116 related articles for article (PubMed ID: 16930912)
21. Inhibition of benzalkonium chloride-induced skin inflammation in mice by an indol-1-ylpropan-2-one inhibitor of cytosolic phospholipase A2 α.
Roebrock K; Wolf M; Bovens S; Lehr M; Sunderkötter C
Br J Dermatol; 2012 Feb; 166(2):306-16. PubMed ID: 21929537
[TBL] [Abstract][Full Text] [Related]
22. In vitro biotransformation of thiazopyr by rat liver microsomes: oxidative cleavage of a carboxylic methylester by monooxygenases.
Feng PC; Solsten RT
Xenobiotica; 1994 Aug; 24(8):729-34. PubMed ID: 7839696
[TBL] [Abstract][Full Text] [Related]
23. 1-Indol-1-yl-propan-2-ones and related heterocyclic compounds as dual inhibitors of cytosolic phospholipase A(2)alpha and fatty acid amide hydrolase.
Forster L; Ludwig J; Kaptur M; Bovens S; Elfringhoff AS; Holtfrerich A; Lehr M
Bioorg Med Chem; 2010 Jan; 18(2):945-52. PubMed ID: 20005725
[TBL] [Abstract][Full Text] [Related]
24. Application of electrospray ionization hybrid ion trap/time-of-flight mass spectrometry in the rapid characterization of quinocetone metabolites formed in vitro.
Liu ZY; Huang LL; Chen DM; Dai MH; Tao YF; Wang YL; Yuan ZH
Anal Bioanal Chem; 2010 Feb; 396(3):1259-71. PubMed ID: 20020112
[TBL] [Abstract][Full Text] [Related]
25. Metabolism of amiodarone (part I): identification of a new hydroxylated metabolite of amiodarone.
Ha HR; Bigler L; Binder M; Kozlik P; Stieger B; Hesse M; Altorfer HR; Follath F
Drug Metab Dispos; 2001 Feb; 29(2):152-8. PubMed ID: 11159805
[TBL] [Abstract][Full Text] [Related]
26. Comparative metabolism of Lappaconitine in rat and human liver microsomes and in vivo of rat using ultra high-performance liquid chromatography-quadrupole/time-of-flight mass spectrometry.
Yang S; Zhang H; Beier RC; Sun F; Cao X; Shen J; Wang Z; Zhang S
J Pharm Biomed Anal; 2015 Jun; 110():1-11. PubMed ID: 25796978
[TBL] [Abstract][Full Text] [Related]
27. Liquid chromatographic-electrospray mass spectrometric determination (LC-ESI-MS) of phase II metabolites of flobufen in rat liver microsomes-Chiral discrimination.
Babú YN; Nemec M; Solich P; Wsól V
Talanta; 2008 Apr; 75(2):494-502. PubMed ID: 18371912
[TBL] [Abstract][Full Text] [Related]
28. 1-(5-carboxyindol-1-yl)propan-2-one inhibitors of human cytosolic phospholipase A(2)alpha with reduced lipophilicity: synthesis, biological activity, metabolic stability, solubility, bioavailability, and topical in vivo activity.
Drews A; Bovens S; Roebrock K; Sunderkötter C; Reinhardt D; Schäfers M; van der Velde A; Schulze Elfringhoff A; Fabian J; Lehr M
J Med Chem; 2010 Jul; 53(14):5165-78. PubMed ID: 20583844
[TBL] [Abstract][Full Text] [Related]
29. Metabolism and excretion of 5-ethyl-2-{5-[4-(2-hydroxyethyl)piperazine-1-sulfonyl]-2-propoxyphenyl}-7-propyl-3,5-dihydropyrrolo[3,2-d]-pyrimidin-4-one (SK3530) in rats.
Lee J; Yoo HH; Rhim KJ; Sohn DR; Kim DH
Rapid Commun Mass Spectrom; 2007; 21(7):1139-49. PubMed ID: 17318927
[TBL] [Abstract][Full Text] [Related]
30. Rapid structural characterization of in vivo and in vitro metabolites of tinoridine using UHPLC-QTOF-MS/MS and in silico toxicological screening of its metabolites.
