BIOMARKERS

Molecular Biopsy of Human Tumors

- a resource for Precision Medicine *

228 related articles for article (PubMed ID: 16949293)

  • 1. Anti-cancer activities of 5-acyl-6-[2-hydroxy/benzyloxy-3-(amino)-propylamino]-1,3-dialkyl-1H-pyrimidin-2,4-diones.
    Singh P; Paul K
    Bioorg Med Chem; 2006 Dec; 14(24):8622-5. PubMed ID: 16949293
    [TBL] [Abstract][Full Text] [Related]  

  • 2. Novel 6-N-arylcarboxamidopyrazolo[4,3-d]pyrimidin-7-one derivatives as potential anti-cancer agents.
    Devegowda VN; Kim JH; Han KC; Yang EG; Choo H; Pae AN; Nam G; Choi KI
    Bioorg Med Chem Lett; 2010 Mar; 20(5):1630-3. PubMed ID: 20138760
    [TBL] [Abstract][Full Text] [Related]  

  • 3. Syntheses and anti-cancer activities of 2-[1-(indol-3-yl-/pyrimidin-5-yl-/pyridine-2-yl-/quinolin-2-yl)-but-3-enylamino]-2-phenyl-ethanols.
    Singh P; Kaur P; Luxami V; Kaur S; Kumar S
    Bioorg Med Chem; 2007 Mar; 15(6):2386-95. PubMed ID: 17275313
    [TBL] [Abstract][Full Text] [Related]  

  • 4. Synthesis and anti-tumor activities of some new pyridines and pyrazolo[1,5-a]pyrimidines.
    Ahmed OM; Mohamed MA; Ahmed RR; Ahmed SA
    Eur J Med Chem; 2009 Sep; 44(9):3519-23. PubMed ID: 19398146
    [TBL] [Abstract][Full Text] [Related]  

  • 5. One pot synthesis of thiazolodihydropyrimidinones and evaluation of their anticancer activity.
    Holla BS; Rao BS; Sarojini BK; Akberali PM
    Eur J Med Chem; 2004 Sep; 39(9):777-83. PubMed ID: 15337290
    [TBL] [Abstract][Full Text] [Related]  

  • 6. Synthesis of new indeno[1,2-e]pyrimido[4,5-b][1,4]diazepine-5,11-diones as potential antitumor agents.
    Insuasty B; Orozco F; Lizarazo C; Quiroga J; Abonia R; Hursthouse M; Nogueras M; Cobo J
    Bioorg Med Chem; 2008 Sep; 16(18):8492-500. PubMed ID: 18752965
    [TBL] [Abstract][Full Text] [Related]  

  • 7. Synthesis of N-{4-[(2,4-diamino-5-methyl-4,7-dihydro-3H-pyrrolo[2,3-d]pyrimidin-6-yl)thio]benzoyl}-L-glutamic acid and N-{4-[(2-amino-4-oxo-5-methyl-4,7-dihydro-3H-pyrrolo[2,3-d]pyrimidin-6-yl)thio]benzoyl}-L-glutamic acid as dual inhibitors of dihydrofolate reductase and thymidylate synthase and as potential antitumor agents.
    Gangjee A; Lin X; Kisliuk RL; McGuire JJ
    J Med Chem; 2005 Nov; 48(23):7215-22. PubMed ID: 16279780
    [TBL] [Abstract][Full Text] [Related]  

  • 8. Synthesis of 2,8-disubstituted imidazo[1,5-a]pyrimidines with potent antitumor activity.
    Matsumoto H; Ikeda K; Nagata N; Takayanagi H; Mizuno Y; Tanaka M; Sasaki T
    J Med Chem; 1999 May; 42(9):1661-6. PubMed ID: 10229634
    [TBL] [Abstract][Full Text] [Related]  

  • 9. Synthesis and antiproliferative activity of 2,4-disubstituted 6-aryl-7H-pyrrolo[3,2-d]pyrimidin-7-one 5-oxides.
    Pudziuvelyte E; Ríos-Luci C; León LG; Cikotiene I; Padrón JM
    Bioorg Med Chem; 2009 Jul; 17(14):4955-60. PubMed ID: 19527934
    [TBL] [Abstract][Full Text] [Related]  

  • 10. Synthesis and antitumor activity of novel pyrido[2,3-d][1,2,4]triazolo[4,3-a]pyrimidin-5-one derivatives.
    El-Nassan HB
    Eur J Med Chem; 2011 Jun; 46(6):2031-6. PubMed ID: 21429629
    [TBL] [Abstract][Full Text] [Related]  

