BIOMARKERS

Molecular Biopsy of Human Tumors

- a resource for Precision Medicine *

211 related articles for article (PubMed ID: 1686464)

  • 1. Carbamate ester prodrugs of dopaminergic compounds: synthesis, stability, and bioconversion.
    Hansen KT; Faarup P; Bundgaard H
    J Pharm Sci; 1991 Aug; 80(8):793-8. PubMed ID: 1686464
    [TBL] [Abstract][Full Text] [Related]  

  • 2. A carbamate-based approach to primaquine prodrugs: antimalarial activity, chemical stability and enzymatic activation.
    Mata G; do Rosário VE; Iley J; Constantino L; Moreira R
    Bioorg Med Chem; 2012 Jan; 20(2):886-92. PubMed ID: 22189276
    [TBL] [Abstract][Full Text] [Related]  

  • 3. Amino Acid Carbamates As Prodrugs Of Resveratrol.
    Mattarei A; Azzolini M; La Spina M; Zoratti M; Paradisi C; Biasutto L
    Sci Rep; 2015 Oct; 5():15216. PubMed ID: 26463125
    [TBL] [Abstract][Full Text] [Related]  

  • 4. Synthesis and evaluation of carbamate prodrugs of a phenolic compound.
    Igarashi Y; Yanagisawa E; Ohshima T; Takeda S; Aburada M; Miyamoto K
    Chem Pharm Bull (Tokyo); 2007 Feb; 55(2):328-33. PubMed ID: 17268110
    [TBL] [Abstract][Full Text] [Related]  

  • 5. Orally active carbamate prodrugs of the selective dopamine agonist N-0437: in-vivo activities in the 6-OHDA turning model and in-vitro activities.
    den Daas I; de Boer P; Tepper PG; Rollema H; Horn AS
    J Pharm Pharmacol; 1991 Jan; 43(1):11-6. PubMed ID: 1676052
    [TBL] [Abstract][Full Text] [Related]  

  • 6. Synthesis and in vitro/in vivo evaluation of novel oral N-alkyl- and N,N-dialkyl-carbamate esters of entacapone.
    Savolainen J; Leppanen J; Forsberg M; Taipale H; Nevalainen T; Huuskonen J; Gynther J; Mannisto PT; Jarvinen T
    Life Sci; 2000; 67(2):205-16. PubMed ID: 10901288
    [TBL] [Abstract][Full Text] [Related]  

  • 7. N-Monosubstituted Methoxy-oligo(ethylene glycol) Carbamate Ester Prodrugs of Resveratrol.
    Mattarei A; Azzolini M; Zoratti M; Biasutto L; Paradisi C
    Molecules; 2015 Sep; 20(9):16085-102. PubMed ID: 26404221
    [TBL] [Abstract][Full Text] [Related]  

  • 8. Improving the oral bioavailability of tapentadol via a carbamate prodrug approach: synthesis, bioactivation, and pharmacokinetics.
    Li Y; Wang Y; Zhang R; Liu C; Wei Y; Sun J; He Z; Xu Y; Zhang T
    Drug Deliv Transl Res; 2018 Oct; 8(5):1335-1344. PubMed ID: 29777509
    [TBL] [Abstract][Full Text] [Related]  

  • 9. Synthesis and Evaluation as Prodrugs of Hydrophilic Carbamate Ester Analogues of Resveratrol.
    Azzolini M; Mattarei A; La Spina M; Marotta E; Zoratti M; Paradisi C; Biasutto L
    Mol Pharm; 2015 Sep; 12(9):3441-54. PubMed ID: 26252229
    [TBL] [Abstract][Full Text] [Related]  

  • 10. Chemical and enzymatic stability of amino acid prodrugs containing methoxy, ethoxy and propylene glycol linkers.
    Gupta D; Gupta SV; Lee KD; Amidon GL
    Mol Pharm; 2009; 6(5):1604-11. PubMed ID: 19566080
    [TBL] [Abstract][Full Text] [Related]  