Kalariya PD; Patel PN; Kavya P; Sharma M; Garg P; Srinivas R; Talluri MV
J Mass Spectrom; 2015 Nov; 50(11):1222-33. PubMed ID: 26505767
[TBL] [Abstract][Full Text] [Related]
31. Structure-activity relationship studies on 1-(5-carboxyindol-1-yl)-propan-2-one inhibitors of human cytosolic phospholipase A2α: variation of the activated ketone moiety.
Kaptur M; Elfringhoff AS; Lehr M
Bioorg Med Chem Lett; 2011 Mar; 21(6):1773-6. PubMed ID: 21316224
[TBL] [Abstract][Full Text] [Related]
32. A new metabolite of nodakenetin by rat liver microsomes and its quantification by RP-HPLC method.
Zhang P; Yang XW
Biomed Chromatogr; 2010 Feb; 24(2):216-21. PubMed ID: 19572262
[TBL] [Abstract][Full Text] [Related]
33. The identification of in vitro metabolites of CKD-732 by liquid chromatography/tandem mass spectrometry.
Myung SW; Kim HY; Min HK; Kim DH; Kim M; Cho HW; Lee HS; Kim JK; Hong CI
Rapid Commun Mass Spectrom; 2002; 16(21):2048-53. PubMed ID: 12391579
[TBL] [Abstract][Full Text] [Related]
34. Structure of the glutathione adduct of activated 3-methylindole indicates that an imine methide is the electrophilic intermediate.
Nocerini MR; Yost GS; Carlson JR; Liberato DJ; Breeze RG
Drug Metab Dispos; 1985; 13(6):690-4. PubMed ID: 2867872
[TBL] [Abstract][Full Text] [Related]
35. Biotransformation of the anti-angiogenic compound SU5416.
Antonian L; Zhang H; Yang C; Wagner G; Shawver LK; Shet M; Ogilvie B; Madan A; Parkinson A
Drug Metab Dispos; 2000 Dec; 28(12):1505-12. PubMed ID: 11095590
[TBL] [Abstract][Full Text] [Related]
36. Biotransformation of 6-methoxy-3-(3',4',5'-trimethoxy-benzoyl)-1H-indole (BPR0L075), a novel antimicrotubule agent, by mouse, rat, dog, and human liver microsomes.
Yao HT; Wu YS; Chang YW; Hsieh HP; Chen WC; Lan SJ; Chen CT; Chao YS; Chang L; Sun HY; Yeh TK
Drug Metab Dispos; 2007 Jul; 35(7):1042-9. PubMed ID: 17403915
[TBL] [Abstract][Full Text] [Related]
37. Structural elucidation of metabolites of ginkgolic acid in rat liver microsomes by ultra-performance liquid chromatography/electrospray ionization tandem mass spectrometry and hydrogen/deuterium exchange.
Liu ZH; Chen J; Yu LS; Jiang HD; Yao TW; Zeng S
Rapid Commun Mass Spectrom; 2009 Jul; 23(13):1899-906. PubMed ID: 19462408
[TBL] [Abstract][Full Text] [Related]
38. In vitro metabolism study of combretastatin A-4 in rat and human liver microsomes.
Aprile S; Del Grosso E; Tron GC; Grosa G
Drug Metab Dispos; 2007 Dec; 35(12):2252-61. PubMed ID: 17890446
[TBL] [Abstract][Full Text] [Related]
39. Metabolism of 7,8-dihydrobenzo(a)pyrene by rat liver microsomal enzymes and mutagenicity of metabolites.
Chiu PL; Yang SK
Cancer Res; 1986 Oct; 46(10):5084-94. PubMed ID: 3756866
[TBL] [Abstract][Full Text] [Related]
40. 1-(5-Carboxyindol-1-yl)propan-2-ones as inhibitors of human cytosolic phospholipase A2alpha: synthesis and properties of bioisosteric benzimidazole, benzotriazole and indazole analogues.
Bovens S; Kaptur M; Elfringhoff AS; Lehr M
Bioorg Med Chem Lett; 2009 Apr; 19(8):2107-11. PubMed ID: 19327988
[TBL] [Abstract][Full Text] [Related]
[Previous] [Next] [New Search]