  • 11. Synthesis and antiviral and cytostatic evaluations of the new C-5 substituted pyrimidine and furo[2,3-d]pyrimidine 4',5'-didehydro-L-ascorbic acid derivatives.
    Gazivoda T; Sokcević M; Kralj M; Suman L; Pavelić K; De Clercq E; Andrei G; Snoeck R; Balzarini J; Mintas M; Raić-Malić S
    J Med Chem; 2007 Aug; 50(17):4105-12. PubMed ID: 17672445
    [TBL] [Abstract][Full Text] [Related]  

  • 12. Induction of intrinsic apoptosis pathway in colon cancer HCT-116 cells by novel 2-substituted-5,6,7,8-tetrahydronaphthalene derivatives.
    Gamal-Eldeen AM; Hamdy NA; Abdel-Aziz HA; El-Hussieny EA; Fakhr IM
    Eur J Med Chem; 2014 Apr; 77():323-33. PubMed ID: 24657569
    [TBL] [Abstract][Full Text] [Related]  

  • 13. Regioselective synthesis and stereochemical structure of anti-tumor active dispiro[3H-indole-3,2'-pyrrolidine-3',3''-piperidine]-2(1H),4''-diones.
    Girgis AS
    Eur J Med Chem; 2009 Mar; 44(3):1257-64. PubMed ID: 18947903
    [TBL] [Abstract][Full Text] [Related]  

  • 14. Synthesis and anti-tumor activities of novel pyrazolo[1,5-a]pyrimidines.
    Li J; Zhao YF; Zhao XL; Yuan XY; Gong P
    Arch Pharm (Weinheim); 2006 Nov; 339(11):593-7. PubMed ID: 17036367
    [TBL] [Abstract][Full Text] [Related]  

  • 15. Synthesis and anti-tumor activities of N'-benzylidene-2-(4-oxothieno[2,3-d]pyrimidin-3(4H)-yl)acetohydrazone derivatives.
    Lou J; Liu Z; Li Y; Zhou M; Zhang Z; Zheng S; Wang R; Li J
    Bioorg Med Chem Lett; 2011 Nov; 21(22):6662-6. PubMed ID: 21986587
    [TBL] [Abstract][Full Text] [Related]  

  • 16. Design, synthesis and anticancer activities of hybrids of indole and barbituric acids--identification of highly promising leads.
    Singh P; Kaur M; Verma P
    Bioorg Med Chem Lett; 2009 Jun; 19(11):3054-8. PubMed ID: 19398334
    [TBL] [Abstract][Full Text] [Related]  

  • 17. Synthesis of novel pyrimidine-2,4-diones and 2-thioxo-pyrimidine-4-ones as potential anticancer and antimicrobial agents.
    Soliman R; Habib NS; Ismail K; Moustafa A; Sarg MT; Fanaki NH
    Boll Chim Farm; 2003 May; 142(4):167-74. PubMed ID: 12918226
    [TBL] [Abstract][Full Text] [Related]  

  • 18. Simplified analogues of immucillin-G retain potent human purine nucleoside phosphorylase inhibitory activity.
    Semeraro T; Lossani A; Botta M; Ghiron C; Alvarez R; Manetti F; Mugnaini C; Valensin S; Focher F; Corelli F
    J Med Chem; 2006 Oct; 49(20):6037-45. PubMed ID: 17004717
    [TBL] [Abstract][Full Text] [Related]  

  • 19. Regioselective synthesis of dispiro[1H-indene-2,3'-pyrrolidine-2',3''-[3H]indole]-1,2''(1''H)-diones of potential anti-tumor properties.
    Girgis AS
    Eur J Med Chem; 2009 Jan; 44(1):91-100. PubMed ID: 18455272
    [TBL] [Abstract][Full Text] [Related]  

  • 20. Discovery of 4-anilino-N-methylthieno[3,2-d]pyrimidines and 4-anilino-N-methylthieno[2,3-d]pyrimidines as potent apoptosis inducers.
    Kemnitzer W; Sirisoma N; May C; Tseng B; Drewe J; Cai SX
    Bioorg Med Chem Lett; 2009 Jul; 19(13):3536-40. PubMed ID: 19464890
    [TBL] [Abstract][Full Text] [Related]  

    [Next]    [New Search]
    of 12.