DR; Mario Pinto B
Bioorg Med Chem; 2006 Dec; 14(24):8332-40. PubMed ID: 17010621
[TBL] [Abstract][Full Text] [Related]
19. Zwitterionic glycosidase inhibitors: salacinol and related analogues.
Mohan S; Pinto BM
Carbohydr Res; 2007 Sep; 342(12-13):1551-80. PubMed ID: 17559821
[TBL] [Abstract][Full Text] [Related]
20. Synthesis and glycosidase inhibitory activities of chain-modified analogues of the glycosidase inhibitors salacinol and blintol.
Nasi R; Sim L; Rose DR; Pinto BM
Carbohydr Res; 2007 Sep; 342(12-13):1888-94. PubMed ID: 17359953
[TBL] [Abstract][Full Text] [Related]
[Next] [New Search]