  • 11. Cyclization-activated prodrugs: N-(substituted 2-hydroxyphenyl and 2-hydroxypropyl)carbamates based on ring-opened derivatives of active benzoxazolones and oxazolidinones as mutual prodrugs of acetaminophen.
    Vigroux A; Bergon M; Zedde C
    J Med Chem; 1995 Sep; 38(20):3983-94. PubMed ID: 7562932
    [TBL] [Abstract][Full Text] [Related]  

  • 12. Triazene drug metabolites. Part 17: Synthesis and plasma hydrolysis of acyloxymethyl carbamate derivatives of antitumour triazenes.
    Carvalho E; Francisco AP; Iley J; Rosa E
    Bioorg Med Chem; 2000 Jul; 8(7):1719-25. PubMed ID: 10976519
    [TBL] [Abstract][Full Text] [Related]  

  • 13. Synthesis, characterization, and biological evaluation of novel diclofenac prodrugs.
    Bandgar BP; Sarangdhar RJ; Ahamed FA; Viswakarma S
    J Med Chem; 2011 Mar; 54(5):1202-10. PubMed ID: 21250699
    [TBL] [Abstract][Full Text] [Related]  

  • 14. New 3'-azido-3'-deoxythymidin-5'-yl O-(omega-hydroxyalkyl) carbonate prodrugs: synthesis and anti-HIV evaluation.
    Vlieghe P; Bihel F; Clerc T; Pannecouque C; Witvrouw M; De Clercq E; Salles JP; Chermann JC; Kraus JL
    J Med Chem; 2001 Mar; 44(5):777-86. PubMed ID: 11262088
    [TBL] [Abstract][Full Text] [Related]  

  • 15. Synthesis, chemical and enzymatic hydrolysis, and bioavailability evaluation in rabbits of metronidazole amino acid ester prodrugs with enhanced water solubility.
    Mahfouz NM; Hassan MA
    J Pharm Pharmacol; 2001 Jun; 53(6):841-8. PubMed ID: 11428660
    [TBL] [Abstract][Full Text] [Related]  

  • 16. In vitro and in vivo evaluations of the metabolism, pharmacokinetics, and bioavailability of ester prodrugs of L-767,679, a potent fibrinogen receptor antagonist: an approach for the selection of a prodrug candidate.
    Prueksaritanont T; Gorham LM; Breslin MJ; Hutchinson JH; Hartman GD; Vyas KP; Baillie TA
    Drug Metab Dispos; 1997 Aug; 25(8):978-84. PubMed ID: 9280406
    [TBL] [Abstract][Full Text] [Related]  

  • 17. Synthesis, characterization and in vitro evaluation of substituted N-(2-phenylcyclopropyl)carbamates as acetyl- and butyrylcholinesterase inhibitors.
    Horáková E; Drabina P; Brož B; Štěpánková Š; Vorčáková K; Královec K; Havelek R; Sedlák M
    J Enzyme Inhib Med Chem; 2016; 31(sup3):173-179. PubMed ID: 27476673
    [TBL] [Abstract][Full Text] [Related]  

  • 18. Phosphoryloxymethyl carbamates and carbonates--novel water-soluble prodrugs for amines and hindered alcohols.
    Safadi M; Oliyai R; Stella VJ
    Pharm Res; 1993 Sep; 10(9):1350-5. PubMed ID: 8234176
    [TBL] [Abstract][Full Text] [Related]  

  • 19. Glycolamide esters as biolabile prodrugs of carboxylic acid agents: synthesis, stability, bioconversion, and physicochemical properties.
    Nielsen NM; Bundgaard H
    J Pharm Sci; 1988 Apr; 77(4):285-98. PubMed ID: 3379586
    [TBL] [Abstract][Full Text] [Related]  

  • 20. Carbamate ester derivatives as potential prodrugs of the presynaptic dopamine autoreceptor agonist (-)-3-(3-hydroxyphenyl)-N-propylpiperidine.
    Thorberg SO; Berg S; Lundström J; Pettersson B; Wijkström A; Sanchez D; Lindberg P; Nilsson JL
    J Med Chem; 1987 Nov; 30(11):2008-12. PubMed ID: 3669008
    [TBL] [Abstract][Full Text] [Related]  

    [Next]    [New Search]
    of 11.