170 related articles for article (PubMed ID: 17081025)
1. Convergent synthesis of complex diketopiperazines derived from pipecolic acid scaffolds and parallel screening against GPCR targets.
Dandapani S; Lan P; Beeler AB; Beischel S; Abbas A; Roth BL; Porco JA; Panek JS
J Org Chem; 2006 Nov; 71(23):8934-45. PubMed ID: 17081025
[TBL] [Abstract][Full Text] [Related]
2. A step-economical multicomponent synthesis of 3D-shaped aza-diketopiperazines and their drug-like chemical space analysis.
Regenass P; Riché S; Péron F; Rognan D; Hibert M; Girard N; Bonnet D
Org Biomol Chem; 2016 Sep; 14(37):8859-8863. PubMed ID: 27722636
[TBL] [Abstract][Full Text] [Related]
3. Diketopiperazines in peptide and combinatorial chemistry.
Fischer PM
J Pept Sci; 2003 Jan; 9(1):9-35. PubMed ID: 12587880
[TBL] [Abstract][Full Text] [Related]
4. Annulation of primary amines to piperazines and diazaspirocycles utilizing alpha-methyl benzyl resin.
Macleod C; Martinez-Teipel BI; Barker WM; Dolle RE
J Comb Chem; 2006; 8(1):132-40. PubMed ID: 16398564
[TBL] [Abstract][Full Text] [Related]
5. Diastereoselective synthesis of novel aza-diketopiperazines via a domino cyclohydrocarbonylation/addition process.
Regenass P; Margathe JF; Mann A; Suffert J; Hibert M; Girard N; Bonnet D
Chem Commun (Camb); 2014 Sep; 50(68):9657-60. PubMed ID: 25019687
[TBL] [Abstract][Full Text] [Related]
6. Comparative Study of the Synthesis and Structural and Physicochemical Properties of Diketopiperazines vs Aza-diketopiperazines.
Regenass P; Bosc D; Riché S; Gizzi P; Hibert M; Karmazin L; Ganesan A; Bonnet D
J Org Chem; 2017 Mar; 82(6):3239-3244. PubMed ID: 28230990
[TBL] [Abstract][Full Text] [Related]
7. Microwave-assisted solid-phase synthesis of 2,5-diketopiperazines: solvent and resin dependence.
Tullberg M; Luthman K; Grøtli M
J Comb Chem; 2006; 8(6):915-22. PubMed ID: 17096581
[TBL] [Abstract][Full Text] [Related]
8. Synthesis of a small library of diketopiperazines as potential inhibitors of calpain.
Zeng Y; Li Q; Hanzlik RP; Aubé J
Bioorg Med Chem Lett; 2005 Jun; 15(12):3034-8. PubMed ID: 15896956
[TBL] [Abstract][Full Text] [Related]
9. Combinatorial aid for underprivileged scaffolds: solution and solid-phase strategies for a rapid and efficient access to novel aza-diketopiperazines (Aza-DKP).
Bonnet D; Margathe JF; Radford S; Pflimlin E; Riché S; Doman P; Hibert M; Ganesan A
ACS Comb Sci; 2012 May; 14(5):323-34. PubMed ID: 22458603
[TBL] [Abstract][Full Text] [Related]
10. Stereochemical and skeletal diversity employing pipecolate ester scaffolds.
Chen Y; Porco JA; Panek JS
Org Lett; 2007 Apr; 9(8):1529-32. PubMed ID: 17367153
[TBL] [Abstract][Full Text] [Related]
11. Synthesis of functionalized, unsymmetrical 1,3,4,6-tetrasubstituted 2,5-diketopiperazines.
Tullberg M; Grøtli M; Luthman K
J Org Chem; 2007 Jan; 72(1):195-9. PubMed ID: 17194099
[TBL] [Abstract][Full Text] [Related]
12. Short and novel stereospecific synthesis of trisubstituted 2,5-diketopiperazines.
Sollis SL
J Org Chem; 2005 Jun; 70(12):4735-40. PubMed ID: 15932312
[TBL] [Abstract][Full Text] [Related]
13. Synthesis, molecular modeling and biological evaluation of aza-proline and aza-pipecolic derivatives as FKBP12 ligands and their in vivo neuroprotective effects.
Wilkinson DE; Thomas BE; Limburg DC; Holmes A; Sauer H; Ross DT; Soni R; Chen Y; Guo H; Howorth P; Valentine H; Spicer D; Fuller M; Steiner JP; Hamilton GS; Wu YQ
Bioorg Med Chem; 2003 Nov; 11(22):4815-25. PubMed ID: 14556798
[TBL] [Abstract][Full Text] [Related]
14. Recycling the versatile Pipecolic linker.
Zajdel P; Masurier N; Sanchez P; Pawlowski M; Kreiter A; Nomezine G; Enjalbal C; Amblard M; Martinez J; Subra G
J Comb Chem; 2010 Sep; 12(5):747-53. PubMed ID: 20715810
[TBL] [Abstract][Full Text] [Related]
15. [Development of Novel Functional Molecules Based on the Molecular Structure Characteristics of Diketopiperazines].
Nakao M
Yakugaku Zasshi; 2017; 137(12):1505-1516. PubMed ID: 29199259
[TBL] [Abstract][Full Text] [Related]
16. A new class of highly cytotoxic diketopiperazines.
Boger DL; Fink BE; Hedrick MP
Bioorg Med Chem Lett; 2000 May; 10(10):1019-20. PubMed ID: 10843206
[TBL] [Abstract][Full Text] [Related]
17. The discovery of potent antagonists of NPBWR1 (GPR7).
Anthony Romero F; Hastings NB; Moningka R; Guo Z; Wang M; Di Salvo J; Lei Y; Trusca D; Deng Q; Tong V; Terebetski JL; Ball RG; Ujjainwalla F
Bioorg Med Chem Lett; 2012 Jan; 22(2):1014-8. PubMed ID: 22197390
[TBL] [Abstract][Full Text] [Related]
18. A new highly versatile handle for chemistry on a solid support: the pipecolic linker.
Zajdel P; Nomezine G; Masurier N; Amblard M; Pawłowski M; Martinez J; Subra G
Chemistry; 2010 Jul; 16(25):7547-53. PubMed ID: 20468039
[TBL] [Abstract][Full Text] [Related]
19. Synthesis of spirohydantoins and spiro-2,5-diketopiperazines via resin-bound cyclic alpha,alpha-disubstituted alpha-amino esters.
Kuster GJ; van Berkom LW; Kalmoua M; van Loevezijn A; Sliedregt LA; van Steen BJ; Kruse CG; Rutjes FP; Scheeren HW
J Comb Chem; 2006; 8(1):85-94. PubMed ID: 16398558
[TBL] [Abstract][Full Text] [Related]
20. Efficient construction of diketopiperazine macroarrays through a cyclative-cleavage strategy and their evaluation as luminescence inhibitors in the bacterial symbiont Vibrio fischeri.
Campbell J; Blackwell HE
J Comb Chem; 2009; 11(6):1094-9. PubMed ID: 19831384
[TBL] [Abstract][Full Text] [Related]
[Next] [New Search]
